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产品名称: AMG 517AMG 517,Inhibitor,inhibit,Transient receptor potential channels,TRP Channel
产品简介:amg 517 is an effective and specific trpv1 antagonist, antagonizes proton (ic50: 0.76 nm), capsaicin (ic50: 0.62 nm), and heat activation (ic50: 1.3 nm) of trpv..产品型号:T6379 原产地:中国大陆价格: ¥0.0
产品名称: CNT2 inhibitor-1CNT-2 inhibitor-1,CNT2 inhibitor 1,CNT2 inhibitor1
产品简介:cnt2 inhibitor-1 is a potent inhibitor of concentrative nucleoside transporter 2 (cnt2; ic50: 640 nm for hcnt2)...产品型号:T10853 原产地:中国大陆价格: ¥0.0
产品名称: Cariprazine hydrochlorideDopamine Receptor,Cariprazine,5-hydroxytryptamine Receptor,RGH188,Inhibitor
产品简介:cariprazine hcl is an antipsychotic drug, is a d3 and d2 receptor partial agonist((ki of 0.085 nm and 0.49 nm, respectively)..产品型号:T8382 原产地:中国大陆价格: ¥0.0
产品名称: GSK-3β inhibitor 2
产品简介:gsk-3β inhibitor 2 is a bbb-crossing and selective inhibitor of gsk-3β (ic50 = 1.1 nm). gsk-3β inhibitor 2 can be used in studies about alzheimer´s diseas..产品型号:T11471 原产地:中国大陆价格: ¥0.0
产品名称: RetapamulinRetapamulin,Bacterial,SB 275833,inhibit,SB275833,Inhibitor,Antibiotic
产品简介:retapamulin, a pleuromutilin antibacterial, binds to both e. coli and s. aureus ribosomes with similar potencies (kd: 3 nm)...产品型号:T6638 原产地:中国大陆价格: ¥0.0
产品名称: OlomoucineOlomoucine,Inhibitor,cyclindependent kinases,cdc2,purines,cell cycle,non-small cell lung c
产品简介:olomoucine is an atp competitive inhibitor of cdk2/cyclin a, cdc2/cyclinb, cdk2/cycline, cdk5/p35, and erk1/p44 map kinase with ic50s of 7, 7, 7, 3 and 25 ?m, r..产品型号:T21588 原产地:中国大陆价格: ¥0.0
产品名称: DacinostatLAQ-824,Dacinostat,Histone deacetylases,inhibit,Autophagy,HDAC,Inhibitor,LAQ 824
产品简介:laq824 (dacinostat) is a novel hdac inhibitor with ic50 of 32 nm and is an activator of the p21 promoter...产品型号:T2454 原产地:中国大陆价格: ¥0.0
产品名称: NBI-31772inhibit,IGF-responsive diseases,IGF-1R,IGFBP,NBI-31772,Inhibitor
产品简介:nbi-31772 is the potent inhibitor of insulin-like growth factor-1 binding protein (igfbp, ki = 47 nm). nbi-31772 can be used in research on igf-responsive disea..产品型号:T8906 原产地:中国大陆价格: ¥0.0
产品名称: N-(Hydroxymethyl)nicotinamideBacterial,Inhibitor,antimicrobic,N(Hydroxymethyl)nicotinamide,N (Hydrox
产品简介:nicoform is an antimicrobial agent...产品型号:T7869 原产地:中国大陆价格: ¥0.0
产品名称: ASK1-IN-1CNS,inhibit,p38 MAPK,ASK1,ASK-1-IN-1,ASK1 IN 1,ASK1IN1,MAPK,Inhibitor,brain,penetrant
产品简介:ask1-in-1 is an inhibitor of apoptosis signal-regulating kinase 1 which is a key mediator in the apoptotic and inflammatory cellular stress response with an ic5..产品型号:T9697 原产地:中国大陆价格: ¥0.0
产品名称: TretazicarTretazicar,NQO1,DNA Alkylator/Crosslinker,rat,bifunctional,Inhibitor,inhibit,agent,cross-l
产品简介:cb1954(tretazicar), an anticancer prodrug, is activated by nad(p)h quinone oxidoreductase 2. it is converted in the presence of the enzyme nqo2 and co-substrate..产品型号:T6798 原产地:中国大陆价格: ¥0.0
产品名称: Scutellarein tetramethyl etherBacterial,Inhibitor,inhibit,Scutellarein tetramethyl ether
产品简介:scutellarein tetramethyl ether is extracted from siam weeds and exhibits anti-inflammatory activity through nf-κb pathway...产品型号:TN1271 原产地:中国大陆价格: ¥0.0
产品名称: BAY-474BAY-474,BAY 474,BAY474,epigenetics,probe,inhibit,Inhibitor,c-Met,SGC,c-Met/HGFR
产品简介:bay-474 is an inhibitor of tyrosine-protein kinase c-met. it acts as an epigenetics probe..产品型号:T7900 原产地:中国大陆价格: ¥0.0
产品名称: SirReal2Sirtuin,Inhibitor,inhibit,SirReal2,SirReal 2,SirReal-2
产品简介:sirreal2 is a potent and selective sirt2 inhibitor with ic50 of 140 nm...产品型号:T6984 原产地:中国大陆价格: ¥0.0
产品名称: Zoledronic Acidactivity,anti-cancer,Inhibitor,bisphosphonate,inhibit,anti-resorptive,CGP-42446,CGP42
产品简介:zoledronate is a bisphosphonate. zometa is used to prevent skeletal fractures in patients with cancers such as multiple myeloma and prostate cancer. it can also..产品型号:T6739 原产地:中国大陆价格: ¥0.0
产品名称: BMP signaling agonist sb4Inhibitor,SMAD,bmp,cell,inhibit,BMP signaling agonist sb4,BRE-luc,BMP signa
产品简介:sb 4 is an agonist of benzoxazole bone morphogenetic protein (bmp) signaling (ec50 :74 nm)..产品型号:T7799 原产地:中国大陆价格: ¥0.0
产品名称: Linderene acetateinhibit,Linderene acetate,Linderene,POP,Prolyl Endopeptidase (PREP),Inhibitor,proly
产品简介:linderene acetate is a competitive inhibitor against prolyl endopeptidase...产品型号:TN4442 原产地:中国大陆价格: ¥0.0
产品名称: Boc-C14-COOHADC Linkers,Antibody-drug conjugates linkers,Inhibitor,PROTAC Linkers,inhibit,Boc-C-14-C
产品简介:boc-c14-cooh is a alkyl-chain-based protac linker. boc-c14-cooh is a non-cleavable adc linker used in the synthesis of antibody-drug conjugates (adcs)...产品型号:T9781 原产地:中国大陆价格: ¥0.0
产品名称: BTSfibers,muscle,Myosin,subfragment,inhibit,BTS,Inhibitor,skeletal,Ca2+,actin,ATPase
产品简介:bts is a potent inhibitor of ca2+-stimulated myosin s1 atpase (ic50 : 5 μm) ...产品型号:T7144 原产地:中国大陆价格: ¥0.0
产品名称: Demethoxydeacetoxypseudolaric acid Binhibit,Demethoxydeacetoxypseudolaric acid B,Inhibitor,Deacetyld
产品简介:demethoxydeacetoxypseudolaric acid b´s the metabolic reaction of tda in vivo is mainly occurred in blood and contributes to be the hydrolysis of plasma es..产品型号:TN3820 原产地:中国大陆价格: ¥0.0