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产品目录

产品展示/Products

  • STING agonist-11;化合物 STING agonist-11STING agonist-11

    产品名称: STING agonist-11;化合物 STING agonist-11STING agonist-11

    产品简介:sting agonist-11 is a potent activator of the small molecule cyclic urea class of sting (ec50: 18 nm).sting activation is a highly promising immunotherapy...

    产品型号:T63458 原产地:中国大陆价格: ¥0.0

  • Tubulin polymerization-IN-4;化合物 Tubulin polymerization-IN-4Tubulin polymerization-IN-4

    产品名称: Tubulin polymerization-IN-4;化合物 Tubulin polymerization-IN-4Tubulin polymerization-IN-4

    产品简介:tubulin polymerization-in-4 is an effective inhibitor of tubulin polymerization (ic50=4.6 μm)。 tubulin polymerization-in-4 can destroy tubulin polymerization, b..

    产品型号:T61940 原产地:中国大陆价格: ¥0.0

  • Telatinib mesylate;化合物 Telatinib mesylateTelatinib mesylate

    产品名称: Telatinib mesylate;化合物 Telatinib mesylateTelatinib mesylate

    产品简介:telatinib mesylate is a potent, orally active inhibitor of vegfr2 (ic50: 6 nm), vegfr3 (ic50: 4 nm), pdgfα (ic50: 15 nm) and c-kit (ic50: 1 nm)...

    产品型号:T63459 原产地:中国大陆价格: ¥0.0

  • WYE-132;化合物WYE-125132WYE 125132|||WYE125132|||WYE-125132;WYE 125132|||WYE125132|||WYE-125132

    产品名称: WYE-132;化合物WYE-125132WYE 125132|||WYE125132|||WYE-125132;WYE 125132|||WYE125132|||WYE-125132

    产品简介:wye-125132 (wye-132 (wye-125132)) is a highly potent, atp-competitive mtor inhibitor with ic50 of 0.19 nm; highly selective for mtor versus pi3ks or pi3k-relate..

    产品型号:T6346 原产地:中国大陆价格: ¥0.0

  • SIRT5 inhibitor 3;化合物 SIRT5 inhibitor 3SIRT5 inhibitor 3

    产品名称: SIRT5 inhibitor 3;化合物 SIRT5 inhibitor 3SIRT5 inhibitor 3

    产品简介:sirt5 inhibitor 3 (compound 46) is an effective and competitive sirt5 inhibitor (ic50=5.9 μ m). sirt5 inhibitor 3 shows inhibitory effect on the deacetylation o..

    产品型号:T61947 原产地:中国大陆价格: ¥0.0

  • Tropesin;化合物 TropesinTropesin

    产品名称: Tropesin;化合物 TropesinTropesin

    产品简介:tropesin is a non-steroidal anti-inflammatory agent (nsaia) that has inhibitory effects on the growth of xylaria green...

    产品型号:T63460 原产地:中国大陆价格: ¥0.0

  • INSCoV-600K(1);化合物 INSCoV-600K(1)INSCoV-600K(1)

    产品名称: INSCoV-600K(1);化合物 INSCoV-600K(1)INSCoV-600K(1)

    产品简介:inscov-600k(1) is a potent mpro(3clpro) inhibitor. proteases (plpro and 3clpro) are associated with viral transcription and replication. inscov-600k(1) has show..

    产品型号:T63461 原产地:中国大陆价格: ¥0.0

  • MraY-IN-2;化合物 MraY-IN-2MraY-IN-2

    产品名称: MraY-IN-2;化合物 MraY-IN-2MraY-IN-2

    产品简介:mray-in-2 (compound 6) is an effective inhibitor of bacterial transposase mray (ic50=4.5 μ m), and can be used for antibacterial research...

    产品型号:T61948 原产地:中国大陆价格: ¥0.0

  • INSCoV-601I(1);化合物 INSCoV-601I(1)INSCoV-601I(1)

    产品名称: INSCoV-601I(1);化合物 INSCoV-601I(1)INSCoV-601I(1)

    产品简介:inscov-601i(1) is a potent mpro(3clpro) inhibitor. proteases (plpro and 3clpro) are associated with viral transcription and replication. inscov-600i(1) has show..

    产品型号:T63462 原产地:中国大陆价格: ¥0.0

  • ERCC1-XPF-IN-1;化合物 ERCC1-XPF-IN-1ERCC1-XPF-IN-1

    产品名称: ERCC1-XPF-IN-1;化合物 ERCC1-XPF-IN-1ERCC1-XPF-IN-1

    产品简介:ercc1-xpf-in-1 is a potent, high-affinity inhibitor of ercc1-xpf (ic50: 0.49 μm). ercc1-xpf-in-1 inhibits the removal of cpds, reduces the toxicity of cyclophos..

    产品型号:T63464 原产地:中国大陆价格: ¥0.0

  • hCAII-IN-5;化合物 hCAII-IN-5hCAII-IN-5

    产品名称: hCAII-IN-5;化合物 hCAII-IN-5hCAII-IN-5

    产品简介:hcaii-in-5 (compound 12h) is a potent, selective inhibitor of human carbonic anhydrase ii (hca ii) with an inhibition constant (ic50) of 4.55 ?m [1]...

    产品型号:T63467 原产地:中国大陆价格: ¥0.0

  • RET-IN-14;化合物 RET-IN-14RET-IN-14

    产品名称: RET-IN-14;化合物 RET-IN-14RET-IN-14

    产品简介:ret-in-14 is a potent inhibitor of ret, capable of acting on ret (wt) (ic50 < 0.51 nm), ret (g810r) (ic50: 9.3 nm), ret (v804m) (ic50: 1.3 nm), btk (c481s) (ic5..

    产品型号:T63468 原产地:中国大陆价格: ¥0.0

  • UIAA-II-232;化合物 UIAA-II-232UIAA-II-232

    产品名称: UIAA-II-232;化合物 UIAA-II-232UIAA-II-232

    产品简介:uiaa-ii-232 (compound 19b) is a potent inhibitor of dna gyrase catalytic (ic 50= 3.5 μm)...

    产品型号:T61950 原产地:中国大陆价格: ¥0.0

  • RIPK1-IN-8;化合物 RIPK1-IN-8RIPK1-IN-8

    产品名称: RIPK1-IN-8;化合物 RIPK1-IN-8RIPK1-IN-8

    产品简介:ripk1-in-8 is an aminoimidazolopyridine and is a selective and potent inhibitor of ripk1 (ic50: 4 nm).ripk1-in-8 has research potential in inflammatory diseases..

    产品型号:T63469 原产地:中国大陆价格: ¥0.0

  • Ki16198;化合物Ki16198Ki16198

    产品名称: Ki16198;化合物Ki16198Ki16198

    产品简介:ki16198 is the methyl ester of ki16425, which is a lpa antagonist and inhibits lpa1- and lpa3-induced inositol phosphate production with ki of 0.34 μm and 0.93 ..

    产品型号:T6347 原产地:中国大陆价格: ¥0.0

  • Mazaticol;化合物 MazaticolMazaticol

    产品名称: Mazaticol;化合物 MazaticolMazaticol

    产品简介:mazaticol is an anticholinergic agent, which blocks the muscarinic acetylcholine receptors and cholinergic nerve activity. mazaticol potently inhibits 3h-qnb an..

    产品型号:T62008 原产地:中国大陆价格: ¥0.0

  • PI3K/mTOR Inhibitor-8;化合物 PI3K/mTOR Inhibitor-8PI3K/mTOR Inhibitor-8

    产品名称: PI3K/mTOR Inhibitor-8;化合物 PI3K/mTOR Inhibitor-8PI3K/mTOR Inhibitor-8

    产品简介:pi3k/mtor inhibitor-8 is a dual inhibitor of pi3k (pi3kα ic50: 0.46 nm) and mtor (mtor ic50: 12 nm). pi3k/mtor inhibitor-8 blocks the cell cycle of hct-116 cell..

    产品型号:T63470 原产地:中国大陆价格: ¥0.0

  • PARP1/BRD4-IN-1;化合物 PARP1/BRD4-IN-1PARP1/BRD4-IN-1

    产品名称: PARP1/BRD4-IN-1;化合物 PARP1/BRD4-IN-1PARP1/BRD4-IN-1

    产品简介:parp1/brd4-in-1 is a highly selective and potent inhibitor of parp1 (ic50: 49 nm) and brd4 (ic50: 202 nm).parp1/brd4-in-1 inhibits the expression and activity o..

    产品型号:T63471 原产地:中国大陆价格: ¥0.0

  • 2α,3β,24-Trihydroxyurs-12-en-28-oic acid;化合物 2α,3β,24-Trihydroxyurs-12-en-28-oic acid2,24-Dihydroxyu

    产品名称: 2α,3β,24-Trihydroxyurs-12-en-28-oic acid;化合物 2α,3β,24-Trihydroxyurs-12-en-28-oic acid2,24-Dihydroxyu

    产品简介:2α,3β,24-trihydroxyurs-12-en-28-oic acid, a natural product, is isolated from salvia palaestina [1]...

    产品型号:T83373 原产地:中国大陆价格: ¥0.0

  • HDAC6-IN-4;化合物 HDAC6-IN-4HDAC6-IN-4

    产品名称: HDAC6-IN-4;化合物 HDAC6-IN-4HDAC6-IN-4

    产品简介:hdac6-in-4 (c10) is an orally active, highly selective, potent and non-significantly toxic hdac6 inhibitor (ic50: 23 nm). hdac6-in-4 induces apoptosis and exhib..

    产品型号:T63472 原产地:中国大陆价格: ¥0.0

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