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产品名称: PARP1/BRD4-IN-2;化合物 PARP1/BRD4-IN-2PARP1/BRD4-IN-2
产品简介:parp1/brd4-in-2 is a potent and selective inhibitor of parp1 (ic50: 197 nm) and brd4 (ic50: 238 nm).parp1/brd4-in-2 inhibits dna damage repair, blocks the g0/g1..产品型号:T62540 原产地:中国大陆价格: ¥0.0
产品名称: JAK3/BTK-IN-4;化合物 JAK3/BTK-IN-4JAK3/BTK-IN-4
产品简介:jak3/btk-in-4 is a potent inhibitor of jak3/btk. btk and jak3 are two important targets in autoimmune diseases. simultaneous inhibition of the btk/jak3 signalin..产品型号:T62553 原产地:中国大陆价格: ¥0.0
产品名称: TGFβRI-IN-4;化合物 TGFβRI-IN-4TGFβRI-IN-4
产品简介:tgfβri-in-4 is a potent, orally active tgfβ receptor type i kinase (tgfβri) inhibitor that acts on alk5 (ic50: 44 nm) and nih3t3 (ic50: 42.5 nm).tgfβri-in-4 inh..产品型号:T62559 原产地:中国大陆价格: ¥0.0
产品名称: TLR7 agonist 4;化合物 TLR7 agonist 4TLR7 agonist 4
产品简介:tlr7 agonist 4 (compound 1.2) is a tlr7 agonist (ec50: 4.3 nm)...产品型号:T62587 原产地:中国大陆价格: ¥0.0
产品名称: TRPC5-IN-4;化合物 TRPC5-IN-4TRPC5-IN-4
产品简介:trpc5-in-4, a potent and safe trpc inhibitor, exhibits ic50 values of 14.07 nm and 65 nm for trpc5 and trpc4, respectively, indicating high efficacy. it does no..产品型号:T62589 原产地:中国大陆价格: ¥0.0
产品名称: Benzyl-piperazine-CO-benzothiazole-4-methylpiperidine;化合物T62461Benzyl-piperazine-CO-benzothiazole-4-
产品简介:benzyl-piperazine-co-benzothiazole-4-methylpiperidine can be used to alter eukaryotic lifespan...产品型号:T62461 原产地:中国大陆价格: ¥0.0
产品名称: Tubulin polymerization-IN-4;化合物 Tubulin polymerization-IN-4Tubulin polymerization-IN-4
产品简介:tubulin polymerization-in-4 is an effective inhibitor of tubulin polymerization (ic50=4.6 μm)。 tubulin polymerization-in-4 can destroy tubulin polymerization, b..产品型号:T61940 原产地:中国大陆价格: ¥0.0
产品名称: PARP1/BRD4-IN-1;化合物 PARP1/BRD4-IN-1PARP1/BRD4-IN-1
产品简介:parp1/brd4-in-1 is a highly selective and potent inhibitor of parp1 (ic50: 49 nm) and brd4 (ic50: 202 nm).parp1/brd4-in-1 inhibits the expression and activity o..产品型号:T63471 原产地:中国大陆价格: ¥0.0
产品名称: HDAC6-IN-4;化合物 HDAC6-IN-4HDAC6-IN-4
产品简介:hdac6-in-4 (c10) is an orally active, highly selective, potent and non-significantly toxic hdac6 inhibitor (ic50: 23 nm). hdac6-in-4 induces apoptosis and exhib..产品型号:T63472 原产地:中国大陆价格: ¥0.0
产品名称: HDAC1-IN-4;化合物 HDAC1-IN-4HDAC1-IN-4
产品简介:hdac1-in-4 is a potent inhibitor of plasmodium falciparum hdac1 (pfhdac1) with low cytotoxicity and antimalarial effects (ic50<5 nm)...产品型号:T63482 原产地:中国大陆价格: ¥0.0
产品名称: IRE1α kinase-IN-4;化合物 IRE1α kinase-IN-4IRE1α kinase-IN-4
产品简介:ire1α kinase-in-4 (compound 6) is a potent inhibitor of ire1α, exhibiting a ki value of 140 nm. it acts as an atp-competitive ligand for ire1α [1]...产品型号:T63511 原产地:中国大陆价格: ¥0.0
产品名称: THR-β agonist 4;化合物 THR-β agonist 4THR-β agonist 4
产品简介:thr-β agonist 4 is a potent agonist of thr-β. thr-β agonist 4 has shown research potential for metabolic diseases such as hyperlipidemia, obesity, hypercholeste..产品型号:T63515 原产地:中国大陆价格: ¥0.0
产品名称: BuChE-IN-4;化合物 BuChE-IN-4BuChE-IN-4
产品简介:buche-in-4 is a potent inhibitor of buche (ic50: 7.7 nm) and exhibits mild antioxidant capacity, non-toxicity, lipophilicity and neuroprotective effects...产品型号:T63517 原产地:中国大陆价格: ¥0.0
产品名称: (3S,4R)-PF-6683324;化合物 (3S,4R)-PF-6683324(3S,4R)-PF-6683324
产品简介:(3s,4r)-pf-6683324 is a pro-myosin-related kinase (trk) inhibitor that has shown research potential for pain and cancer...产品型号:T63641 原产地:中国大陆价格: ¥0.0
产品名称: A 922500;化合物A922500A922500|||DGAT-1 Inhibitor 4a;A922500|||(1R,2R)-2-[[4-[[(苯基氨基)羰基]氨基][1,1-联苯]-4-基]
产品简介:a 922500 (dgat-1 inhibitor 4a) is an inhibitor for human and mouse dgat-1 with ic50 of 7 nm and 24 nm, respectively, good selectivity over related acyltransfera..产品型号:T6365 原产地:中国大陆价格: ¥0.0
产品名称: A-966492化合物A9664922-[2-氟-4-[(2S)-2-吡咯烷基]苯基]-1H-苯并咪唑-7-甲酰胺
产品简介:a-96649 is a new-type and effective inhibitor. the ki of a-966492 for parp1 and parp2 is 1 nm and 1.5 nm, respectively...产品型号:T6366 原产地:中国大陆价格: ¥0.0
产品名称: FGFR4-IN-9;化合物 FGFR4-IN-9FGFR4-IN-9
产品简介:fgfr4-in-9 is a selective inhibitor of fgfr4 (ic50: 75.3 nm) that effectively inhibits the growth and angiogenesis of hepatocellular carcinoma cells...产品型号:T63662 原产地:中国大陆价格: ¥0.0
产品名称: FGFR4-IN-7;化合物 FGFR4-IN-7FGFR4-IN-7
产品简介:fgfr4-in-7 is a covalent, reversible fgfr4 inhibitor (ic50: 0.42 μm) that blocks the fgfr4 signaling pathway, thereby inducing apoptosis...产品型号:T63692 原产地:中国大陆价格: ¥0.0
产品名称: sEH inhibitor-4;化合物 sEH inhibitor-4sEH inhibitor-4
产品简介:seh inhibitor-4 (compound b15) has been identified as a potent soluble epoxide hydrolase (seh) inhibitor with a remarkable inhibitory potency of 0.03 ± 0.01 nm...产品型号:T63700 原产地:中国大陆价格: ¥0.0
产品名称: DENV-IN-4;化合物 DENV-IN-4DENV-IN-4
产品简介:denv-in-4 is a potent inhibitor of denv (denv ec50=4.79 μm, vero cc50>100 μm, si>20.9). the antiviral effect was demonstrated by the concentration-dependent red..产品型号:T63598 原产地:中国大陆价格: ¥0.0