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产品名称: CYC-116CYC116,inhibit,Inhibitor,CYC-116,CYC 116,Aurora Kinase
产品简介:cyc116 is a potent inhibitor of aurora a/b with ki of 8.0 nm/9.2 nm, is less potent to vegfr2 (ki of 44 nm), with 50-fold greater potency than cdks, not active ..产品型号:T6458 原产地:中国大陆价格: ¥0.0
产品名称: GSK-1520489AGSK1520489A,inhibit,GSK 1520489A,HT29,GSK-1520489A,Inhibitor,active protein kinase
产品简介:gsk-1520489a is an active pkmyt1 inhibitor...产品型号:T9966 原产地:中国大陆价格: ¥0.0
产品名称: BAY1125976inhibit,Inhibitor,Protein kinase B,Akt,BAY 1125976,BAY1125976,PKB,BAY-1125976
产品简介:bay1125976 is an allosteric inhibitor of akt1 and akt2 (ic50s of 5.2 and 18 nm, respectively, in a time-resolved fret assay)..产品型号:T7315 原产地:中国大陆价格: ¥0.0
产品名称: FLLL32FLLL32,Apoptosis,inhibit,JAK,Inhibitor,STAT,Janus kinase,FLLL-32,FLLL 32
产品简介:flll32 is an effective jak2/stat3 inhibitor (ic50 of <5 μm)...产品型号:T6838 原产地:中国大陆价格: ¥0.0
产品名称: BDP5290inhibit,Rho-kinase,Rho-associated kinase,BDP-5290,BDP5290,Rho-associated protein kinase,ROK,B
产品简介:bdp5290 is a potent inhibitor of both rock and mrck(ic50s of 5 nm, 50 nm, 10 nm and 100 nm for rock1, rock2, mrckα and mrckβ, respectively.)..产品型号:T7301 原产地:中国大陆价格: ¥0.0
产品名称: AZD-8835inhibit,PI3K,Inhibitor,AZD 8835,AZD-8835,Phosphoinositide 3-kinase
产品简介:azd8835 is a mixed inhibitor of pi3kα/δ (ic50: 6.2/5.7 nm), also with selectivity against pi3kβ/γ (ic50: 431/90 nm)...产品型号:T6774 原产地:中国大陆价格: ¥0.0
产品名称: NepodinInhibitor,AMP-activated protein kinase,Musizin,Parasite,AMPK,Nepodin,inhibit
产品简介:nepodin has antimalarial, and anti-inflammatory activities, it shows significant cyclooxygenase (cox) inhibitory activity. nepodin has an antidiabetic effect, w..产品型号:TN1100 原产地:中国大陆价格: ¥0.0
产品名称: THZ2inhibit,THZ2,Cyclin dependent kinase,CDK,THZ-2,Inhibitor,THZ 2
产品简介:thz2, an analog of thz1, is a potent and selective cdk7 inhibitor(ic50:13.9 nm),with the potential to treat triple-negative breast cancer (tnbc)...产品型号:T7296 原产地:中国大陆价格: ¥0.0
产品名称: Opaganibinhibit,SphK,Opaganib,Sphingosine kinase,ABC-294640,Inhibitor,ABC 294640
产品简介:abc294640 is an orally active and specific sphingosine kinase-2 (sphk2) inhibitor (ic50: 60 μm)...产品型号:T6750 原产地:中国大陆价格: ¥0.0
产品名称: Epiblastin Ainduces reprogramming,ATP competitive,epiblast stem cells,inhibit,Casein Kinase,Inhibito
产品简介:epiblastin a is an inhibitor of casein kinase 1 (ck1). epiblastin a engages ck1 isoenzymes in cell lysate and induces efficient conversion of epiblast stem cell..产品型号:T8987 原产地:中国大陆价格: ¥0.0
产品名称: TAK-733inhibit,Inhibitor,TAK-733,MAP2K,MAPKK,MEK,Mitogen-activated protein kinase kinase
产品简介:mek inhibitor tak-733 is an orally bioavailable small-molecule inhibitor of mek1 and mek2 (mek1/2) with potential antineoplastic activity...产品型号:T6692 原产地:中国大陆价格: ¥0.0
产品名称: TBK1/IKKε-IN-5I kappa B kinase,Inhibitor,inhibit,IKK,IκB kinase,TBK1/IKKε IN 5,TBK-1/IKKε-IN-5,TBK1/
产品简介:tbk1/ikkε-in-5 is a dual tbk1 and ikkε inhibitor(ic50 of 1 nm and 5.6 nm, respectively)...产品型号:T7951 原产地:中国大陆价格: ¥0.0
产品名称: KY19382Glycogen synthase kinase 3,Beta catenin,β-catenin,GSK-3,KY 19382,inhibit,Wnt,Inhibitor,KY-193
产品简介:ky19382 is a potent and orally active dual inhibitor of cxxc5-dvl and gsk3β( ic50s of 19 and 10 nm, respectively). it activates wnt/β-catenin signaling through ..产品型号:T9025 原产地:中国大陆价格: ¥0.0
产品名称: BI-847325BI 847325,inhibit,Apoptosis,MEK,MAPKK,MAP2K,Inhibitor,Aurora Kinase,Mitogen-activated prote
产品简介:bi-847325 is a selective dual inhibitor of mek and aurora kinases (ak) with ic50 values of 4 and 15 nm for human mek2 and ak-c, respectively...产品型号:T6785 原产地:中国大陆价格: ¥0.0
产品名称: Povorcitinib phosphateJAK,Povorcitinib,Povorcitinib phosphate,CLE,Janus kinase,JAK1 inhibitor,Inhibi
产品简介:povorcitinib phosphate is a selective jak1 inhibitor and can be used in studies about the treatment of cutaneous lupus erythematosus and lichen planus...产品型号:T39113L 原产地:中国大陆价格: ¥0.0
产品名称: MK2-IN-3MAPK activated protein kinase 2,Mitogen-activated protein kinase activated protein kinase 2,
产品简介:mk2-in-3 is a potent, cell-permeable inhibitor of mitogen-activated protein kinase-activated protein kinase 2 (mapkap-k2 or mk-2) and can be used for the treatm..产品型号:T9034 原产地:中国大陆价格: ¥0.0
产品名称: FlavopiridolHMR1275,inhibit,L86-8275,CDK,Cyclin dependent kinase,Inhibitor,Autophagy,HMR 1275,Human
产品简介:flavopiridol (alvocidib) competes with atp to inhibit cdks including cdk1, cdk2, cdk4 and cdk6 with ic50 of ~ 40 nm. it is 7.5-fold more selective for cdk1, 2, ..产品型号:T6837 原产地:中国大陆价格: ¥0.0
产品名称: CCT245737CCT245737,Inhibitor,CCT 245737,inhibit,Checkpoint Kinase (Chk),CCT-245737
产品简介:cct245737 is an orally active and selective chk1 inhibitor (ic50: 1.3 nm); cct245737 shows much less activity against chk2 (ic50: 2440 nm)...产品型号:T7080 原产地:中国大陆价格: ¥0.0
产品名称: CAY10505PI3K,CAY10505,Apoptosis,Phosphoinositide 3-kinase,CAY-10505,CAY 10505,inhibit,Inhibitor
产品简介:cay10505, a form of dehydroxyl of as-252424, is a pi3kγ inhibitor (ic50: 33 nm)...产品型号:T6433 原产地:中国大陆价格: ¥0.0
产品名称: SAR407899SAR 407899,Rho-associated kinase,ROK,Rho-kinase,ROCK,Rho-associated protein kinase,SAR40789
产品简介:sar407899 is rho kinase inhibitor potently inhibits endothelin-1-induced constriction of renal resistance arteries...产品型号:T7391 原产地:中国大陆价格: ¥0.0