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产品名称: BI 2536化合物BI 25364-[[(7R)-8-环戊基-7-乙基-5,6,7,8-四氢-5-甲基-6-氧代-2-喋啶基]氨基]-3-甲氧基-N-(1-甲基-4-哌啶基)苯甲酰胺
产品简介:bi2536 is an effective plk1 inhibitor (ic50: 0.83 nm). it has 4- and 11-fold greater selectivity than plk2 and plk3...产品型号:T6173 原产地:中国大陆价格: ¥0.0
产品名称: HPK1-IN-25;化合物 HPK1-IN-25HPK1-IN-25
产品简介:hpk1-in-25 (example 94), an inhibitor of hematopoietic progenitor kinase 1 (hpk1), demonstrates enzymatic activity with an ic50 value of 129 nm, indicating its ..产品型号:T61733 原产地:中国大陆价格: ¥0.0
产品名称: MI-1;化合物 MI-1MI-1
产品简介:mi-1 inhibits menin-mll interaction with an ic 50 of 1.9 μm [1]...产品型号:T61735 原产地:中国大陆价格: ¥0.0
产品名称: CB1/2 agonist 3;化合物 CB1/2 agonist 3CB1/2 agonist 3
产品简介:cb1/2 agonist 3 (compound 52), a potent non-selective cannabinoid ligand, is a competitive agonist for the cb1/cb2 receptors. it exhibits cb1/cb2 agonistic acti..产品型号:T61736 原产地:中国大陆价格: ¥0.0
产品名称: Dyrk1A-IN-5;化合物 Dyrk1A-IN-5Dyrk1A-IN-5
产品简介:dyrk1a-in-5 (compound 5j) is a highly potent and selective inhibitor of dyrk1a, exhibiting an ic50 of 6 nm. it dose-dependently diminishes the phosphorylation o..产品型号:T61739 原产地:中国大陆价格: ¥0.0
产品名称: Enpp-1-IN-12;化合物 Enpp-1-IN-12Enpp-1-IN-12
产品简介:enpp-1-in-12 (compound 43), an orally active and potent inhibitor of ecto-nucleotide pyrophosphatase/phosphodiesterases 1 (enpp1) with a k i of 41 nm, exhibits ..产品型号:T61514 原产地:中国大陆价格: ¥0.0
产品名称: 5-HT7 receptor ligand 1;化合物 5-HT7 receptor ligand 15-HT7 receptor ligand 1
产品简介:5-ht7 receptor ligand 1 (compound 5c) is a potent ligand for the 5-ht7 receptor, with a k i value of 8 nm. the compound demonstrates non-hepatotoxic properties ..产品型号:T61515 原产地:中国大陆价格: ¥0.0
产品名称: Nrf2/HO-1 activator 2;化合物 Nrf2/HO-1 activator 2Nrf2/HO-1 activator 2
产品简介:nrf2/ho-1 activator 2 (compound 13m), a difluoro-substituted derivative, is a highly potent activator of nrf2/ho-1. it exhibits substantial neuroprotective and ..产品型号:T61522 原产地:中国大陆价格: ¥0.0
产品名称: Tubulin/HDAC-IN-1;化合物 Tubulin/HDAC-IN-1Tubulin/HDAC-IN-1
产品简介:tubulin/hdac-in-1 is a compound that functions as a dual inhibitor for tubulin and hdac-in-1. it achieves this by interacting with tubulin through ch/π interact..产品型号:T61524 原产地:中国大陆价格: ¥0.0
产品名称: NFATc1-IN-1;化合物NFATc1-IN-1NFATc1-IN-1
产品简介:nfatc1-in-1 (also known as compound a04) is a highly effective inhibitor of osteoclast formation induced by rankl, with an ic50 of 1.57 μm. it exerts its anti-o..产品型号:T61531 原产地:中国大陆价格: ¥0.0
产品名称: A1AR antagonist 4;化合物 A1AR antagonist 4A1AR antagonist 4
产品简介:a1ar antagonist 4 (compound 22) is a highly developed chemical compound that acts as a potent and selective antagonist of the a1 adenosine receptor (a1ar). it p..产品型号:T61536 原产地:中国大陆价格: ¥0.0
产品名称: ASIC-IN-1;化合物 ASIC-IN-1ASIC-IN-1
产品简介:asic-in-1 is a potent inhibitor of acid-sensing ion channels, demonstrating an ic 50 value of less than 10 μm. it effectively reduces pain intensity in a dose-d..产品型号:T61537 原产地:中国大陆价格: ¥0.0
产品名称: CLK1/4-IN-1;化合物 CLK1/4-IN-1CLK1/4-IN-1
产品简介:clk1/4-in-1 (compound 31) is a highly potent and selective inhibitor of clk1 and clk4, with ic50 values of 9.7 nm and 6.6 nm, respectively. it effectively inhib..产品型号:T61543 原产地:中国大陆价格: ¥0.0
产品名称: CSF1R-IN-13;化合物 CSF1R-IN-13CSF1R-IN-13
产品简介:csf1r-in-13 is a powerful csf1r inhibitor with potential applications in researching cancer diseases [1]. csf1r, also known as colony stimulating factor 1 recep..产品型号:T61554 原产地:中国大陆价格: ¥0.0
产品名称: Ruxolitinib (S enantiomer);环丙基[4-[3-(1H-咪唑-5-基)丙氧基]苯S-Ruxolitinib|||Ruxolitinib S enantiomer|||INCB0
产品简介:ruxolitinib s enantiomer (incb18424) is the s-enantiomer of ruxolitinib. ruxolitinib is the first potent, selective jak1/2 inhibitor...产品型号:T6156 原产地:中国大陆价格: ¥0.0
产品名称: CB1R Allosteric modulator 3;CB1R变构调节剂3CB1R Allosteric modulator 3
产品简介:cb1r allosteric modulator 3 is a potent cb1r modulator.cb1r allosteric modulator 3 inhibits camp and β-arrestin, and can be used for the study of obesity and ni..产品型号:T61562 原产地:中国大陆价格: ¥0.0
产品名称: HSV-1/HSV-2-IN-2;化合物 HSV-1/HSV-2-IN-2HSV-1/HSV-2-IN-2
产品简介:hsv-1/hsv-2-in-2 is a compound that acts as an inhibitor of hsv-1, hsv-2, and vv, demonstrating antiviral activity with ec50 values of 6.8, 8.9, and 8.9 μm, res..产品型号:T61563 原产地:中国大陆价格: ¥0.0
产品名称: Liproxstatin-1 hydrochloride;化合物 Liproxstatin-1 hydrochlorideLiproxstatin-1 hydrochloride
产品简介:liproxstatin-1 hydrochloride is a high-potency ferroptosis inhibitor capable of effectively preventing ferroptotic cell death, with an ic50 value of 22 nm [1]...产品型号:T61567 原产地:中国大陆价格: ¥0.0
产品名称: Vanin-1-IN-3;化合物 Vanin-1-IN-3Vanin-1-IN-3
产品简介:vanin-1-in-3 (omp-7) is a vanin-1 inhibitor with an ic 50 of 0.038 μm [1]...产品型号:T61568 原产地:中国大陆价格: ¥0.0
产品名称: Mt KARI-IN-1;化合物 Mt KARI-IN-1Mt KARI-IN-1
产品简介:mt kari-in-1 is a lead compound that demonstrates strong inhibitory activity towards mycobacterium tuberculosis ketol-acid reductoisomerase (mtb kari), with a k..产品型号:T61569 原产地:中国大陆价格: ¥0.0