联系我们
产品目录
产品展示/Products
产品名称: N6-(2-Phenylethyl)adenosineP1 receptor,A1AR,derivative,N-6-(2-Phenylethyl)adenosine,Adenosine Recept
产品简介:n6-(2-phenylethyl)adenosine is an adenosine derivative and an agonist of adenosine receptors with ki values of 11.8 nm and 30.1 nm for rat and human a1...产品型号:T12163 原产地:中国大陆价格: ¥0.0
产品名称: Rotundine5-hydroxytryptamine Receptor,Inhibitor,Dopamine Receptor,Rotundine,5-HT Receptor,inhibit,Se
产品简介:rotundine (l-tetrahydropalmatine, l-thp) is a selective dopamine d1 receptor antagonist with ic50 of 166 nm...产品型号:T6648 原产地:中国大陆价格: ¥0.0
产品名称: NSC 228155Epidermal growth factor receptor,Histone Acetyltransferase,EGFR,HER1,HATs,inhibit,Inhibito
产品简介:nsc228155 is an activator of egfr, binding to the segfr dimerization domain ii and modulate egfr tyrosine phosphorylation...产品型号:T6908 原产地:中国大陆价格: ¥0.0
产品名称: RS102895CC chemokine receptor,CCR,Inhibitor,RS102895,inhibit,RS-102895,RS 102895
产品简介:rs102895 is a potent ccr2 antagonist (ic50: 360 nm) and shows no effect on ccr1...产品型号:TQ0283 原产地:中国大陆价格: ¥0.0
产品名称: Practololreceptor,inhibit,arrhythmias,β1-adrenergic,Practolol,Beta Receptor,Adrenergic Receptor,card
产品简介:practolol is a selective β-adrenoceptor blocker...产品型号:T8595 原产地:中国大陆价格: ¥0.0
产品名称: PRN1371inhibit,CSF1R,PRN 1371,Inhibitor,colony stimulating factor 1 receptor,c-Fms,CSF-1R,FGFR,CSF-1
产品简介:prn1371 is a specific and potent fgfr1-4 and csf1r inhibitor (ic50s: 0.6/1.3/4.1/19.3/8.1 nm for fgfr1/2/3/4 and csf1r)...产品型号:TQ0015 原产地:中国大陆价格: ¥0.0
产品名称: HS024selective,melanocortin,intake,Inhibitor,Melanocortin Receptor,MC Receptor,HS-024,food,HS024,inh
产品简介:highly potent melanocortin mc4 receptor antagonist (ki values are 0.29, 18.6, 5.45 and 3.29 nm for cloned human mc4, mc1, mc3 and mc5 receptors respectively). i..产品型号:TP1898 原产地:中国大陆价格: ¥0.0
产品名称: OXOMEMAZINEhistamine H1-receptor,OXOMEMAZINE,Histamine Receptor,inhibit,phenothiazine,antimuscarinic
产品简介:oxomemazine is a phenothiazine-based histamine h1-receptor blocker with pronounced antimuscarinic activity. oxomemazine is a selective antagonist of mycotoxins ..产品型号:T9353 原产地:中国大陆价格: ¥0.0
产品名称: LM22A-4LM-22A-4,Inhibitor,Trk Receptor,inhibit,LM22A4,LM22A-4,Tropomyosin related kinase receptor,LM
产品简介:lm22a-4 is a brain-derived neurotrophic factor (bdnf) mimetic and agonist of the receptor tropomyosin-related kinase b (trkb; ic50 : 47 nm in a fluorescence ani..产品型号:T7568 原产地:中国大陆价格: ¥0.0
产品名称: Galanin (1-16), mouse, porcine, ratGalanin (1-16), mouse, porcine, rat,Neuropeptide Y Receptor,Inhib
产品简介:galanin (1-16), mouse, porcine, rat is a hippocampal galanin receptor agonist(kd = 3 nm) with high biological activity on locus coeruleus neurons...产品型号:TP1380 原产地:中国大陆价格: ¥0.0
产品名称: Methylbenactyzium BromideInhibitor,Muscarinic acetylcholine receptor,Methylbenactyzium Bromide,inhib
产品简介:dimethadione is an anticonvulsant that is the active metabolite of trimethadione...产品型号:T6744 原产地:中国大陆价格: ¥0.0
产品名称: Bepotastine BesilateInhibitor,Bepotastine Besilate,Bepotastine,inhibit,pruritus,Histamine Receptor,u
产品简介:bepotastine is a non-sedating and selective h1 receptor antagonist (pic50: 5.7)...产品型号:T6405 原产地:中国大陆价格: ¥0.0
产品名称: Atopaxarplatelets,Atopaxar,receptor-1,signaling,PAR-1,inhibit,E-5555,Inhibitor,receptor,Protease Act
产品简介:atopaxar, a reversible par-1 thrombin receptor antagonist, interferes with platelet signaling. atopaxar has been investigated for the treatment of coronary arte..产品型号:T1986 原产地:中国大陆价格: ¥0.0
产品名称: WIN 55,212-2 MesylateCannabinoid Receptor,WIN 55,212-2,inhibit,WIN 55,212 2 Mesylate,Inhibitor,WIN 5
产品简介:win 55, 212-2 (mesylate) is a potent aminoalkylindole cannabinoid (cb) receptor agonist with kis of 62.3 and 3.3 nm for human recombinant cb1 and cb2 receptors,..产品型号:T4458 原产地:中国大陆价格: ¥0.0
产品名称: Necrostatin-34Necrostatin 34,RIP kinase,FADD,Necrostatin-34,RIPK,inhibit,RIPK1,Receptor-interacting
产品简介:necrostatin-34 is a ripk1 kinase inhibitor, stabilizing ripk1 kinase in an inactive conformation by occupying a distinct binding pocket in the kinase domain...产品型号:T9095 原产地:中国大陆价格: ¥0.0
产品名称: VU0238441mAChR,Inhibitor,VU-0238441,VU0238441,Muscarinic acetylcholine receptor,VU 0238441,inhibit
产品简介:vu0238441 is agonist of muscarinic acetylcholine receptor m5 (human) with ec50 of 2.1μm...产品型号:T8219 原产地:中国大陆价格: ¥0.0
产品名称: AR 231453inhibit,GPR119,AR-231453,G Protein-Coupled Receptor 119,diabetes,AR231453,AR 231453,insulin
产品简介:ar 231453 is a selective and orally available gpr119 agonist,can stimulate β-cell replication and improve islet graft function...产品型号:T8329 原产地:中国大陆价格: ¥0.0
产品名称: DarolutamideBAY1841788,BAY 1841788,ODM201,ODM 201,Inhibitor,Androgen Receptor,Darolutamide,inhibit
产品简介:odm-201 is an androgen receptor (ar) antagonist that blocks ar nuclear translocation (ki: 11 nm)...产品型号:T6915 原产地:中国大陆价格: ¥0.0
产品名称: DS-1205TRKA,c-Met/HGFR,migration,Axl,Tyro3,Trk Receptor,MET,DS 1205,Mer,Tropomyosin related kinase r
产品简介:ds-1205 is a potent and selective inhibitor of axl kinase, with an ic50 of 1.3 nm. ds-1205 also inhibits mer, met, and trka, with ic50s of 63, 104, and 407 nm, ..产品型号:T9123 原产地:中国大陆价格: ¥0.0
产品名称: Bevantolol hydrochlorideBevantolol hydrochloride,Beta Receptor,Ca2+ channels,cerebral,Inhibitor,inhi
产品简介:bevantolol hydrochloride is a β1-adrenoceptor antagonist that treatment angina pectoris and hypertension...产品型号:T8143 原产地:中国大陆价格: ¥0.0