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产品名称: α-MSHMelanocortin Receptor,hormone,αMSH,inhibit,Inhibitor,α MSH,neuroimmunomodulatory,inflammation,e
产品简介:α-msh is amide stimulates melanocortin 1 receptor that results in the activation of adenylyl cyclase...产品型号:T7813 原产地:中国大陆价格: ¥0.0
产品名称: JHU37152JHU37152,inhibit,hM3Dq,Clozapine,Inhibitor,DREADD,Muscarinic acetylcholine receptor,mAChR,hM
产品简介:jhu 37152 is a designer receptors exclusively activated by designer drug (dreadd) agonist with ki of 1.8 nm and 8.7 nm for human muscarinic acetylcholine m3 rec..产品型号:T9019 原产地:中国大陆价格: ¥0.0
产品名称: BAY-545Inhibitor,BAY 545,BAY545,Adenosine Receptor,BAY-545,P1 receptor,inhibit
产品简介:bay-545 is an antagonist of a2b adenosine receptor(ic50 : 59 nm)...产品型号:T8512 原产地:中国大陆价格: ¥0.0
产品名称: TozadenantP1 receptor,SYN-115,Adenosine Receptor,SYN 115,Tozadenant,Inhibitor,inhibit
产品简介:tozadenant is an adenosine a2a receptor antagonist(ki of 11.5 nm and 6 nm on human and rhesus,respectively)..产品型号:T7320 原产地:中国大陆价格: ¥0.0
产品名称: NPS2390Inhibitor,NPS2390,Calcium-sensing receptor,NPS-2390,mGluR,inhibit,Metabotropic glutamate rece
产品简介:nps2390 is a first generation quinoxaline derivative that acts as a noncompetitive antagonist of mglur1 and mglur5 (ic50 of 5.2 and 82 nm, respectively)..产品型号:T8457 原产地:中国大陆价格: ¥0.0
产品名称: GLP-1 receptor agonist 9GLP 1 receptor agonist 9,Inhibitor,inhibit,Glucagon Receptor,GLP-1 receptor
产品简介:1h-benzimidazole-6-carboxylic acid is a glp-1 receptor agonist...产品型号:T9579 原产地:中国大陆价格: ¥0.0
产品名称: DerazantinibARQ 087,Derazantinib,Fibroblast growth factor receptor,inhibit,FGFR,ARQ087,Inhibitor
产品简介:derazantinib (arq-087) is an atp competitive tyrosine kinase inhibitor. it exhibits potent activity against fgfr1/fgfr2/fgfr3 chondrocytes (ic50s: 4.5 nm/1.8 nm..产品型号:TQ0228 原产地:中国大陆价格: ¥0.0
产品名称: Temgicolurilinhibit,Inhibitor,γ-Aminobutyric acid Receptor,Mebicar,Temgicoluril,Gamma-aminobutyric a
产品简介:temgicoluril acts on?gaba receptor...产品型号:T9424 原产地:中国大陆价格: ¥0.0
产品名称: Pimavanserin tartrateInhibitor,Pimavanserin hemitartrate,5-hydroxytryptamine Receptor,ACP-103 hemita
产品简介:pimavanserin is an effective and specific serotonin 5-ht2a inverse agonist (pic50: 8.73), used in the therapy of psychosis associated with parkinson´s dis..产品型号:T6946 原产地:中国大陆价格: ¥0.0
产品名称: TH1020interaction,inhibit,Bacterial,flagellin,TH-1020,TH1020,Toll-like Receptor (TLR),TLR5,protein-p
产品简介:th1020 is a novel inhibitor of toll-like receptor 5 (tlr5)/flagellin complex with promising activity (ic50 =0.85±0.12 μm) and specificity...产品型号:T8727 原产地:中国大陆价格: ¥0.0
产品名称: MyristicinMyristicin,Serotonin Receptor,Inhibitor,5-hydroxytryptamine Receptor,5-HT Receptor,inhibit
产品简介:myristicin is a natural product found in spices and umbelliferous plants. myristicin has anti-cholinergic, antibacterial, and hepatoprotective effects, it also ..产品型号:T9113 原产地:中国大陆价格: ¥0.0
产品名称: BinodenosonMRE 0470,imaging,P1 receptor,stress,oxidative,WRC0470,neutrophil,inhibit,radiotracers,Bin
产品简介:binodenoson is a potent and selective a2a adenosine receptor agonist (kd=270 nm). binodenoson is being developed as a short-acting coronary vasodilator as an ad..产品型号:T9516 原产地:中国大陆价格: ¥0.0
产品名称: Tiagabine hydrochlorideNO050328,TGB,NO-050328,γ-Aminobutyric acid Receptor,NO 050328,inhibit,NO-328,
产品简介:tiagabine hydrochloride is the hydrochloride salt form of tiagabine, a nipecotic acid derivative with anticonvulsant property. a selective gamma-aminobutyric ac..产品型号:T7000 原产地:中国大陆价格: ¥0.0
产品名称: Eplivanserin5-hydroxytryptamine Receptor,Serotonin Receptor,5-HT2A,5-HT Receptor,Eplivanserin,SR4634
产品简介:eplivanserin is an effective and selective antagonist of 5-ht2a receptor with a kd of 1.14 nm and an ic50 value of 5.8 nm in rat cortical membrane...产品型号:T11217 原产地:中国大陆价格: ¥0.0
产品名称: Procyanidin B1Procyanidin B1,Toll-like Receptor (TLR),Inhibitor,Procyanidin B-1,inhibit,Procyanidin
产品简介:procyanidin b1, isolated from commonly eaten fruits, binds to the tlr4/md-2 complex and has anti-inflammatory activity...产品型号:TQ0205 原产地:中国大陆价格: ¥0.0
产品名称: BradykininBradykinin Receptor,Bradykinin,Serine endopeptidases,inhibit,Threonine proteases,Inhibitor
产品简介:bradykinin is an inflammatory mediator. it is a peptide that causes blood vessels to dilate (enlarge) via the release of prostacyclin, nitric oxide, and endothe..产品型号:TP1277 原产地:中国大陆价格: ¥0.0
产品名称: Pazopanib Hydrochlorideinhibit,CD117,CSF1R,GW-786034,Vascular endothelial growth factor receptor,col
产品简介:pazopanib hcl (gw786034 hcl) is a novel multi-target inhibitor of vegfr1, vegfr2, vegfr3, pdgfr, fgfr, c-kit and c-fms with ic50 of 10 nm, 30 nm, 47 nm, 84 nm, ..产品型号:T6930 原产地:中国大陆价格: ¥0.0
产品名称: DAPTAHIV,DAPTA,CC chemokine receptor,Human immunodeficiency virus,inhibit,CCR,Inhibitor
产品简介:dapta(tfa) is an inhibitor of ccr5, shows potent anti-hiv activities...产品型号:T7624 原产地:中国大陆价格: ¥0.0
产品名称: N6-(4-Hydroxybenzyl)adenosineinhibit,P2Y Receptor,Inhibitor
产品简介:n6-(4-hydroxybenzyl)adenosine is a platelet aggregation inhibitor...产品型号:T12164 原产地:中国大陆价格: ¥0.0
产品名称: Motilin (26-47), human, porcineMotilin (26-47), human, porcine,MLNR,Motilin Receptor,Motilin (26 47)
产品简介:motilin (26-47), human and pig are endogenous motilin receptor ligands in chinese hamster ovarian cell lines, with ki and ec50 at 2.3 nm and 0.3 nm, respectivel..产品型号:TP1425 原产地:中国大陆价格: ¥0.0