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产品名称: TheliatinibATP-competitive,inhibit,EGFR,ERK,cancer,esophageal,Epidermal growth factor receptor,HMPL-
产品简介:theliatinib, a potent and highly selective egfr inhibitor, with anti-tumor activity. ki of 0.05 nm for wild type egfr, and ic50s of 3 and 22 nm for egfr and egf..产品型号:T7322 原产地:中国大陆价格: ¥0.0
产品名称: Eltoprazine hydrochlorideDU-28853,5-hydroxytryptamine Receptor,Inhibitor,DU 28853,5-HT Receptor,DU28
产品简介:eltoprazine hydrochloride is a partial agonist at serotonin 5-ht1a, 5-ht1b, and 5-ht2b receptors (ki value of 40, 52, and 81 nm, respectively)...产品型号:T7498 原产地:中国大陆价格: ¥0.0
产品名称: LML134inhibit,LML134,LML 134,Inhibitor,Histamine Receptor
产品简介:lml-134 is an inverse agonist of histamine 3 receptor (h3r)(hh3r camp and hh3r bdg with kis of 0.3 nm and 12 nm)...产品型号:T8514 原产地:中国大陆价格: ¥0.0
产品名称: Ripretinibc-Kit,Inhibitor,DCC2618,Vascular endothelial growth factor receptor,CD135,CD117,Platelet-d
产品简介:ripretinib is an orally bioavailable inhibitor of kit and pdgfra...产品型号:T8482 原产地:中国大陆价格: ¥0.0
产品名称: PRX-07034 hydrochlorideflexibility,5-HT6,PRX 07034,working,Serotonin Receptor,cognitive,Inhibitor,in
产品简介:prx-07034 is a selective antagonist of 5-ht6 receptor. it has cognition and memory-enhancing properties and potently decreases food intake and body weight in ro..产品型号:T8720 原产地:中国大陆价格: ¥0.0
产品名称: Indophagolininhibit,formation,Inhibitor,Indophagolin,5-hydroxytryptamine Receptor,autophagosome,Sero
产品简介:indophagolin is a potent, indoline-containing autophagy inhibitor with ic50 of 140 nm. indophagolin antagonizes the purinergic receptor p2x4 as well as p2x1 and..产品型号:T8946 原产地:中国大陆价格: ¥0.0
产品名称: OglufanideM21 human melanoma,anti-angiogenesis,Vascular endothelial growth factor receptor,HCV,inhib
产品简介:oglufanide is a naturally occurring thymic immunomodulator,and inhibits vascular endothelial growth factor (vegf)...产品型号:T7203 原产地:中国大陆价格: ¥0.0
产品名称: Xaliproden hydrochloride5-HT Receptor,Xaliproden hydrochloride,SR57746A,Serotonin Receptor,dopamine,
产品简介:xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-ht1a receptor agonist...产品型号:T9272 原产地:中国大陆价格: ¥0.0
产品名称: Vatalanib dihydrochloridePTK-787,Inhibitor,Vascular endothelial growth factor receptor,VEGFR,PTK 787
产品简介:vatalanib (ptk787) (ic50=37 nm) is an inhibitor of vegfr2/kdr. it exhibits less effective against vegfr1/flt-1 and 18-fold against vegfr3/flt-4...产品型号:T6720 原产地:中国大陆价格: ¥0.0
产品名称: OkaninToll-like Receptor (TLR),Nuclear factor-κB,NF-κB,Inhibitor,Nuclear factor-kappaB,Okanin,inhibi
产品简介:okanin shows significant activities on both linoleic acid peroxidation inhibition and dpph radical scavenging effect...产品型号:TN2008 原产地:中国大陆价格: ¥0.0
产品名称: A-317491flux,calcium,P2X Receptor,A 317491,Inhibitor,neuropathic,inhibit,P2X2/3,A317491,P2X3,P2XRs,p
产品简介:a-317491 is a non-nucleotide p2x3 ( ki: 22 nm) and p2x2/3 receptor (ki: 9 nm) antagonist, which inhibits calcium flux mediated by the receptors...产品型号:TQ0002 原产地:中国大陆价格: ¥0.0
产品名称: SU 5402SU-5402,SU 5402,VEGFR,inhibit,Inhibitor,Fibroblast growth factor receptor,FGFR,Platelet-deriv
产品简介:su5402 is a potent multi-targeted receptor tyrosine kinase inhibitor with ic50 of 20 nm, 30 nm, and 510 nm for vegfr2, fgfr1, and pdgf-rβ, respectively...产品型号:T6996 原产地:中国大陆价格: ¥0.0
产品名称: Deltorphin 2inhibit,Deltorphin2,Inhibitor,Deltorphin 2,Opioid Receptor,Deltorphin-2
产品简介:deltorphin 2(tfa) is an agonist of δ opioid receptor(ic50:0.41 nm)..产品型号:T7639 原产地:中国大陆价格: ¥0.0
产品名称: BepotastineBepotastine,Histamine Receptor,conjunctivitis,LTB 4,pruritus,Inhibitor,atopic dermatitis,
产品简介:bepotastine free base is a histamine 1 (h1) receptor antagonis...产品型号:T7893 原产地:中国大陆价格: ¥0.0
产品名称: SB-408124SB408124,SB 408124,inhibit,water,membrane,selectivity,Inhibitor,Orexin Receptor (OX Recepto
产品简介:sb408124 is a non-peptide antagonist for ox1 receptor with ki of 57 nm and 27 nm in both whole cell and membrane, respectively, exhibits 50-fold selectivity ove..产品型号:T6658 原产地:中国大陆价格: ¥0.0
产品名称: TianeptineTianeptine,Serotonin Receptor,Inhibitor,inhibit,5-HT Receptor,5-hydroxytryptamine Receptor
产品简介:tianeptine is a selective 5-ht uptake facilitator in vitro and in vivo...产品型号:T8140 原产地:中国大陆价格: ¥0.0
产品名称: BMS986188BMS986188,Opioid Receptor,inhibit,BMS-986188,Inhibitor,BMS 986188
产品简介:bms986188 is a novel potent and selective positive allosteric modulator of the delta-opioid receptor...产品型号:T8992 原产地:中国大陆价格: ¥0.0
产品名称: AtrasentanAtrasentan,Endothelin Receptor,A 147627,ABT627,Inhibitor,inhibit,A147627,ABT 627
产品简介:atrasentan (abt-627) is an endothelin receptor antagonist (ic50: 0.0551 nm for eta)...产品型号:TQ0259 原产地:中国大陆价格: ¥0.0
产品名称: Galanin Receptor Ligand M35 TFAGalanin Receptor Ligand M35 TFA,Galanin Receptor Ligand M-35 TFA
产品简介:galanin receptor ligand m35 tfa is a high-affinity ligand and antagonist of galanin receptor (kd=0.1 nm)...产品型号:TP1704 原产地:中国大陆价格: ¥0.0
产品名称: Exendin-4 acetateExenatide,Exendin 4 acetate,Glucagon Receptor,Exendin-4,inhibit,Exendin4 acetate,Ex
产品简介:exendin-4 acetate is a 39 amino acid peptide.exendin-4 acetate is a long-acting glp-1 receptor agonist(ic50 = 3.22 nm)...产品型号:T8748 原产地:中国大陆价格: ¥0.0