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产品目录

产品展示/Products

  • IDO1/TDO-IN-4;化合物 IDO1/TDO-IN-4IDO1/TDO-IN-4

    产品名称: IDO1/TDO-IN-4;化合物 IDO1/TDO-IN-4IDO1/TDO-IN-4

    产品简介:ido1/tdo-in-4 displays potent inhibition of both ido1 (ic50 = 3.53 μm) and tdo (ic50 = 1.15 μm) and has an acceptable safety profile and pharmacokinetic propert..

    产品型号:T60318 原产地:中国大陆价格: ¥0.0

  • AZ8838;化合物 AZ8838AZ8838

    产品名称: AZ8838;化合物 AZ8838AZ8838

    产品简介:az8838 is an effective, competitive, allosteric, orally active non-peptide small molecule antagonist of par2 with a pk i of 6.4 for hpar2 [1]...

    产品型号:T60319 原产地:中国大陆价格: ¥0.0

  • Birabresib;化合物BirabresibOTX-015|||OTX015 (MK 8628/Birabresib)|||MK-8628;OTX-015|||OTX015 (MK 8628/Bi

    产品名称: Birabresib;化合物BirabresibOTX-015|||OTX015 (MK 8628/Birabresib)|||MK-8628;OTX-015|||OTX015 (MK 8628/Bi

    产品简介:birabresib (mk-8628) is a synthetic, small molecule inhibitor of the bet (bromodomain and extra-terminal) family of bromodomain-containing proteins 2, 3 and 4 w..

    产品型号:T6032 原产地:中国大陆价格: ¥0.0

  • Antifungal agent 36;化合物 Antifungal agent 36Antifungal agent 36

    产品名称: Antifungal agent 36;化合物 Antifungal agent 36Antifungal agent 36

    产品简介:antifungal agent 36 is a potent anti-fungal agent that shows anti-fungal activity for basidiomycetes [1]...

    产品型号:T60320 原产地:中国大陆价格: ¥0.0

  • Tubulysin IM-3;化合物 Tubulysin IM-3Tubulysin IM-3

    产品名称: Tubulysin IM-3;化合物 Tubulysin IM-3Tubulysin IM-3

    产品简介:tubulysin im-3 is an adc cytotoxin as well as tubulin binder. tubulysin im-3 can be used as anti-microtubule toxins...

    产品型号:T60321 原产地:中国大陆价格: ¥0.0

  • Mopivabil;化合物 MopivabilMopivabil

    产品名称: Mopivabil;化合物 MopivabilMopivabil

    产品简介:mopivabil is the angiotensin ii receptor antagonist[1]...

    产品型号:T60323 原产地:中国大陆价格: ¥0.0

  • Fungicide4;化合物 Fungicide4Fungicide4

    产品名称: Fungicide4;化合物 Fungicide4Fungicide4

    产品简介:fungicide4 exhibits the high activity against the p. infestans strain...

    产品型号:T60324 原产地:中国大陆价格: ¥0.0

  • CAPSO;化合物 CAPSOCAPSO

    产品名称: CAPSO;化合物 CAPSOCAPSO

    产品简介:capso is a biological zwitterionic buffer with a useful ph range from 8.9 to 10.3 [1]...

    产品型号:T60326 原产地:中国大陆价格: ¥0.0

  • Falimint;化合物 FalimintFalimint

    产品名称: Falimint;化合物 FalimintFalimint

    产品简介:falimint is a compound with antipyretic and analgesic activity [1]...

    产品型号:T60327 原产地:中国大陆价格: ¥0.0

  • CDK4/6-IN-12;化合物 CDK4/6-IN-12CDK4/6-IN-12

    产品名称: CDK4/6-IN-12;化合物 CDK4/6-IN-12CDK4/6-IN-12

    产品简介:cdk4/6-in-12 is a potent cyclin-dependent kinase 4/6 (cdk4/6) inhibitor. cdk4/6-in-12 has enzymatic inhibitory activity against cdk4 and cdk6 with ic 50 of 592...

    产品型号:T60328 原产地:中国大陆价格: ¥0.0

  • Mepixetil;化合物 MepixetilMepixetil

    产品名称: Mepixetil;化合物 MepixetilMepixetil

    产品简介:mepixetil is a potent angiotensin ii receptor antagonist[1]...

    产品型号:T60329 原产地:中国大陆价格: ¥0.0

  • Acridone-4-carboxylic acid;化合物 Acridone-4-carboxylic acidAcridone-4-carboxylic acid

    产品名称: Acridone-4-carboxylic acid;化合物 Acridone-4-carboxylic acidAcridone-4-carboxylic acid

    产品简介:acridone-4-carboxylic acid (aca) (compound 2c), a heme-interacting acridone derivative, inhibits free heme-mediated protein oxidation and degradation, and reduc..

    产品型号:T60331 原产地:中国大陆价格: ¥0.0

  • Methacholine bromide;化合物 Methacholine bromideMethacholine bromide

    产品名称: Methacholine bromide;化合物 Methacholine bromideMethacholine bromide

    产品简介:methacholine bromide (acetyl-β-methylcholine bromide) is a potent muscarinic-3 (m3) agonist that specifically acts on acetylcholine receptors located on smooth ..

    产品型号:T60332 原产地:中国大陆价格: ¥0.0

  • DYRK1-IN-1;化合物 DYRK1-IN-1DYRK1-IN-1

    产品名称: DYRK1-IN-1;化合物 DYRK1-IN-1DYRK1-IN-1

    产品简介:dyrk1-in-1 is a highly selective and ligand-efficient dyrk1a inhibitor. dyrk1-in-1 inhibits dyrk1a phosphorylation activity with an ic 50 value of 220 nm. dyrk1..

    产品型号:T60334 原产地:中国大陆价格: ¥0.0

  • Procyclidine;化合物 ProcyclidineProcyclidine

    产品名称: Procyclidine;化合物 ProcyclidineProcyclidine

    产品简介:procyclidine (tricyclamol; (±)-procyclidine) is an anticholinergic agent which is a muscarinic receptor antagonist as well as an n-methyl-d-aspartate ( nmda ) a..

    产品型号:T60578 原产地:中国大陆价格: ¥0.0

  • CEase-IN-1;化合物 CEase-IN-1CEase-IN-1

    产品名称: CEase-IN-1;化合物 CEase-IN-1CEase-IN-1

    产品简介:cease-in-1 (compound a1h3) is a potent and selective inhibitor of cholesterol esterase (cease) with an ic 50 of 0.36 μm. it can be used in hypercholesterolemia ..

    产品型号:T60579 原产地:中国大陆价格: ¥0.0

  • LY2886721;化合物LY2886721LY2886721

    产品名称: LY2886721;化合物LY2886721LY2886721

    产品简介:ly2886721, a bace inhibitor, is used for the therapy of alzheimer´s disease...

    产品型号:T6058 原产地:中国大陆价格: ¥0.0

  • A1AR antagonist 2;化合物 A1AR antagonist 2A1AR antagonist 2

    产品名称: A1AR antagonist 2;化合物 A1AR antagonist 2A1AR antagonist 2

    产品简介:a1ar antagonist 2 (compound 18h) is a potent antagonist of the a1 adenosine receptor (ar). a1ar antagonist 2 has ki values of 1.49, 10.2, and 50.1 nm for ha 1, ..

    产品型号:T60580 原产地:中国大陆价格: ¥0.0

  • Alkannin;化合物 AlkanninAlkannin

    产品名称: Alkannin;化合物 AlkanninAlkannin

    产品简介:alkannin is a potent and specific tumor-specific pyruvate kinase-m2 (pkm2) inhibitor that does not inhibit pkm1 and pyruvate kinase-l (pkl). alkannin is a poten..

    产品型号:T60581 原产地:中国大陆价格: ¥0.0

  • Antibacterial agent 74;化合物 Antibacterial agent 74Antibacterial agent 74

    产品名称: Antibacterial agent 74;化合物 Antibacterial agent 74Antibacterial agent 74

    产品简介:antibacterial agent 74 (compound 36) has anti-salmonella activity [1]...

    产品型号:T60582 原产地:中国大陆价格: ¥0.0

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