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产品名称: BCR-ABL-IN-7;BCR-ABL抑制剂7BCR-ABL-IN-7
产品简介:bcr-abl-in-7 is a wt and t315i mutant abl kinase inhibitor.bcr-abl-in-7 potently inhibits wt and t315i mutant abl kinase activity.bcr-abl-in-7 can be used in ch..产品型号:T72958 原产地:中国大陆价格: ¥0.0
产品名称: THZ2;化合物THZ2CDK7-IN-1;CDK7-IN-1
产品简介:thz2 (cdk7-in-1), an analog of thz1, is a potent and selective cdk7 inhibitor(ic50:13.9 nm),with the potential to treat triple-negative breast cancer (tnbc)...产品型号:T7296 原产地:中国大陆价格: ¥0.0
产品名称: STAT3-IN-7;化合物 STAT3-IN-7STAT3-IN-7
产品简介:stat3-in-7, an orally active aryl sulfonamido azetidine compound, serves as a stat3 inhibitor with anticancer activities...产品型号:T73114 原产地:中国大陆价格: ¥0.0
产品名称: USP7-IN-7;化合物 USP7-IN-7USP7-IN-7
产品简介:usp7-in-7, a potent usp7 inhibitor, exhibits an ic50 value of <10 nm. demonstrating cytotoxicity against both p53-mutant and p53 wild-type blood cancer, as well..产品型号:T73234 原产地:中国大陆价格: ¥0.0
产品名称: EZH2-IN-7;化合物 EZH2-IN-7EZH2-IN-7
产品简介:ezh2-in-7, a potent inhibitor of ezh2, addresses overexpression or mutations in the set region (y641f, y641n, a687v, a677g point mutations) that cause an abnorm..产品型号:T73246 原产地:中国大陆价格: ¥0.0
产品名称: USP7-IN-9;化合物 USP7-IN-9USP7-IN-9
产品简介:usp7-in-9, a potent inhibitor of ubiquitin-specific protease 7 (usp7) with an ic50 of 40.8 nm, effectively induces apoptosis and arrests cell progression at the..产品型号:T73257 原产地:中国大陆价格: ¥0.0
产品名称: USP7-IN-10;化合物 USP7-IN-10USP7-IN-10
产品简介:usp7-in-10 is a potent inhibitor of ubiquitin-specific protease 7 (usp7), exhibiting an inhibition concentration half-maximal (ic50) value of 13.39 nm...产品型号:T73136 原产地:中国大陆价格: ¥0.0
产品名称: CDK7-IN-20;化合物 CDK7-IN-20CDK7-IN-20
产品简介:cdk7-in-20 is a potent, selective, and irreversible inhibitor of cyclin-dependent kinase 7 (cdk7) with an ic50 value of 4 nm, exhibiting over 206-fold selectivi..产品型号:T73163 原产地:中国大陆价格: ¥0.0
产品名称: LRRK2-IN-7;化合物 LRRK2-IN-7LRRK2-IN-7
产品简介:lrrk2-in-7 is a potent lrrk2 kinase inhibitor that demonstrates high selectivity and central nervous system (cns) penetration, possessing an ic50 value of 0.9 n..产品型号:T73176 原产地:中国大陆价格: ¥0.0
产品名称: BuChE-IN-7;化合物 BuChE-IN-7BuChE-IN-7
产品简介:buche-in-7 is a selective inhibitor targeting human butyrylcholinesterase (hbuche) and equine butyrylcholinesterase (eqbuche), demonstrating ic50 values of 40 n..产品型号:T73187 原产地:中国大陆价格: ¥0.0
产品名称: 7-Methylguanosine;7-甲基鸟苷7-Methylguanosine
产品简介:7-methylguanosine is a novel cniiib nucleotidase inhibitor (ic50 : 87.8 ± 7.5 μm)...产品型号:T7319 原产地:中国大陆价格: ¥0.0
产品名称: Tozadenant;化合物TozadenantSYN115;SYN115|||4-羟基-N-[4-甲氧基-7-(4-吗啉基)-2-苯并噻唑基]-4-甲基-1-哌啶甲酰胺
产品简介:tozadenant (syn115) is an adenosine a2a receptor antagonist(ki of 11.5 nm and 6 nm on human and rhesus,respectively)..产品型号:T7320 原产地:中国大陆价格: ¥0.0
产品名称: HIF-2α-IN-7;化合物 HIF-2α-IN-7HIF-2α-IN-7
产品简介:hif-2α-in-7 is a hypoxia inducible factor 2α (hif-2α) inhibitor. hif-2α-in-7 can inhibit hif-2α with an ec 50 value of 6 nm. hif-2α-in-7 can be used for the res..产品型号:T72997 原产地:中国大陆价格: ¥0.0
产品名称: PARP7-IN-12;化合物 PARP7-IN-12PARP7-IN-12
产品简介:parp7-in-12, a potent inhibitor targeting parp7, exhibits an ic50 of 7.836 nm. this compound is applicable in cancer research...产品型号:T73025 原产地:中国大陆价格: ¥0.0
产品名称: KIF18A-IN-7;化合物 KIF18A-IN-7KIF18A-IN-7
产品简介:kif18a-in-7 is an orally active inhibitor targeting kif18a, demonstrating potent inhibition with an ic50 value of 9.4 nm against the microtubule-dependent atpas..产品型号:T73050 原产地:中国大陆价格: ¥0.0
产品名称: ASP-8497;化合物 T30169UNII-GC7THT248G|||ASP8497|||ASP 8497;UNII-GC7THT248G|||ASP8497|||ASP 8497
产品简介:asp8497 is a potent, long-acting dpp-iv inhibitor that improves glucose tolerance by elevating glp-1 levels in a glucose-dependent insulin-stimulating manner. t..产品型号:T30169 原产地:中国大陆价格: ¥0.0
产品名称: ATH-18534;化合物 T30194UNII-V78F7TLP21|||ATH 18534|||SCHEMBL3236065;UNII-V78F7TLP21|||ATH 18534|||SCHEM
产品简介:ath-18534 is a bio-active chemical...产品型号:T30194 原产地:中国大陆价格: ¥0.0
产品名称: Brecanavir;化合物 T30585GW-640385|||GW-640385X|||UNII-E367I8C7FI|||CHEMBL206031|||GW-0385;GW-640385|||G
产品简介:brecanavir is a tyrosyl-based arylsulfonamide, high affinity, protease inhibitor (pi) for the treatment of human immunodeficiency virus type 1...产品型号:T30585 原产地:中国大陆价格: ¥0.0
产品名称: BMS-587101;化合物 T30533UNII-5V7E4UQL93;UNII-5V7E4UQL93
产品简介:bms-587101 is a small molecule antagonist of lfa-1, which can reduce inflammation and joint destruction in the mouse model of arthritis...产品型号:T30533 原产地:中国大陆价格: ¥0.0
产品名称: CHIR98014 HCl (252935-94-7 free base);化合物 T3074LCT-98014|||CHIR-98014 hydrochloride|||CHIR-98014|||C
产品简介:chir98014 is a reversible, cell-permeable inhibitor of gsk3α and gsk3β (ic50s: 0.65 and 0.58 nm). through its effects on gsk3, chir98014 stimulates glycogen syn..产品型号:T3074L 原产地:中国大陆价格: ¥0.0