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产品名称: Top/HDAC-IN-1;化合物 Top/HDAC-IN-1Top/HDAC-IN-1
产品简介:top/hdac-in-1 is a dual topoisomerase (top)/hdac inhibitor that acts on hdac1 (ic50: 18 nm), hdac2 (ic50: 230 nm), hdac3 (ic50: 790 nm), hdac6 (ic50: 87 nm) and..产品型号:T63509 原产地:中国大陆价格: ¥0.0
产品名称: MGCD-265 analog;化合物MGCD-265 analogMGCD-265|||Glesatinib;MGCD-265|||Glesatinib
产品简介:mgcd-265 analog (glesatinib) is an orally bioavailable multitargeted tyrosine kinase inhibitor with potential antineoplastic activity with ic50 of 29 nm and 10 ..产品型号:T6351 原产地:中国大陆价格: ¥0.0
产品名称: ATX inhibitor 21;化合物 ATX inhibitor 21ATX inhibitor 21
产品简介:atx inhibitor 21 is a potent inhibitor of atx (ic50: 3490 nm)...产品型号:T63510 原产地:中国大陆价格: ¥0.0
产品名称: IRE1α kinase-IN-4;化合物 IRE1α kinase-IN-4IRE1α kinase-IN-4
产品简介:ire1α kinase-in-4 (compound 6) is a potent inhibitor of ire1α, exhibiting a ki value of 140 nm. it acts as an atp-competitive ligand for ire1α [1]...产品型号:T63511 原产地:中国大陆价格: ¥0.0
产品名称: LpxC-IN-10;化合物 LpxC-IN-10LpxC-IN-10
产品简介:lpxc-in-10 is a selective lpxc inhibitor with an mic of 0.5 μg/ml against e. coli and k. pneumoniae and is capable of being used to study bacterial infections...产品型号:T63512 原产地:中国大陆价格: ¥0.0
产品名称: Antitumor agent-71;化合物 Antitumor agent-71Antitumor agent-71
产品简介:antitumor agent-71 is an antitumor compound that exhibits an inhibitory effect on tubulin aggregation. antitumor agent-71 possesses an anti-proliferative effect..产品型号:T63513 原产地:中国大陆价格: ¥0.0
产品名称: PPARγ agonist 1;化合物 PPARγ agonist 1PPARγ agonist 1
产品简介:pparγ agonist 1 is a potent agonist of pparγ that efficiently activates hpparγ without causing full agonism, thereby avoiding adverse effects. pparγ agonist 1 h..产品型号:T63514 原产地:中国大陆价格: ¥0.0
产品名称: THR-β agonist 4;化合物 THR-β agonist 4THR-β agonist 4
产品简介:thr-β agonist 4 is a potent agonist of thr-β. thr-β agonist 4 has shown research potential for metabolic diseases such as hyperlipidemia, obesity, hypercholeste..产品型号:T63515 原产地:中国大陆价格: ¥0.0
产品名称: NRX-252114;化合物NRX-252114NRX252114|||NRX 252114;NRX252114|||NRX 252114
产品简介:nrx-252114 (nrx252114) induces degradation of mutant β-catenin nrx-252114 is a potent enhancer of the interaction of β-catenin with the homologous e3 ligase scf..产品型号:T63516 原产地:中国大陆价格: ¥0.0
产品名称: BuChE-IN-4;化合物 BuChE-IN-4BuChE-IN-4
产品简介:buche-in-4 is a potent inhibitor of buche (ic50: 7.7 nm) and exhibits mild antioxidant capacity, non-toxicity, lipophilicity and neuroprotective effects...产品型号:T63517 原产地:中国大陆价格: ¥0.0
产品名称: CCG-273463;化合物 CCG-273463CCG-273463
产品简介:ccg-273463 is a potent, covalent, selective inhibitor of grk5 (ic50: 9 nm). ccg-273463 can be used to study heart failure, hypertrophic cardiomyopathy and cance..产品型号:T63640 原产地:中国大陆价格: ¥0.0
产品名称: (3S,4R)-PF-6683324;化合物 (3S,4R)-PF-6683324(3S,4R)-PF-6683324
产品简介:(3s,4r)-pf-6683324 is a pro-myosin-related kinase (trk) inhibitor that has shown research potential for pain and cancer...产品型号:T63641 原产地:中国大陆价格: ¥0.0
产品名称: CQ211;化合物CQ211CQ211
产品简介:cq211 is a potent and selective riok2 inhibitor with a kd of 6.1 nm.cq211 has shown potent proliferation inhibitory activity against various cancer cell lines i..产品型号:T63642 原产地:中国大陆价格: ¥0.0
产品名称: BI-4142;化合物BI-4142BI-4142
产品简介:bi-4142 is an orally active, potent and selective her2 inhibitor that inhibits cancer cell proliferation, suppresses her2-dependent cell lines and inhibits down..产品型号:T63643 原产地:中国大陆价格: ¥0.0
产品名称: ONO-9780307;化合物 ONO-9780307ONO-9780307
产品简介:ono-9780307 is a specific antagonist of lpa1 (lysophosphatidic acid receptor 1) (ic50: 2.7 nm)...产品型号:T63645 原产地:中国大陆价格: ¥0.0
产品名称: COX-2-IN-9;化合物 COX-2-IN-9COX-2-IN-9
产品简介:cox-2-in-9 is a selective, potent, orally active cox-2 inhibitor (ic50: 10.17 μm).cox-2-in-9 has a higher cox-2 selectivity than celecoxib.cox-2-in-9 exhibits g..产品型号:T63646 原产地:中国大陆价格: ¥0.0
产品名称: DCN1-UBC12-IN-1;化合物 DCN1-UBC12-IN-1DCN1-UBC12-IN-1
产品简介:dcn1-ubc12-in-1 is a potent and specific dcn1-ubc12 inhibitor with an ic50 value of 2.86 nm and anti-cardiac fibrogenic activity...产品型号:T63647 原产地:中国大陆价格: ¥0.0
产品名称: EGFR kinase inhibitor 1;化合物 EGFR kinase inhibitor 1EGFR kinase inhibitor 1
产品简介:egfr kinase inhibitor 1 is a potent inhibitor of egfr that acts on wt (ic50: 37 nm), l885r/t790m (ic50: 1.7 nm), and l858r/t790m/c797s (ic50>300 nm). egfr kinas..产品型号:T63648 原产地:中国大陆价格: ¥0.0
产品名称: Ned-K;化合物 Ned-KNed-K
产品简介:ned-k is a nicotinic acid adenine dinucleotide phosphate (naadp) antagonist that exhibits an inhibitory effect on myocardial ischemia and reperfusion (sir)-indu..产品型号:T63649 原产地:中国大陆价格: ¥0.0
产品名称: Desfesoterodine fumarate;化合物 T6364LPNU-200577 fumarate|||UNII-607O3D83YQ;PNU-200577 fumarate|||UNII-
产品简介:desfesoterodine fumarate is a bio-active chemical. detailed information has not been published...产品型号:T6364L 原产地:中国大陆价格: ¥0.0