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产品名称: A2A/A1 AR antagonist-1;化合物 A2A/A1?AR antagonist-1A2A/A1 AR antagonist-1
产品简介:a2a/a1 ar antagonist-1 (compound 1a) has the potential for ischemic stroke research which is potent a 2a /a 1 ar dual antagonist with ki s of 5.58 and 24.2 nm, ..产品型号:T60732 原产地:中国大陆价格: ¥0.0
产品名称: MNK1/2-IN-5;化合物 MNK1/2-IN-5MNK1/2-IN-5
产品简介:mnk1/2-in-5 is a potent and selective inhibitor of mnk1/2...产品型号:T60733 原产地:中国大陆价格: ¥0.0
产品名称: HIV-1 integrase inhibitor 8;HIV-1整合酶抑制剂8HIV-1 integrase inhibitor 8
产品简介:hiv-1 integrase inhibitor 8 is an inhibitor of hiv-1 integrase. integration is a required step in hiv replication [1]...产品型号:T60742 原产地:中国大陆价格: ¥0.0
产品名称: HbF inducer-1;化合物 HbF inducer-1HbF inducer-1
产品简介:hbf inducer-1 is a fetal hemoglobin inducer which is orally bioavailable...产品型号:T60898 原产地:中国大陆价格: ¥0.0
产品名称: ERCC1-XPF-IN-2;化合物ERCC1-XPF-IN-2ERCC1-XPF-IN-2
产品简介:ercc1-xpf-in-2 is active in nucleotide excision repair, cisplatin enhancement and γh2ax assays. ercc1-xpf-in-2 is a potent inhibitor of ercc1-xpf endonuclease w..产品型号:T60904 原产地:中国大陆价格: ¥0.0
产品名称: SARM1-IN-2;SARM1抑制剂2SARM1-IN-2
产品简介:sarm1-in-2 is a potent sarm1 inhibitor for the study of metabolic and neurological related diseases...产品型号:T60908 原产地:中国大陆价格: ¥0.0
产品名称: A1AR antagonist 5;化合物 A1AR antagonist 5A1AR antagonist 5
产品简介:a1ar antagonist 5 (compound 20) is a potent and selective antagonist of a1 adenosine receptor (a1ar) with a pki of 6.11 and a pic 50 of 5.83 [1]...产品型号:T60915 原产地:中国大陆价格: ¥0.0
产品名称: Dopamine D4 receptor antagonist-1;化合物 Dopamine D4 receptor antagonist-1Dopamine D4 receptor antagoni
产品简介:dopamine d4 receptor antagonist-1 can be used in schizophrenia study. dopamine d4 receptor antagonist-1 is a selective antagonist of dopamine d4 receptor (drd4)..产品型号:T60917 原产地:中国大陆价格: ¥0.0
产品名称: RSK-IN-1;化合物 RSK-IN-1RSK-IN-1
产品简介:rsk-in-1 (compound 7d) shows anti-tumor activity. rsk-in-1 is an inhibitor of rsk that inhibits the phosphorylation of yb-1 [1]...产品型号:T60922 原产地:中国大陆价格: ¥0.0
产品名称: PknB-IN-1;化合物 PknB-IN-1PknB-IN-1
产品简介:pknb-in-1 (compound 2) is an inhibitor of protein kinase b (pknb) with a concentration causing 50% inhibition (ic50) of 14.4 μm. this compound demonstrates anti..产品型号:T61772 原产地:中国大陆价格: ¥0.0
产品名称: Keap1-Nrf2-IN-4;化合物 Keap1-Nrf2-IN-4Keap1-Nrf2-IN-4
产品简介:keap1-nrf2-in-4, a powerful neddylation inhibitor, demonstrates significant anti-proliferation activity against mgc-803 cells (ic50 = 2.55 μm), effectively impe..产品型号:T61773 原产地:中国大陆价格: ¥0.0
产品名称: SARS 3CLpro-IN-1;化合物 SARS 3CLpro-IN-1SARS 3CLpro-IN-1
产品简介:sars 3clpro-in-1 (compound 3b) is a stereo-specific sars 3cl protease inhibitor that belongs to the octahydroisochromene scaffold. it demonstrates inhibition ag..产品型号:T61774 原产地:中国大陆价格: ¥0.0
产品名称: mGlu4 receptor agonist 1;化合物 mGlu4 receptor agonist 1mGlu4 receptor agonist 1
产品简介:mglu4 receptor agonist 1 (compound 62) is a highly effective positive allosteric modulator of mglu4 receptors, displaying an ec 50 of 308 nm. additionally, it e..产品型号:T61775 原产地:中国大陆价格: ¥0.0
产品名称: NPP1-IN-1;化合物 NPP1-IN-1NPP1-IN-1
产品简介:npp1-in-1 is a highly potent inhibitor of npp enzymes, effectively inhibiting npp1 with an ic 50 value of 0.15 μm and npp3 with an ic 50 value of 40 μm [1]...产品型号:T61782 原产地:中国大陆价格: ¥0.0
产品名称: Antimicrobial agent-1;化合物 Antimicrobial agent-1Antimicrobial agent-1
产品简介:antimicrobial agent-1 (compound 6c) shows strong activity (mic = 2 μg/ml) against tolc mutant e. coli. additionally, it synergistically interacts with colistin ..产品型号:T61783 原产地:中国大陆价格: ¥0.0
产品名称: GlcN-6-P Synthase-IN-1;化合物 GlcN-6-P Synthase-IN-1GlcN-6-P Synthase-IN-1
产品简介:glcn-6-p synthase-in-1 (compound 4d) is a potent inhibitor of glucosamine-6-phosphate (glcn-6-p) synthase, with an ic50 of 3.47 μm. this compound demonstrates r..产品型号:T61784 原产地:中国大陆价格: ¥0.0
产品名称: TRPV1 antagonist 3;化合物 TRPV1 antagonist 3TRPV1 antagonist 3
产品简介:trpv1 antagonist 3 (compound 7q) is a highly potent antagonist of the trpv1 receptor with an ic50 of 2.66 nm against capsaicin. it exhibits selectivity towards ..产品型号:T61788 原产地:中国大陆价格: ¥0.0
产品名称: IDO1-IN-14;化合物 IDO1-IN-14IDO1-IN-14
产品简介:ido1-in-14 (compound 4a) is a highly effective inhibitor of the ido1 enzyme, exhibiting an ic50 value of 396.9 nm. additionally, ido1-in-14 demonstrates excelle..产品型号:T61789 原产地:中国大陆价格: ¥0.0
产品名称: BRD4-BD1/2-IN-1;化合物 BRD4-BD1/2-IN-1BRD4-BD1/2-IN-1
产品简介:brd4-bd1/2-in-1 is a highly effective inhibitor of brd4, specifically targeting the brd4 bd-1 and brd4 bd-2 domains with ic 50 values of <100 nm each (us2015014..产品型号:T61791 原产地:中国大陆价格: ¥0.0
产品名称: hCAIX/XII-IN-1;化合物 hCAIX/XII-IN-1hCAIX/XII-IN-1
产品简介:hcaix/xii-in-1, a potent inhibitor of both caix and caxii, exhibits ki values of 0.48 μm for caix and 0.83 μm for caxii, respectively. this compound demonstrate..产品型号:T61873 原产地:中国大陆价格: ¥0.0