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产品名称: BSJ-4-116CDK,degrader,antiproliferative,inhibit,Kelly,C1039F,BSJ 4 116,Cyclin dependent kinase,PROTA
产品简介:bsj-4-116 is a highly potent and selective cdk12 degrader (protac) with an ic50 of 6 nm. it downregulates ddr genes through a premature termination of transcrip..产品型号:T9117 原产地:中国大陆价格: ¥0.0
产品名称: SelitrectinibInhibitor,LOXO195,Tropomyosin related kinase receptor,LOXO 195,Selitrectinib,Trk Recept
产品简介:selitrectinib is a potent and selective inhibitor of the receptor tyrosine kinases(trk)( trka and trkc with ic50s of 0.6 and <2.5 nm, respectively)..产品型号:T7435 原产地:中国大陆价格: ¥0.0
产品名称: DRB5,6-Dichlorobenzimidazole riboside,DRB,inhibit,Inhibitor,CDK,Cyclin dependent kinase
产品简介:drb is a nucleoside analog that inhibits several carboxyl-terminal domain (ctd) kinases including casein kinase ii (ic50 range of 4-10 μm)..产品型号:T7789 原产地:中国大陆价格: ¥0.0
产品名称: BIX 02565Inhibitor,BIX02565,BIX-02565,Ribosomal S6 Kinase (RSK),S6K,BIX 02565,inhibit
产品简介:bix 02565 is a potent inhibitor of ribosomal s6 kinase 2 (rsk2, ic50: 1.1 nm)...产品型号:T5428 原产地:中国大陆价格: ¥0.0
产品名称: SincalidePI3K/Akt,cardiovascular hormone,Inhibitor,SQ 19844,PI3K,Akt,Protein kinase B,Apoptosis,SQ-1
产品简介:sincalide (inn) is a cholecystokinetic drug administered by injection to aid in diagnosing disorders of the gallbladder and pancreas. it is the 8-amino acid c-t..产品型号:TP1197 原产地:中国大陆价格: ¥0.0
产品名称: VTX-27Inhibitor,VTX27,VTX 27,PKC,Protein kinase C,inhibit,VTX-27
产品简介:vtx-27 is a selective inhibitor of protein kinase c θ (pkc θ) (kis: 0.08 nm and 16 nm for pkc θ and pkc δ)...产品型号:T13314 原产地:中国大陆价格: ¥0.0
产品名称: NarciclasineRho-associated kinase,ROCK,inhibit,Inhibitor,ROK,Narciclasine,Rho-associated protein kin
产品简介:narciclasine, a natural product, modulates the rho/rho-kinase/lim kinase/cofilin signaling pathway, greatly increasing gtpase rhoa activity...产品型号:TQ0183 原产地:中国大陆价格: ¥0.0
产品名称: Batatasin IIIFocal adhesion kinase,Batatasin III,Inhibitor,inhibit,PTK2 protein tyrosine kinase 2,PK
产品简介:batatasin iii inhibits cancer migration and invasion by suppressing epithelial to mesenchymal transition and fak-akt signals and possesses anti-cancer activitie..产品型号:TN1433 原产地:中国大陆价格: ¥0.0
产品名称: Tyrphostin AG1296Fms like tyrosine kinase 3,PDGF,Apoptosis,CD117,inhibit,platelet-derived,CD135,SCFR
产品简介:tyrphostin ag 1296 is an inhibitor of pdgfr with ic50 of 0.3-0.5 μm, no activity to egfr...产品型号:T6711 原产地:中国大陆价格: ¥0.0
产品名称: Thymidylate Kinase Inhibitor, YMU1YMU 1,inhibit,YMU-1,YMU1,Thymidylate Kinase Inhibitor, YMU1,Inhibi
产品简介:ymu1 is a human thymidylate kinase (htmpk) inhibitor. ymu1 stabilizes the conformation of ligand-induced degradation (lid) region of htmpk and blocks the cataly..产品型号:T8864 原产地:中国大陆价格: ¥0.0
产品名称: ASK1-IN-2colitis,ulcerative,signal-regulating,ASK1 IN 2,ASK1IN2,inhibit,MAP kinase kinase kinase, ME
产品简介:ask1-in-2 is a potent and orally active inhibitor of apoptosis signal-regulating kinase 1 (ask1), with an ic50 of 32.8 nm. ask1-in-2 can potentially be used as ..产品型号:T9377 原产地:中国大陆价格: ¥0.0
产品名称: CGP 57380CGP-57380,CGP 57380,Mitogen activated protein kinase interacting kinase,Inhibitor,MAPK inte
产品简介:cgp 57380 is a potent mnk1 inhibitor with ic50 of 2.2 μm, exhibiting no inhibitory activity on p38, jnk1, erk1 and -2, pkc, or c-src-like kinases...产品型号:T6440 原产地:中国大陆价格: ¥0.0
产品名称: ROCK-IN-2inhibit,Rho-kinase,Rho-associated protein kinase,Azaindole-1,ROCKIN2,Rho-associated kinase,
产品简介:azaindole 1 is a selective and atp-competitive rock inhibitor with ic50 of 0.6 and 1.1 nm for human rock-1 and rock-2...产品型号:TQ0110 原产地:中国大陆价格: ¥0.0
产品名称: GNE-493GNE493,Mammalian target of Rapamycin,PI3K,Inhibitor,inhibit,GNE-493,Phosphoinositide 3-kinase
产品简介:gne-493 is potent, selective, and orally available pi3k and mtor inhibitor with potential anticancer activity.ic50s of 3.4 nm, 12 nm, 16 nm, 16 nm and 32 nm for..产品型号:T7166 原产地:中国大陆价格: ¥0.0
产品名称: 4SC-203tumor,antineoplastic,Fms like tyrosine kinase 3,Vascular endothelial growth factor receptor,4
产品简介:4sc-203 is a multikinase inhibitor with potential antineoplastic activity. 4sc-203 selectively inhibits fms-related tyrosine kinase 3 (flt3/stk1), flt3 mutated ..产品型号:T9473 原产地:中国大陆价格: ¥0.0
产品名称: TL-895anti-viral,TL-895,Inhibitor,Bruton tyrosine kinase,TL895,Myelofibrosis,Solid Tumor,Carcinoma,A
产品简介:tl-895 is an atp-competitive, and highly selective irreversible inhibitor of bruton’s tyrosine kinase(btk). tl-895 showed good potency with an ic50 of 1.5 nm an..产品型号:T9705 原产地:中国大陆价格: ¥0.0
产品名称: GSK-1070916Inhibitor,Aurora Kinase,GSK-1070916,GSK 1070916,Apoptosis,inhibit
产品简介:gsk1070916 is a reversible and atp-competitive inhibitor of aurora b/c with ic50 of 3.5 nm/6.5 nm. it displays >100-fold selectivity against the closely related..产品型号:T6129 原产地:中国大陆价格: ¥0.0
产品名称: Abrocitinibinhibit,Abrocitinib,Inhibitor,JAK,PF04965842,Janus kinase,PF 04965842
产品简介:abrocitinib (pf-04965842) is a potent, specific and orally-active jak1 inhibitor (ic50s: 29/803 nm for jak1/2)...产品型号:TQ0037 原产地:中国大陆价格: ¥0.0
产品名称: ARN-3236inhibit,ARN3236,Salt-inducible Kinase (SIK),ARN-3236,ARN 3236,Inhibitor
产品简介:arn-3236 is an oral active and selective inhibitor of salt-inducible kinase 2 (sik2), (sik2, sik1 and sik3 with ic50s of <1 nm, 21.63 nm and 6.63 nm respectivel..产品型号:T5993 原产地:中国大陆价格: ¥0.0
产品名称: Ro 5126766MAPKK,CH 5126766,MEK,Ro 5126766,Raf kinases,Raf,Mitogen-activated protein kinase kinase,in
产品简介:ro5126766 (ch5126766) is a dual raf/mek inhibitor with ic50 of 8.2 nm, 19 nm, 56 nm, and 160 nm for braf v600e, braf, craf, and mek1, respectively. phase 1...产品型号:T6971 原产地:中国大陆价格: ¥0.0