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产品名称: SilmitasertibCX-4945;5-[(3-氯苯基)氨基]-苯并[C]-2,6-萘啶-8-羧酸
产品简介:cx-4945 is a potent, orally bioavailable inhibitor of casein kinase 2 (ck2; ki: 0.38 nm)...产品型号:T2259 原产地:中国大陆价格: ¥0.0
产品名称: AM2811-(2,4-二氯苯基)-5-(4-碘苯基)-4-甲基-N-4-吗啉基-1H-吡唑-3-甲酰胺
产品简介:am 281, a cannabinoid antagonist, reduces neurologic dysfunction and mortality rate after cecal ligation and puncture in rats...产品型号:T2264 原产地:中国大陆价格: ¥0.0
产品名称: AG-120 (racemic)1-(4-氰基-2-吡啶基)-5-氧代-L-脯氨酰-2-(2-氯苯基)-N-(3,3-二氟环丁基)-N2-(5-氟-3-吡啶基)甘氨酰胺
产品简介:ag-120 (racemic), the racemic mixture of ag-120, is an orally available isocitrate dehydrogenase type 1 (idh1) inhibitor, and shows potential antineoplastic act..产品型号:T22253 原产地:中国大陆价格: ¥0.0
产品名称: TCS JNK 5aN-(3-氰基-4,5,6,7-四氢苯并[b]噻吩-2-基)-1-萘甲酰胺;SC-202671;SC202671;SC 202671;N-(3-Cyano-4,5,6,7-tetr
产品简介:tcs jnk 5a is an effective, specific inhibitor of jnk3(pic50= 6.7), jnk2(pic50=6.5)...产品型号:T2234 原产地:中国大陆价格: ¥0.0
产品名称: DactolisibNVP-BEZ235;BEZ235;2-甲基-2-[4-[3-甲基-2-氧代-8-(喹啉-3-基)-2,3-二氢咪唑并[4,5-c]喹啉-1-基]苯基]丙腈
产品简介:dactolisib is an orally bioavailable inhibitor of pi3k and mtor (ic50s: 4 nm/5 nm/7 nm/75 nm, and 20.7 nm for p110α/p110γ/p110δ/p110β and mtor)...产品型号:T2235 原产地:中国大陆价格: ¥0.0
产品名称: RU 588414-[3-(4-羟基丁基)-4,4-二甲基-2,5-二氧代-1-咪唑烷基]-2-(三氟甲基)苯腈;HMR-3841;RU58841;PSK-3841
产品简介:ru 58841 is a specific androgen receptor antagonist or anti-androgen; ru 58841 has a significant effect on hair regrowth...产品型号:T2236 原产地:中国大陆价格: ¥0.0
产品名称: MYF-01-371-[3-Methyl-3-[3-(trifluoromethyl)anilino]pyrrolidin-1-yl]prop-2-en-1-one
产品简介:myf-01-37 is a novel covalent tead inhibitor...产品型号:T22372 原产地:中国大陆价格: ¥0.0
产品名称: Nor-benzetimideNorbenzetimide;3-苯基-[3,4-联哌啶]-2,6-二酮
产品简介:norbenzetimide, an organic compound, is prepared from benzetimide by catalytic transfer hydrogenolysis...产品型号:T22380 原产地:中国大陆价格: ¥0.0
产品名称: Wnt-C594-(2-甲基-4-吡啶基)-N-[4-(3-吡啶基)苯基]苯乙酰胺;C59
产品简介:wnt-c59(c59) is a highly effective and specific wnt signaling antagonis with porcn enzymatic activity...产品型号:T2242 原产地:中国大陆价格: ¥0.0
产品名称: 1-(4-Chloro-3-(trifluoromethyl)phenyl)-3-(4-(4-cyanophenoxy)phenyl)urea
产品简介:sc-1 is a a derivative of the multiple tyrosine kinase inhibitor sorafenib. sc-1 potently inhibits the phosphorylation of stat3 by blocking stat3 phosphorylatio..产品型号:T22424 原产地:中国大陆价格: ¥0.0
产品名称: AM-2232AM2232;AM 2232;UNII-40KCH8YIKP;3-(1-萘基羰基)-1H-吲哚-1-戊腈
产品简介:am-2232 is a potent and unselective agonist of the cannabinoid receptors...产品型号:T21450 原产地:中国大陆价格: ¥0.0
产品名称: Temozolomide Acid3,4-二氢-3-甲基-4-氧代咪唑并[5,1-D]-1,2,3,5-四嗪-8-甲酰胺酸;TMZA
产品简介:temozolomide acid is a metabolite of temozolomide (tmz). temozolomide processes anticancer activity in vitro. temozolomide (tmz) is an oral alkylating agent use..产品型号:T21463 原产地:中国大陆价格: ¥0.0
产品名称: AZD-5597(S)-(4-((5-Fluoro-4-(1-isopropyl-2-methyl-1H-imidazol-5-yl)pyrimidin-2-yl)amino)phenyl)(3-(m
产品简介:azd-5597 is a potent imidazole pyrimidine amide cdk inhibitor...产品型号:T21544 原产地:中国大陆价格: ¥0.0
产品名称: SKF-96365 hydrochloride1-[2-(4-甲氧基)-2-[3-(4-甲氧基苯基)丙氧基]乙基]咪唑;SKF96365
产品简介:skf-96365, a soce inhibitor, exhibits potent anti-neoplastic activity by inducing cell-cycle arrest and apoptosis in colorectal y cells. skf-96365 can induce cy..产品型号:T2170 原产地:中国大陆价格: ¥0.0
产品名称: S-23S23;(S)-3-(4-chloro-3-fluorophenoxy)-N-(4-cyano-3-(trifluoromethyl)phenyl)-2-hydroxy-2-methylpro
产品简介:s-23 is an oral selective androgen receptor modulator (sarm) with a ki of 1.7 nm. s-23 increases prostate, seminal vesicle, and levator ani muscle weights in ca..产品型号:T20789 原产地:中国大陆价格: ¥0.0
产品名称: RU 24969 hemisuccinate5-甲氧基-3-(1,2,5,6-四氢-4-吡啶基)-1H-吲哚半琥珀酸盐
产品简介:ru 24969 is a selective agonist at the 5-ht1a and 5-ht1b receptors...产品型号:T2289 原产地:中国大陆价格: ¥0.0
产品名称: m-Chlorophenylbiguanide hydrochloride1-(3-氯苯基)双胍;1-(3-Chlorophenyl)biguanidehydrochloride
产品简介:m-chlorophenylbiguanide hydrochloride is a 5-ht3 receptor agonist. m-chlorophenylbiguanide hydrochloride selectively binds 5-ht3(ki: 0.002 ?m) over 5-ht1a(ki: 1..产品型号:T22959 原产地:中国大陆价格: ¥0.0
产品名称: DL-AP3DL-2-氨基-3-磷丙酸
产品简介:dl-ap3 is a competitive group i metabotropic glutamate receptor antagonist and inhibitor of phosphoserine phosphatase...产品型号:T22730 原产地:中国大陆价格: ¥0.0
产品名称: YK-4-2794,7-二氯-1,3-二氢-3-羟基-3-[2-(4-甲氧基苯基)-2-氧代乙基]-2H-吲哚-2-酮
产品简介:yk 4-279, an inhibitor of rna helicase a (rha), binds to the oncogenic transciption factor ews-fli1...产品型号:T2275 原产地:中国大陆价格: ¥0.0
产品名称: RI-1RI-1; 3-氯-1-(3,4-二氯苯基)-4-(4-吗啉基)-1H-吡咯-2,5-二酮;RI1;RI 1;RAD51 inhibitor 1
产品简介:ri-1 is a rad51 inhibitor (ic50: 5-30 μm)...产品型号:T2276 原产地:中国大陆价格: ¥0.0