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产品目录

产品展示/Products

  • PI3Kα-IN-6;化合物 PI3Kα-IN-6PI3Kα-IN-6

    产品名称: PI3Kα-IN-6;化合物 PI3Kα-IN-6PI3Kα-IN-6

    产品简介:pi3kα-in-6 (compound 5b) is a pi3kα inhibitor that exhibits anticancer effects without toxicity to normal cells. pi3kα-in-6 increases ros production, decreases ..

    产品型号:T62073 原产地:中国大陆价格: ¥0.0

  • COX-2/PI3K-IN-1;化合物 COX-2/PI3K-IN-1COX-2/PI3K-IN-1

    产品名称: COX-2/PI3K-IN-1;化合物 COX-2/PI3K-IN-1COX-2/PI3K-IN-1

    产品简介:cox-2/pi3k-in-1 (compound 5d) is a potent inhibitor of pi3k (ic50: 1.14 nm). cox-2/pi3k-in-1 is a selective inhibitor of cox-2 (ki: 3.24 nm)...

    产品型号:T62103 原产地:中国大陆价格: ¥0.0

  • PI3Kγ inhibitor 4;化合物 PI3Kγ inhibitor 4PI3Kγ inhibitor 4

    产品名称: PI3Kγ inhibitor 4;化合物 PI3Kγ inhibitor 4PI3Kγ inhibitor 4

    产品简介:pi3kγ inhibitor 4 is a selective, potent, orally active pi3kγ inhibitor (ic50: 40 nm). pi3kγ inhibitor 4 is ~7-fold more selective for pi3kγ than the α subtype,..

    产品型号:T62165 原产地:中国大陆价格: ¥0.0

  • PI3KC2α-IN-1;化合物 PI3KC2α-IN-1PI3KC2α-IN-1

    产品名称: PI3KC2α-IN-1;化合物 PI3KC2α-IN-1PI3KC2α-IN-1

    产品简介:pi3kc2α-in-1 is a potent inhibitor of pi3kc2α with an ic50 value of 95 nm. pi3kc2α-in-1 interacts with the atp binding site of pi3kc2α. pi3kc2α-in-1 impairs the..

    产品型号:T62289 原产地:中国大陆价格: ¥0.0

  • PI3K/HDAC-IN-2;化合物 PI3K/HDAC-IN-2PI3K/HDAC-IN-2

    产品名称: PI3K/HDAC-IN-2;化合物 PI3K/HDAC-IN-2PI3K/HDAC-IN-2

    产品简介:pi3k/hdac-in-2 is a potent dual pi3k/hdac inhibitor, capable of acting on pi3kα (ic50: 226 nm), pi3kβ (ic50: 279 nm), pi3kγ (ic50: 467 nm), pi3kδ (ic50: 29 nm),..

    产品型号:T62912 原产地:中国大陆价格: ¥0.0

  • PI3Kδ/γ-IN-3;化合物 PI3Kδ/γ-IN-3PI3Kδ/γ-IN-3

    产品名称: PI3Kδ/γ-IN-3;化合物 PI3Kδ/γ-IN-3PI3Kδ/γ-IN-3

    产品简介:pi3kδ/γ-in-3 (compound 58) is an orally active dual inhibitor of pi3kδ (ic50: 1 nm) and pi3kγ (ic50: 16 nm). pi3kδ/γ-in-3 can induce apoptosis of tumor cells, w..

    产品型号:T63078 原产地:中国大陆价格: ¥0.0

  • PI3Kβ-IN-1;化合物 PI3Kβ-IN-1PI3Kβ-IN-1

    产品名称: PI3Kβ-IN-1;化合物 PI3Kβ-IN-1PI3Kβ-IN-1

    产品简介:pi3kβ-in-1 is a selective, orally active pi3kβ inhibitor (ic50: 2 nm)...

    产品型号:T62948 原产地:中国大陆价格: ¥0.0

  • PI3K/AKT-IN-1;化合物 PI3K/AKT-IN-1PI3K/AKT-IN-1

    产品名称: PI3K/AKT-IN-1;化合物 PI3K/AKT-IN-1PI3K/AKT-IN-1

    产品简介:pi3k/akt-in-1 is a potent, dual pi3k/akt inhibitor that acts on pi3kγ (ic50: 6.99 μm), pi3kδ (ic50: 4.01 μm) and akt (ic50: 3.36 μm). pi3k/akt-in-1 induces casp..

    产品型号:T62997 原产地:中国大陆价格: ¥0.0

  • PI3K/mTOR Inhibitor-7;化合物 PI3K/mTOR Inhibitor-7PI3K/mTOR Inhibitor-7

    产品名称: PI3K/mTOR Inhibitor-7;化合物 PI3K/mTOR Inhibitor-7PI3K/mTOR Inhibitor-7

    产品简介:pi3k/mtor inhibitor-7 is a potent dual pi3k/mtor inhibitor. pi3k/mtor inhibitor-7 is 4.7-fold more potent than gedatolisib, with ic50 values of 1.4 μm and 0.3 μ..

    产品型号:T64041 原产地:中国大陆价格: ¥0.0

  • PI4KIIIbeta-IN-11;化合物 PI4KIIIbeta-IN-11PI4KIIIbeta-IN-11

    产品名称: PI4KIIIbeta-IN-11;化合物 PI4KIIIbeta-IN-11PI4KIIIbeta-IN-11

    产品简介:pi4kiiibeta-in-11 is a pi4kiiiβ inhibitor (mean pic50=9.1) that can be used to study diseases caused by rna viruses and plasmodium falciparum...

    产品型号:T64106 原产地:中国大陆价格: ¥0.0

  • PI3K/mTOR Inhibitor-6;化合物 PI3K/mTOR Inhibitor-6PI3K/mTOR Inhibitor-6

    产品名称: PI3K/mTOR Inhibitor-6;化合物 PI3K/mTOR Inhibitor-6PI3K/mTOR Inhibitor-6

    产品简介:pi3k/mtor inhibitor-6 (compound 19c) is a potent dual pi3k/mtor inhibitor that is more stable than gedatolisib in artificial gastric fluid. 10 μm of pi3k/mtor i..

    产品型号:T64219 原产地:中国大陆价格: ¥0.0

  • PI3Kδ-IN-16;PI3Kδ抑制剂16PI3Kδ-IN-16

    产品名称: PI3Kδ-IN-16;PI3Kδ抑制剂16PI3Kδ-IN-16

    产品简介:pi3kδ-in-16 is a selective and potent pi3kδ inhibitor with anticancer and antiproliferative activity, induces cell cycle arrest and apoptosis...

    产品型号:T77667 原产地:中国大陆价格: ¥0.0

  • PI5P4Kα-IN-1;化合物 PI5P4Kα-IN-1PI5P4Kα-IN-1

    产品名称: PI5P4Kα-IN-1;化合物 PI5P4Kα-IN-1PI5P4Kα-IN-1

    产品简介:pi5p4kα-in-1 (compound 13) is a phosphatidylinositol 5-phosphate 4-kinase (pi5p4k) inhibitor, displaying ic50 values of 2 μm for pi5p4kα and 9.4 μm for pi5p4kβ,..

    产品型号:T78178 原产地:中国大陆价格: ¥0.0

  • IHMT-PI3K-455;化合物 IHMT-PI3K-455IHMT-PI3K-455

    产品名称: IHMT-PI3K-455;化合物 IHMT-PI3K-455IHMT-PI3K-455

    产品简介:ihmt-pi3k-455 (compound 15u) is a potent, selective pi3kγ/δ dual inhibitor, demonstrating oral activity, with ic50 values of 7.1 nm for pi3kγ and 0.57 nm for pi..

    产品型号:T78836 原产地:中国大陆价格: ¥0.0

  • PI3Kα-IN-12;化合物 PI3Kα-IN-12PI3Kα-IN-12

    产品名称: PI3Kα-IN-12;化合物 PI3Kα-IN-12PI3Kα-IN-12

    产品简介:pi3kα-in-12 (compound 13), a potent and selective pi3kα inhibitor (ic50: 1.2 nm), effectively suppresses hct-116 and u87-mg cell proliferation with ic50 values ..

    产品型号:T78804 原产地:中国大陆价格: ¥0.0

  • PI3K-IN-47;化合物 PI3K-IN-47PI3K-IN-47

    产品名称: PI3K-IN-47;化合物 PI3K-IN-47PI3K-IN-47

    产品简介:pi3k-in-47 (compound 27) is a potent bivalent inhibitor targeting the phosphoinositide 3-kinases (pi3k) family, exhibiting inhibitory concentration (ic50) value..

    产品型号:T78853 原产地:中国大陆价格: ¥0.0

  • PI3K-IN-41;化合物 PI3K-IN-41PI3K-IN-41

    产品名称: PI3K-IN-41;化合物 PI3K-IN-41PI3K-IN-41

    产品简介:pi3k-in-41 (compound 2), a photocaged pi3k inhibitor (ic50=18.92 nm) with anticancer properties, demonstrates potent pi3k inhibition following uv light irradiat..

    产品型号:T79566 原产地:中国大陆价格: ¥0.0

  • PI5P4K-β-IN-2;化合物 PI5P4K-β-IN-2PI5P4K-β-IN-2

    产品名称: PI5P4K-β-IN-2;化合物 PI5P4K-β-IN-2PI5P4K-β-IN-2

    产品简介:pi5p4k-β-in-2 (compound d5) is a potent inhibitor of the pi5p4k-β enzyme, demonstrating an ic50 value of 0.35 μm and exhibiting antitumor activity...

    产品型号:T81464 原产地:中国大陆价格: ¥0.0

  • PI5P4K-β-IN-1;化合物 PI5P4K-β-IN-1PI5P4K-β-IN-1

    产品名称: PI5P4K-β-IN-1;化合物 PI5P4K-β-IN-1PI5P4K-β-IN-1

    产品简介:pi5p4k-β-in-1 (compound vs1) is a potent pi5p4k-β inhibitor with an ic50 of 0.80 μm [1]...

    产品型号:T81465 原产地:中国大陆价格: ¥0.0

  • PI5P4Ks-IN-3;化合物 PI5P4Ks-IN-3PI5P4Ks-IN-3

    产品名称: PI5P4Ks-IN-3;化合物 PI5P4Ks-IN-3PI5P4Ks-IN-3

    产品简介:pi5p4ks-in-3 (compound 30) is a covalent inhibitor of pi5p4k, exhibiting inhibition constants (ic50s) of 1.34 μm for pi5p4kα and 9.9 μm for pi5p4kβ. notably, th..

    产品型号:T81466 原产地:中国大陆价格: ¥0.0

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