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产品名称: ITK degrader 1;化合物 ITK degrader 1ITK degrader 1
产品简介:itk degrader 1, a highly selective interleukin-2-inducible t-cell kinase (itk; dc50=3.6 nm in vivo in mice) degrader, induces rapid and prolonged degradation of..产品型号:T74843 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC pan-IAP degrader-1;化合物 PROTAC pan-IAP degrader-1PROTAC pan-IAP degrader-1
产品简介:protac pan-iap degrader-1 (compound 9) is a pan- iap degrader protac . protac pan-iap degrader-1 degrades xiap , ciap1 and ciap2 with dc 50 s of 0.7, 2.4, and 6..产品型号:T74847 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC CDK9 degrader-5;化合物 PROTAC CDK9 degrader-5PROTAC CDK9 degrader-5
产品简介:protac cdk9 degrader-5 is a selective protac that mediates degradation of cdk9 via the proteasome pathway. it efficiently degrades the cdk9 42 and cdk9 55 isofo..产品型号:T74851 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC CDK9 degrader-6;化合物 PROTAC CDK9 degrader-6PROTAC CDK9 degrader-6
产品简介:protac cdk9 degrader-6 is a specific protac targeting cdk9 that mediates its degradation through the proteasome pathway. this compound effectively degrades cdk9..产品型号:T74852 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC CDK9 degrader-7;化合物 PROTAC CDK9 degrader-7PROTAC CDK9 degrader-7
产品简介:protac cdk9 degrader-7 is a proteolysis-targeting chimera (protac) specifically designed to target and mediate the degradation of cyclin-dependent kinase 9 (cdk..产品型号:T74853 原产地:中国大陆价格: ¥0.0
产品名称: ER degrader 4;化合物 ER degrader 4ER degrader 4
产品简介:er degrader 4, a selective and orally active compound, effectively degrades estrogen receptors and exhibits anti-tumor activity [1]...产品型号:T74856 原产地:中国大陆价格: ¥0.0
产品名称: ER degrader 5;化合物 ER degrader 5ER degrader 5
产品简介:er degrader 5 is a potent compound that degrades the estrogen receptor (er), exhibits anti-proliferation activity, and has potential applications in breast canc..产品型号:T74857 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC STING Degrader-1;化合物 PROTAC STING Degrader-1PROTAC STING Degrader-1
产品简介:protac sting degrader-1 (compound sp23) is a sting-targeted protac degrader exhibiting a dc50 of 3.2 μm and demonstrates anti-inflammatory activity [1]...产品型号:T74896 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC FLT3/CDK9 degrader-1;化合物 PROTAC FLT3/CDK9 degrader-1PROTAC FLT3/CDK9 degrader-1
产品简介:protac flt3/cdk9 degrader-1, a potent dual degrader of flt3 and cdk9, effectively induces apoptosis and targets protein degradation of flt3 and cdk9. this compo..产品型号:T74707 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC PTPN2 degrader-1;化合物 PROTAC PTPN2 degrader-1PROTAC PTPN2 degrader-1
产品简介:protac ptpn2 degrader-1 (compound example 77) is a potent entity capable of degrading ptpn2, showing promise for research applications in cancer or metabolic di..产品型号:T74732 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC AR-NTD degrader 1;化合物 PROTAC AR-NTD degrader 1PROTAC AR-NTD degrader 1
产品简介:protac ar-ntd antagonist 1 (compound 18) is a small molecule belonging to the protein-targeting chimeras (protacs) that selectively targets the n-terminal domai..产品型号:T78811 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC CDK9 degrader-8;化合物 PROTAC CDK9 degrader-8PROTAC CDK9 degrader-8
产品简介:protac cdk9 degrader-8 (compound 21) is a potent degrader of cdk9 with an ic50 of 0.01 μm, utilized in cancer research [1]...产品型号:T78928 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC BTK Degrader-6;化合物 PROTAC BTK Degrader-6PROTAC BTK Degrader-6
产品简介:protac btk degrader-6 (compound 15), with a dc50 of 3.18 nm, exhibits anti-inflammatory properties by inhibiting nf-κb activation and suppressing the expression..产品型号:T78782 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC BRD3/BRD4-L degrader-2;化合物 PROTAC BRD3/BRD4-L degrader-2PROTAC BRD3/BRD4-L degrader-2
产品简介:protac brd3/brd4-l degrader-2, a protac molecule, selectively degrades cellular brd3 and brd4-l with k i values of 16.91 and 2.8 nm, respectively, and exhibits ..产品型号:T78956 原产地:中国大陆价格: ¥0.0
产品名称: STAT3 degrader-2;化合物 STAT3 degrader-2STAT3 degrader-2
产品简介:stat3 degrader-2 is a protac-based compound that effectively reduces the total stat3 protein levels, and is utilized in the research of cancer and various disea..产品型号:T78983 原产地:中国大陆价格: ¥0.0
产品名称: ER degrader 6;化合物 ER degrader 6ER degrader 6
产品简介:er degrader 6 (compound 35s) is a potent selective estrogen receptor modulator (serm) with the capacity to degrade estrogen receptor (er)α. it disrupts the micr..产品型号:T79382 原产地:中国大陆价格: ¥0.0
产品名称: ER degrader 7;化合物 ER degrader 7ER degrader 7
产品简介:er degrader 7 (compound 35t) is a selective degrader of both erα and erβ, and possesses activity as a tubulin polymerization inhibitor. it exhibits potent cell ..产品型号:T79383 原产地:中国大陆价格: ¥0.0
产品名称: GSPT1 degrader-1;化合物 GSPT1 degrader-1GSPT1 degrader-1
产品简介:gspt1 degrader-1 (compound 9q) effectively facilitates the degradation of g1 to s phase transition 1 (gspt1) through the ubiquitin-proteasome system and induces..产品型号:T79474 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC TG2 degrader-1;化合物 PROTAC TG2 degrader-1PROTAC TG2 degrader-1
产品简介:protac tg2 degrader-1 (compound 11) is a vhl-based protac that targets tissue transglutaminase (tg2) and exhibits a binding affinity with a k d of 68.9 μm. this..产品型号:T79505 原产地:中国大陆价格: ¥0.0
产品名称: NAMPT degrader-3;化合物 NAMPT degrader-3NAMPT degrader-3
产品简介:nampt degrader-3 (compound c5) is a nampt degrader that functions through a vhl- and proteasome-dependent mechanism. it exhibits cytotoxic properties and inhibi..产品型号:T79437 原产地:中国大陆价格: ¥0.0