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产品名称: (E)-AG 99;化合物AG 99(E)-Tyrphostin AG 99|||(E)-Tyrphostin 46|||AG 99|||Tyrphostin 46;(E)-Tyrphostin AG
产品简介:(e)-ag 99 ((e)-tyrphostin ag 99) is an inhibitor of egfr kinase (ic50: 10 μm in the human epidermoid carcinoma cell line a431)...产品型号:T5155 原产地:中国大陆价格: ¥0.0
产品名称: 2,3,2’’,3’’-Tetrahydroochnaflavone化合物 T5156金银花
产品简介:2,3,2´´,3´´-tetrahydroochnaflavone is a natural product of lonicera, caprifoliaceae. the catalog number is t5156 and the cas number is 6..产品型号:T5156 原产地:中国大陆价格: ¥0.0
产品名称: 9,13-Epidioxy-8(14)-abieten-18-oic acid;化合物 T51579,13-Epidioxy-8(14)-abieten-18-oic acid
产品简介:9,13β-epidioxy-8(14)-abieten-18-oic acid has anti-inflammatory activities, it exhibits moderate activities on no levels in lps-stimulated murine microglia bv2 c..产品型号:T5157 原产地:中国大陆价格: ¥0.0
产品名称: SR3335;化合物SR3335ML 176;ML 176
产品简介:sr3335 (ml 176) is a selective inverse agonist of rorα, competitively inhibiting the binding of 25-hydroxycholesterol to the ligand binding domain (ki: 220 nm)...产品型号:T5160 原产地:中国大陆价格: ¥0.0
产品名称: SR1001;化合物SR1001SR1001
产品简介:sr 1001 is an inverse agonist for rorα/rorγ (kis: 172/111 nm)...产品型号:T5163 原产地:中国大陆价格: ¥0.0
产品名称: Leniolisib;化合物LeniolisibCDZ173;CDZ173
产品简介:leniolisib (cdz173) (cdz173) is a potent and selective pi3kδ inhibitor (ic50: 11 nm)...产品型号:T5166 原产地:中国大陆价格: ¥0.0
产品名称: Leniolisib phosphate;化合物 T5166LLeniolisib monophosphate;Leniolisib monophosphate
产品简介:leniolisib phosphate is an effective pi3k inhibitor...产品型号:T5166L 原产地:中国大陆价格: ¥0.0
产品名称: FM-381;化合物FM381FM381;FM381
产品简介:fm381 is a potent covalent reversible inhibitor of jak3. fm-381 has an ic50 of 127 pm for jak3, with 410, 2700 and 3600-fold selectivity over jak1, jak2 and tyk..产品型号:T5091 原产地:中国大陆价格: ¥0.0
产品名称: AIM-100;化合物AIM-100AIM100;AIM100
产品简介:aim-100 is a ack1 inhibitor (ic50: 24 nm)...产品型号:T5092 原产地:中国大陆价格: ¥0.0
产品名称: Pim1/AKK1-IN-1;化合物Pim1/AKK1-IN-1LKB1/AAK1 dual inhibitor|||MDK-2275;LKB1/AAK1 dual inhibitor|||MDK-2
产品简介:pim1/akk1-in-1 (lkb1/aak1 dual inhibitor) is a potent multi-kinase inhibitor with kd values of 35 nm/53 nm/75 nm/380 nm for pim1/akk1/mst2/lkb1 respectively, an..产品型号:T5093 原产地:中国大陆价格: ¥0.0
产品名称: SRT 1720化合物SRT 1720N-[2-[3-(1-哌嗪基甲基)咪唑并[2,1-B]噻唑-6-基]苯基]-2-喹喔啉甲酰胺
产品简介:srt 1720 is a selective activator of human sirt1 (ec1.5: 0.16 μm) and is >230-fold less potent for sirt2 and sirt3...产品型号:T5096 原产地:中国大陆价格: ¥0.0
产品名称: Ezatiostat;化合物EzatiostatTER199(free base)|||TLK199;TER199(free base)|||TLK199
产品简介:ezatiostat (ter199(free base)) is a tripeptide analog of glutathione that can selectively inhibit gstp1-1 catalytic activity...产品型号:T5097 原产地:中国大陆价格: ¥0.0
产品名称: Gefapixant;化合物GefapixantRO 4926219|||AF219|||MK-7264;RO 4926219|||AF219|||MK-7264
产品简介:gefapixant (af219) is a p2x3 receptor (p2x3r) antagonist with ic50 of ~30 nm at recombinant hp2x3 homotrimers and 100-250 nm at hp2x2/3 heterotrimeric receptors..产品型号:T5099 原产地:中国大陆价格: ¥0.0
产品名称: DJ-V-159化合物DJ-V159DJ-V159
产品简介:dj-v-159 is a gprc6a agonist, targeting the g protein-coupled receptor family c group 6 member a (gprc6a)...产品型号:T5100 原产地:中国大陆价格: ¥0.0
产品名称: BW-A 78U;化合物BW-A78UBW-A78U;BW-A78U
产品简介:bw-a 78u is a pde4 inhibitor (ic50: 3 μm). it is not inhibition on the lipopolysaccharide (lps)-induced tnf-α release...产品型号:T5101 原产地:中国大陆价格: ¥0.0
产品名称: TGN-020;化合物TGN020TGN020;TGN020
产品简介:tgn-020 is an inhibitor of aquaporin 4 (aqp4, ic50: 3.1 μm), the most abundant water channel in the brain...产品型号:T5102 原产地:中国大陆价格: ¥0.0
产品名称: AKOS B018304化合物AKOS B018304(5E)-5-(2-硝基苯亚甲基)-2-硫代-四氢噻唑-4-酮
产品简介:akos b018304 is an arylalkylidene derivative with polar substitution at para-position...产品型号:T5103 原产地:中国大陆价格: ¥0.0
产品名称: BTSA1;化合物BTSA1BTSA1
产品简介:btsa1 is a bax activator that binds with high affinity and specificity to the n-terminal activation site and induces conformational changes to bax leading to ba..产品型号:T5104 原产地:中国大陆价格: ¥0.0
产品名称: BRL-50481;化合物BRL 50481BRL-50481
产品简介:brl-50481 is a novel and selective inhibitor of pde7 with ic50s of 0.15, 12.1, 62 and 490 μm for pde7a, pde7b, pde4 and pde3, respectively...产品型号:T5106 原产地:中国大陆价格: ¥0.0
产品名称: ML311;化合物ML311ML311
产品简介:ml311 is a selective inhibitor of the mcl-1/bim interaction...产品型号:T5108 原产地:中国大陆价格: ¥0.0