联系我们
产品目录
产品展示/Products
产品名称: BorussertibBorussertib,Inhibitor,PKB,Akt,Protein kinase B,inhibit
产品简介:borussertib is a covalent-allosteric and first-in-class inhibitor of protein kinase akt(ic50 of 0.8 nm and a ki of 2.2 nm for aktwt)..产品型号:T8427 原产地:中国大陆价格: ¥0.0
产品名称: WYE-687mTOR,Mammalian target of Rapamycin,WYE-687,Phosphoinositide 3-kinase,WYE687,PI3K,WYE 687,inhi
产品简介:wye-687 is an atp-competitive and selective inhibitor of mtor with ic50 of 7 nm; blocks mtorc1/ps6k(t389) and mtorc2/p-akt(s473) but no effect observed on p-akt..产品型号:T6732 原产地:中国大陆价格: ¥0.0
产品名称: DASA-58DASA58,inhibit,Inhibitor,DASA 58,DASA-58,glycolysis,TXNIP,cancer metabolism,Pyruvate Kinase,p
产品简介:dasa-58 is a specific and potent pyruvate kinase m2 (pkm2) activator...产品型号:T6816 原产地:中国大陆价格: ¥0.0
产品名称: LY3405105anticancer,Cyclin dependent kinase,CDK,MCF7,SNU-16,Cyclin-dependent kinase,LY 3405105,LY340
产品简介:ly3405105 is a novel cdk7 inhibitors...产品型号:T9078 原产地:中国大陆价格: ¥0.0
产品名称: TH-257LIM Kinase (LIMK),LIMKs,Inhibitor,TH-257,inhibit,TH257
产品简介:th 257 is a potent and selective allosteric limk 1/2 inhibitor(limk1 and limk2, ic50 of 84 nm and 39 nm)...产品型号:T7128 原产地:中国大陆价格: ¥0.0
产品名称: RSVA405RSVA-405,Autophagy,Inhibitor,anti-inflammatory,STAT,AMP-activated protein kinase,disease,Kina
产品简介:rsva 405 is an ampk activator (ec50 = 1 μm), and is stat3 inhibitor..产品型号:T8476 原产地:中国大陆价格: ¥0.0
产品名称: R547Glycogen synthase kinase 3,kinase,multiple,tumor,cyclin-dependent,R547,Apoptosis,Cyclin dependen
产品简介:r547 is a potent atp-competitive inhibitor of cdk1/2/4 with ki of 2 nm/3 nm/1 nm. it is less potent to cdk7 and gsk3α/β, while inactive to other kinases. phase ..产品型号:T6312 原产地:中国大陆价格: ¥0.0
产品名称: ChelerythrineBcl-2 Family,Apoptosis,Protein kinase C,PKC,Inhibitor,Chelerythrine,inhibit,Autophagy
产品简介:1. chelerythrine may have antimanic effect . 2. chelerythrine can inhibit telomerase activity. 3. chelerythrine is a well-known protein kinase c inhibitor . 4. ..产品型号:T6S0052 原产地:中国大陆价格: ¥0.0
产品名称: CHR-6494 TFACHR-6494,inhibit,apoptosis,Haspin Kinase,NRAS mutant melanoma cells,CHR 6494,mitotic cat
产品简介:chr-6494 tfa is a potent haspin inhibitor, with an?ic50?of 2 nm. it inhibits histone h3t3 phosphorylation. chr-6494 tfa induces the?apoptosis?of cancer cells, i..产品型号:T9521 原产地:中国大陆价格: ¥0.0
产品名称: (E/Z)-GSK-3β inhibitor 1Glycogen synthase kinase 3,Inhibitor,Glycogen synthase kinase-3,inhibit,(E/Z
产品简介:gsk-3β inhibitor 1 is a glycogen synthase kinase 3β (gsk-3β) inhibitor and demonstrates high antidiabetic efficacy...产品型号:T9178 原产地:中国大陆价格: ¥0.0
产品名称: EML4-ALK kinase inhibitor 1
产品简介:eml4-alk kinase inhibitor 1 is a potent oral active inhibitor of echinoderm microtubule-associated protein-like 4-anaplastic lymphoma kinase (eml4-alk), with an..产品型号:T11184 原产地:中国大陆价格: ¥0.0
产品名称: GDC-0623Mitogen-activated protein kinase kinase,Apoptosis,inhibit,MEK,Inhibitor,MAP2K,MAPKK,MEK inhi
产品简介:gdc-0623 is a potent and atp-uncompetitive mek1 inhibitor with ki of 0.13 nm. phase 1...产品型号:T6843 原产地:中国大陆价格: ¥0.0
产品名称: GSK547Inhibitor,RIP kinase,inhibit,GSK-547,GSK547,Receptor-interacting protein kinases,RIPK,GSK 547
产品简介:gsk547 is a highly selective and potent inhibitor of rip1 kinase,inhibits macrophage-mediated adaptive immune tolerance in pancreatic cancer...产品型号:T7397 原产地:中国大陆价格: ¥0.0
产品名称: HG-10-102-01Parkinson’s disease,Leucine-rich repeat kinase 2,inhibit,Ser910,BBB,HG 10 102 01,Radiosy
产品简介:hg-10-102-01 is an inhibitor of leucine-rich repeat kinase 2 (lrrk2, ic50 of 20.3 nm)...产品型号:T7196 原产地:中国大陆价格: ¥0.0
产品名称: dCeMM3?degradation,dCeMM 3,dCeMM3?,Inhibitor,inhibit,CDK,CDK12,Cyclin dependent kinase,glue degrader
产品简介:dcemm3 is a glue degrader. dcemm3 prompts an interaction of cdk12-cyclin k with a crl4b ligase complex, result in inducing ubiquitination and degradation of cyc..产品型号:T9758 原产地:中国大陆价格: ¥0.0
产品名称: KahweolInhibitor,inhibit,Kahweol,AMPK,Apoptosis,AMP-activated protein kinase
产品简介:kahweol has anticarcinogenic, anti-angiogenic,and anti-inflammatory activities, it can block the lps-induced activation of nf-kappab by preventing ikappab degra..产品型号:TN1828 原产地:中国大陆价格: ¥0.0
产品名称: K145 hydrochlorideK-145,K 145,ERK,K145 hydrochloride,K145,Sphingosine kinase,anti-proliferative,SphK
产品简介:k145 hydrochloride is a selective sphk2 inhibitor with substrate competitiveness and oral activity, with ic50 of 4.3 ?m and ki of 6.4 ?m. k145 hydrochloride can..产品型号:TQ0138 原产地:中国大陆价格: ¥0.0
产品名称: AMG 900AMG 900,Inhibitor,Aurora Kinase,inhibit
产品简介:amg 900 is a potent and highly selective pan-aurora kinases inhibitor for aurora a/b/c with ic50 of 5 nm/4 nm /1 nm. it is >10-fold selective for aurora kinases..产品型号:T6380 原产地:中国大陆价格: ¥0.0
产品名称: ZimlovisertibInterleukin-1 receptor associated kinase,inhibit,Zimlovisertib,Inhibitor,IL-1R associat
产品简介:pf06650833 is an effective, selective and orally active inhibitor of interleukin-1 receptor-associated kinase 4 (irak4) (ic50s: 0.2 and 2.4 nm in the cell and p..产品型号:TQ0167 原产地:中国大陆价格: ¥0.0
产品名称: AZD3264inhibit,I kappa B kinase,IκB kinase,AZD 3264,AZD-3264,AZD3264,IKK,Inhibitor
产品简介:azd3264 is a new type ikk2 inhibitor...产品型号:T6771 原产地:中国大陆价格: ¥0.0