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产品名称: AMG-1694;化合物AMG-1694AMG-1694
产品简介:amg-1694, a potent disruptor of the glucokinase–glucokinase regulatory protein (gk-gkrp) complex, operates by promoting the dissociation of this complex, thereb..产品型号:T14212 原产地:中国大陆价格: ¥0.0
产品名称: Tapotoclax;化合物 T14213AMG-176;AMG-176
产品简介:amg-176 is a mcl-1 inhibitor (ki: 0.13 nm)...产品型号:T14213 原产地:中国大陆价格: ¥0.0
产品名称: AMG 511;化合物AMG 511AMG 511
产品简介:amg 511 is a potent and orally available pan inhibitor of class i pi3ks(kis of 4 nm, 6 nm, 2 nm and 1 nm for pi3kα, β, δ and γ, respectively). it exhibits anti-..产品型号:T14214 原产地:中国大陆价格: ¥0.0
产品名称: AMG 837 sodium salt;化合物 T14215AMG 837 sodium salt
产品简介:amg 837 sodium salt is a potent gpr40 agonist(ec50=13 nm) with a superior pharmacokinetic profile and robust glucose-dependent stimulation of insulin secretion ..产品型号:T14215 原产地:中国大陆价格: ¥0.0
产品名称: AMG 837;化合物 T14216AMG 837
产品简介:amg 837 is a partial gpr40 agonist with an ec50 value of 13 nm, showcasing 85% of the maximal activity displayed by dha in standard assay conditions, indicating..产品型号:T14216 原产地:中国大陆价格: ¥0.0
产品名称: AMG 579;化合物AMG 579AMG-579;AMG-579
产品简介:amg 579 is an efficacious and selective inhibitor of pde10a (ic50 = 0.1 nm)...产品型号:T14217 原产地:中国大陆价格: ¥0.0
产品名称: Azelaprag;化合物AzelapragAMG 986;AMG 986
产品简介:azelaprag (amg 986) is an effective small-molecule apelin receptor agonist. azelaprag can be used to treat neurological diseases and cardiovascular diseases...产品型号:T14390 原产地:中国大陆价格: ¥0.0
产品名称: Vidupiprant;化合物VidupiprantAMG 853;AMG 853
产品简介:vidupiprant (amg 853) is an effective dual antagonist of crth2 and prostanoid d receptor with ic50s of 8 nm and 35 nm in human plasma. vidupiprant can be used i..产品型号:T17232 原产地:中国大陆价格: ¥0.0
产品名称: c-Kit-IN-5-1;化合物AMG-253-(2-Aminoquinazolin-6-yl)-4-methyl-1-(4-(oxazol-2-yl)phenyl)pyridin-2(1H)-one
产品简介:c-kit-in-5-1 (amg-25) is a novel selective and potent c-kit inhibitor...产品型号:T22256 原产地:中国大陆价格: ¥0.0
产品名称: (S)-AMG-510;化合物(S)-AMG-510AMG-510 racemate;AMG-510 racemate
产品简介:(s)-amg-510 是 amg-510 的 s型化合物,是 kras g12c 的强效共价抑制剂,具有潜在的抗肿瘤活性。..产品型号:T22258 原产地:中国大陆价格: ¥0.0
产品名称: AMG-Tie2-1;4-甲基-3-[[3-[2-(甲基氨基)-4-嘧啶基]-2-吡啶基]氧基]-N-[3-(三氟甲基)苯基]苯甲酰胺AMG-Tie2;AMG-Tie2|||4-甲基-3-[[3-[2
产品简介:amg-tie2-1 is a dual inhibitor of vegf receptor 2 (vegfr2) and tunica interna endothelial cell kinase 2 (tie2)...产品型号:T22259 原产地:中国大陆价格: ¥0.0
产品名称: Cinacalcet hydrochloride;盐酸西那卡塞AMG-073 HCl|||Cinacalcet HCl|||AMG-073 hydrochloride|||Cinacalcet;AMG
产品简介:cinacalcet hydrochloride (amg-073 hydrochloride) is a naphthalene derivative and calcimimetic agent that increases the sensitivity of parathyroid gland calcium-..产品型号:T2406 原产地:中国大陆价格: ¥0.0
产品名称: AMG131;化合物INT-131INT-131|||AMG-131|||CHS 131;INT-131|||AMG-131|||CHS 131
产品简介:amg131 (chs 131) , is a novel, non-thiazolidinedione (tzd), selective peroxisome proliferator-activated receptor (ppar)gamma modulator, which can be used for th..产品型号:T8780 原产地:中国大陆价格: ¥0.0
产品名称: Kira8 Hydrochloride;化合物 T11762AMG-18 Hydrochloride;AMG-18 Hydrochloride
产品简介:kira8 hydrochloride is a mono-selective ire1α inhibitor that allosterically attenuates ire1α rnase activity with an ic50 of 5.9 nm...产品型号:T11762 原产地:中国大陆价格: ¥0.0
产品名称: Kira8;化合物Kira8AMG-18;AMG-18
产品简介:kira8 (amg-18) is a mono-selective ire1α inhibitor that allosterically attenuates ire1α rnase activity (ic50: 5.9 nm)...产品型号:T11762L 原产地:中国大陆价格: ¥0.0
产品名称: Raleukin;阿那白滞素AMG-719|||Anakinra;AMG-719|||阿那白滞素|||Anakinra
产品简介:anakinra (raleukin) is an antagonist of recombinant, nonglycosylated human il-1r. it is the first biological agent to block the pro-inflammatory effects...产品型号:T10317 原产地:中国大陆价格: ¥0.0
产品名称: AMG 487 (S-enantiomer);化合物 T10297AMG 487 (S-enantiomer)
产品简介:amg 487 s-enantiomer is the s enantiomer of amg 487. amg 487 is an cxcr3 antagonist...产品型号:T10297 原产地:中国大陆价格: ¥0.0
产品名称: AMG 487;化合物AMG 487AMG 487
产品简介:amg 487 is a potent and selective antagonist of chemokine (c-x-c motif) receptor 3 (cxcr3) which inhibits the binding of cxcl10 and cxcl11 to cxcr3 with ic50s o..产品型号:T10297L 原产地:中国大陆价格: ¥0.0
产品名称: AMG-548 hydrochloride (864249-60-5 free base);化合物 T10298AMG-548 hydrochloride;AMG-548 hydrochloride
产品简介:amg-548 hydrochloride is an orally active and selective p38α inhibitor (ki: 0.5 nm) and shows slightly selective over p38β (ki: 36 nm) and >1000 fold selective ..产品型号:T10298 原产地:中国大陆价格: ¥0.0
产品名称: AMG-548;化合物 T10298LAMG-548
产品简介:amg-548 is an orally active and selective p38α inhibitor (ki=0.5 nm), shows slightly selective over p38β (ki=36 nm) and >1000 fold selective against p38γ and p3..产品型号:T10298L 原产地:中国大陆价格: ¥0.0