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产品名称: AKR1C3-IN-6;化合物 AKR1C3-IN-6AKR1C3-IN-6
产品简介:akr1c3-in-6 (compound 1) is a powerful and specific inhibitor of akr1c3, with ic50 values of 0.31 μm and 73.23 μm against akr1c3 and akr1c2, respectively. it de..产品型号:T61790 原产地:中国大陆价格: ¥0.0
产品名称: PARP1-IN-7;化合物 PARP1-IN-7PARP1-IN-7
产品简介:parp1-in-7 functions as an anticancer agent by inhibiting poly(adp-ribose) polymerase-1 (parp1)...产品型号:T61879 原产地:中国大陆价格: ¥0.0
产品名称: RIPK1-IN-13;化合物 RIPK1-IN-13RIPK1-IN-13
产品简介:ripk1-in-13 (compound 8) is an effective ripk1 inhibitor (ic50=1139 nm). by inhibiting ripk1, ripk1-in-13 can block the activation of necrotic apoptosis pathway..产品型号:T61887 原产地:中国大陆价格: ¥0.0
产品名称: mTOR/HDAC6-IN-1;化合物 mTOR/HDAC6-IN-1mTOR/HDAC6-IN-1
产品简介:mtor/hdac6-in-1 is an effective dual inhibitor of histone deacetylase (hdac6) and mammalian rapamycin (mtor). the ic50 values for hdac6 and mtor are 56 nm and 1..产品型号:T61888 原产地:中国大陆价格: ¥0.0
产品名称: CSF1R-IN-12;化合物 CSF1R-IN-12CSF1R-IN-12
产品简介:csf1r-in-12 is an effective csf1r inhibitor. csf1r-in-12 has research potential in cancer diseases...产品型号:T61893 原产地:中国大陆价格: ¥0.0
产品名称: SMO-IN-1;化合物 SMO-IN-1SMO-IN-1
产品简介:smo-in-1 (compound 15) is an oral effective smoothened (smo) inhibitor. the ec50 value of sonic hh protein (shh) is 89 nm...产品型号:T61897 原产地:中国大陆价格: ¥0.0
产品名称: VEGFR2-IN-1;VEGFR2 抑制剂1VEGFR2-IN-1
产品简介:vegfr2-in-1 is a selective and potent vegfr2 inhibitor with antitumor activity that inhibits cell proliferation and migration and can be used in the study of br..产品型号:T61899 原产地:中国大陆价格: ¥0.0
产品名称: 5-HT6/5-HT2AR antagonist-1;化合物 5-HT6/5-HT2AR antagonist-15-HT6/5-HT2AR antagonist-1
产品简介:5-ht6/5-ht2ar antagonist-1 is a powerful and effective compound that acts as a dual antagonist for both the 5-ht6 and 5-ht2a receptors. it exhibits high potency..产品型号:T61837 原产地:中国大陆价格: ¥0.0
产品名称: SCD1-IN-1;化合物 SCD1-IN-1SCD1-IN-1
产品简介:scd1-in-1, a potent inhibitor of scd1 (ic50: 5.8 nm), is valuable in dermatologic research [1]...产品型号:T61841 原产地:中国大陆价格: ¥0.0
产品名称: HIV-1 inhibitor-9;化合物 HIV-1 inhibitor-9HIV-1 inhibitor-9
产品简介:hiv-1 inhibitor-9 exhibits potent inhibition activity at low nanomolar concentrations against both the wild-type (wt) hiv-1 strain and multiple strains that hav..产品型号:T61844 原产地:中国大陆价格: ¥0.0
产品名称: Nrf2-ARE/hMAO-B/QR2 modulator 1;化合物 Nrf2-ARE/hMAO-B/QR2 modulator 1Nrf2-ARE/hMAO-B/QR2 modulator 1
产品简介:nrf2-are/hmao-b/qr2 modulator 1 is a new resveratrol-based multitarget-directed ligands (mtdls) that showed a well-balanced mtdl profile: cellular activation of..产品型号:T60395 原产地:中国大陆价格: ¥0.0
产品名称: ART-IN-1;化合物 ART-IN-1ART-IN-1
产品简介:art-in-1 (compound 7) is a selective inhibitor of parp with ic 50 s of 19, 22, 2.4, >100, 1.1 μm for parp2, tnks2, parp10, parp14, parp15, respectively [1]...产品型号:T60410 原产地:中国大陆价格: ¥0.0
产品名称: Adenosine receptor inhibitor 1;化合物 Adenosine receptor inhibitor 1Adenosine receptor inhibitor 1
产品简介:adenosine receptor inhibitor 1 is a highly potent and selective antagonist of adenosine receptor (ar). it exhibits exceptional affinity for a1 ar, a2a ar, a2b a..产品型号:T61850 原产地:中国大陆价格: ¥0.0
产品名称: PTP1B-IN-3 diammonium;化合物 PTP1B-IN-3 diammoniumPTP1B-IN-3 diammonium
产品简介:ptp1b-in-3 diammonium is a highly effective and orally bioavailable inhibitor of the protein tyrosine phosphatase 1b (ptp1b) enzyme, with an ic50 value of 120 n..产品型号:T61851 原产地:中国大陆价格: ¥0.0
产品名称: Antimycobacterial agent-1;化合物 Antimycobacterial agent-1Antimycobacterial agent-1
产品简介:antimycobacterial agent-1 (compound 33) demonstrates potent antimycobacterial activity against mycobacterium tuberculosis h37ra, with a minimal inhibitory conce..产品型号:T61853 原产地:中国大陆价格: ¥0.0
产品名称: Antistaphylococcal agent 1;化合物 Antistaphylococcal agent 1Antistaphylococcal agent 1
产品简介:antistaphylococcal agent 1 is an antistaphylococcal therapeutic agent...产品型号:T61855 原产地:中国大陆价格: ¥0.0
产品名称: HIF-1α-IN-5;化合物 HIF-1α-IN-5HIF-1α-IN-5
产品简介:hif-1α-in-5 is an inhibitor of hif-1α with an ic 50 value of 24 nm in hek293t cells that also inhibits the activity of mao-a. hif-1α-in-5 downregulates the mrna..产品型号:T60532 原产地:中国大陆价格: ¥0.0
产品名称: TRAP-6-IN-1;化合物 TRAP-6-IN-1TRAP-6-IN-1
产品简介:trap-6-in-1 (compound 8) is a dual inhibitor of collagen and trap-6 with ic 50 values of 17.12 μm and 11.88 μm, respectively. trap-6-in-1 non-competitively inh..产品型号:T60557 原产地:中国大陆价格: ¥0.0
产品名称: Enpp-1-IN-9;化合物 Enpp-1-IN-9Enpp-1-IN-9
产品简介:enpp-1-in-9, a powerful inhibitor of ectonucleotide pyrophosphatase-phosphodiesterase 1 (enpp1), exhibits wide substrate specificity, capable of cleaving variou..产品型号:T61860 原产地:中国大陆价格: ¥0.0
产品名称: Quorum Sensing-IN-1;化合物 Quorum Sensing-IN-1Quorum Sensing-IN-1
产品简介:quorum sensing-in-1 is a small-molecule inhibitor of quorum sensing...产品型号:T60595 原产地:中国大陆价格: ¥0.0