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产品目录

产品展示/Products

  • PPARα/δ agonist 1;化合物 PPARα/δ agonist 1PPARα/δ agonist 1

    产品名称: PPARα/δ agonist 1;化合物 PPARα/δ agonist 1PPARα/δ agonist 1

    产品简介:pparα/δ agonist 1 is a potent pparα/pparδ dual agonist with ec50 values of 7.0 nm for pparα and 8.4 nm for pparδ. pparα/δ agonist 1 exhibits high selectivity fo..

    产品型号:T62968 原产地:中国大陆价格: ¥0.0

  • CDK1-IN-1;化合物 CDK1-IN-1CDK1-IN-1

    产品名称: CDK1-IN-1;化合物 CDK1-IN-1CDK1-IN-1

    产品简介:cdk1-in-7 is a potent inhibitor of cdk1 with an ic50 value of 161.2 nm for cdk1/cycb. cdk1-in-7 induces apoptosis in a p53-dependent manner via the apoptosis-in..

    产品型号:T62970 原产地:中国大陆价格: ¥0.0

  • FLT3/CDK4-IN-1;化合物 FLT3/CDK4-IN-1FLT3/CDK4-IN-1

    产品名称: FLT3/CDK4-IN-1;化合物 FLT3/CDK4-IN-1FLT3/CDK4-IN-1

    产品简介:flt3/cdk4-in-1 is a highly selective, potent, orally active dual inhibitor of flt3/cdk4, acting on flt3 (ic50: 7 nm) and cdk4 (ic50: 11 nm).flt3/cdk4-in-1 has g..

    产品型号:T63135 原产地:中国大陆价格: ¥0.0

  • Glutaminyl cyclases-IN-1;化合物 Glutaminyl cyclases-IN-1Glutaminyl cyclases-IN-1

    产品名称: Glutaminyl cyclases-IN-1;化合物 Glutaminyl cyclases-IN-1Glutaminyl cyclases-IN-1

    产品简介:glutaminyl cyclases-in-1 (isoqc-in-1) is a potent inhibitor of glutaminyl cyclases (qc), which acts on human qc (ic50: 12 nm) and isoqc (ic 50:73 nm). glutaminy..

    产品型号:T63139 原产地:中国大陆价格: ¥0.0

  • LSD1-IN-20;LSD1抑制剂20LSD1-IN-20

    产品名称: LSD1-IN-20;LSD1抑制剂20LSD1-IN-20

    产品简介:lsd1-in-20 is a potent dual inhibitor of lsd1/g9a with ki values of 0.44 and 0.68 μm, respectively. lsd1-in-20 showed antiproliferative activity against thp-1 l..

    产品型号:T63140 原产地:中国大陆价格: ¥0.0

  • AChE/HDAC-IN-1;化合物 AChE/HDAC-IN-1AChE/HDAC-IN-1

    产品名称: AChE/HDAC-IN-1;化合物 AChE/HDAC-IN-1AChE/HDAC-IN-1

    产品简介:cox-2-in-23 (compound a10) is a potent inhibitor of ache (ic50: 0.12 nm) and hdac (ic50: 0.23 nm).cox-2-in-23 exhibits antioxidant and metal chelating propertie..

    产品型号:T63142 原产地:中国大陆价格: ¥0.0

  • JAK2/TYK2-IN-1;化合物 JAK2/TYK2-IN-1JAK2/TYK2-IN-1

    产品名称: JAK2/TYK2-IN-1;化合物 JAK2/TYK2-IN-1JAK2/TYK2-IN-1

    产品简介:jak2/tyk2-in-2 is a potent and selective inhibitor of tyk2 (ic50: 9 nm) and jak2 (ic50: 157 nm) with anti-inflammatory effects...

    产品型号:T63146 原产地:中国大陆价格: ¥0.0

  • Calcitriol;骨化三醇Topitriol|||Rocaltrol|||Calcijex|||RO215535|||1,25-Dihydroxyvitamin D3;Topitriol|||Ro

    产品名称: Calcitriol;骨化三醇Topitriol|||Rocaltrol|||Calcijex|||RO215535|||1,25-Dihydroxyvitamin D3;Topitriol|||Ro

    产品简介:calcitriol (1,25-dihydroxyvitamin d3) is a metabolite of vitamin d and a vitamin d receptor (vdr) agonist (ic50=0.4 nm). calcitriol increases intestinal absorpt..

    产品型号:T6316 原产地:中国大陆价格: ¥0.0

  • HIV-1 inhibitor-21;化合物 HIV-1 inhibitor-21HIV-1 inhibitor-21

    产品名称: HIV-1 inhibitor-21;化合物 HIV-1 inhibitor-21HIV-1 inhibitor-21

    产品简介:hiv-1 inhibitor-21 (compound 9b) is a potent inhibitor of hiv-1 non-nucleoside reverse transcriptase (rt) and acts on hiv-1 rt (ic50: 0.55 μm). hiv-1 inhibitor-..

    产品型号:T63113 原产地:中国大陆价格: ¥0.0

  • SOS1-IN-8;化合物 SOS1-IN-8SOS1-IN-8

    产品名称: SOS1-IN-8;化合物 SOS1-IN-8SOS1-IN-8

    产品简介:sos1-in-8 is an inhibitor of sos1 and acts on sos1-g12d (ic50: 11.6 nm) and sos1-g12v (ic50: 40.7 nm)...

    产品型号:T63118 原产地:中国大陆价格: ¥0.0

  • NF-κB/MAPK-IN-1;NF-κB/MAPK抑制剂1NF-κB/MAPK-IN-1

    产品名称: NF-κB/MAPK-IN-1;NF-κB/MAPK抑制剂1NF-κB/MAPK-IN-1

    产品简介:nf-κb/mapk-in-1 is a potent dual inhibitor of the nf-κb and mapk pathways with potential anti-inflammatory activity, inhibition of no production, and inhibition..

    产品型号:T63119 原产地:中国大陆价格: ¥0.0

  • ZIKV-IN-1;化合物 ZIKV-IN-1ZIKV-IN-1

    产品名称: ZIKV-IN-1;化合物 ZIKV-IN-1ZIKV-IN-1

    产品简介:zikv-in-1 is a potent inhibitor of zika virus (ec50: 2.8 μm, ec90: 6.8 μm). zikv-in-1 has anti-zikv effects and low cytotoxicity. zikv-in-1 shows high affinity ..

    产品型号:T63131 原产地:中国大陆价格: ¥0.0

  • (R)-MALT1-IN-7;化合物 (R)-MALT1-IN-7(R)-MALT1-IN-7

    产品名称: (R)-MALT1-IN-7;化合物 (R)-MALT1-IN-7(R)-MALT1-IN-7

    产品简介:(r)-malt1-in-7 (compound 142a) is a potent inhibitor of malt1 protease and has potential for cancer research...

    产品型号:T63133 原产地:中国大陆价格: ¥0.0

  • MALT1-IN-7;化合物 MALT1-IN-7MALT1-IN-7

    产品名称: MALT1-IN-7;化合物 MALT1-IN-7MALT1-IN-7

    产品简介:malt1-in-7 (compound 142b) is a potent inhibitor of malt1 protease with potential for cancer research...

    产品型号:T63134 原产地:中国大陆价格: ¥0.0

  • iNOs-IN-1;化合物 iNOs-IN-1iNOs-IN-1

    产品名称: iNOs-IN-1;化合物 iNOs-IN-1iNOs-IN-1

    产品简介:inos-in-1 (ypw) is a potent inhibitor of inducible nitric oxide synthase (inos) with anti-inflammatory effects. inos-in-1 significantly inhibits il-6 and inos e..

    产品型号:T62987 原产地:中国大陆价格: ¥0.0

  • Mpro/PLpro-IN-1;化合物 Mpro/PLpro-IN-1Mpro/PLpro-IN-1

    产品名称: Mpro/PLpro-IN-1;化合物 Mpro/PLpro-IN-1Mpro/PLpro-IN-1

    产品简介:mpro/plpro-in-1 (compound 29) is a dual-acting inhibitor of sars-cov-2 protease.mpro/plpro-in-1 is also a potent inhibitor of mpro/plpro, with micromolar inhibi..

    产品型号:T62991 原产地:中国大陆价格: ¥0.0

  • BACE-1 inhibitor 2;化合物 BACE-1 inhibitor 2BACE-1 inhibitor 2

    产品名称: BACE-1 inhibitor 2;化合物 BACE-1 inhibitor 2BACE-1 inhibitor 2

    产品简介:bace-1 inhibitor 2 is a potent, cns-permeable inhibitor of bace-1, exhibiting an ic50 value of 1.5 nm in enzymatic assays [1]...

    产品型号:T62995 原产地:中国大陆价格: ¥0.0

  • PI3K/AKT-IN-1;化合物 PI3K/AKT-IN-1PI3K/AKT-IN-1

    产品名称: PI3K/AKT-IN-1;化合物 PI3K/AKT-IN-1PI3K/AKT-IN-1

    产品简介:pi3k/akt-in-1 is a potent, dual pi3k/akt inhibitor that acts on pi3kγ (ic50: 6.99 μm), pi3kδ (ic50: 4.01 μm) and akt (ic50: 3.36 μm). pi3k/akt-in-1 induces casp..

    产品型号:T62997 原产地:中国大陆价格: ¥0.0

  • COX-2/15-LOX-IN-1;化合物 COX-2/15-LOX-IN-1COX-2/15-LOX-IN-1

    产品名称: COX-2/15-LOX-IN-1;化合物 COX-2/15-LOX-IN-1COX-2/15-LOX-IN-1

    产品简介:cox-2/15-lox-in-1 (compound 14) is a cox-2 and 15-lipoxygenase (15-lox) inhibitor that acts on cox-1 (ic50: 10.65 μm), cox-2 (ic50: 0.075 μm) and 15-lox (ic50: ..

    产品型号:T62998 原产地:中国大陆价格: ¥0.0

  • Germination-IN-1;化合物 Germination-IN-1Germination-IN-1

    产品名称: Germination-IN-1;化合物 Germination-IN-1Germination-IN-1

    产品简介:germination-in-1 (compound 11) is a potent germination inhibitor (ic50: 4 μm) with anti-germination effects (germination rate = 14%)...

    产品型号:T62999 原产地:中国大陆价格: ¥0.0

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