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产品名称: PROTAC FLT3/CDK9 degrader-1;化合物 PROTAC FLT3/CDK9 degrader-1PROTAC FLT3/CDK9 degrader-1
产品简介:protac flt3/cdk9 degrader-1, a potent dual degrader of flt3 and cdk9, effectively induces apoptosis and targets protein degradation of flt3 and cdk9. this compo..产品型号:T74707 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC PTPN2 degrader-1;化合物 PROTAC PTPN2 degrader-1PROTAC PTPN2 degrader-1
产品简介:protac ptpn2 degrader-1 (compound example 77) is a potent entity capable of degrading ptpn2, showing promise for research applications in cancer or metabolic di..产品型号:T74732 原产地:中国大陆价格: ¥0.0
产品名称: GSPT1 degrader-1;化合物 GSPT1 degrader-1GSPT1 degrader-1
产品简介:gspt1 degrader-1 (compound 9q) effectively facilitates the degradation of g1 to s phase transition 1 (gspt1) through the ubiquitin-proteasome system and induces..产品型号:T79474 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC TG2 degrader-1;化合物 PROTAC TG2 degrader-1PROTAC TG2 degrader-1
产品简介:protac tg2 degrader-1 (compound 11) is a vhl-based protac that targets tissue transglutaminase (tg2) and exhibits a binding affinity with a k d of 68.9 μm. this..产品型号:T79505 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC TTK degrader-1;化合物 PROTAC TTK degrader-1PROTAC TTK degrader-1
产品简介:protac ttk degrader-1, a potent threonine tyrosine kinase (ttk) protac degrader, demonstrates dc50 values of 1.7 nm in colo-205 cells and 5.8 nm in hct-116 cell..产品型号:T81375 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC NSD3 degrader-1;化合物 PROTAC NSD3 degrader-1PROTAC NSD3 degrader-1
产品简介:protac nsd3 degrader-1 (compound 56) is a targeted degradation agent for the nuclear receptor binding set domain protein nsd3. it effectively induces the degrad..产品型号:T81377 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC GDI2 Degrader-1;化合物 PROTAC GDI2 Degrader-1PROTAC GDI2 Degrader-1
产品简介:protac gdi2 degrader-1 (compound 21) is a potent degrader of protac gdi2, demonstrating outstanding antitumor activity in vivo within pancreatic xenograft model..产品型号:T81379 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC eDHFR Degrader-1;化合物 PROTAC eDHFR Degrader-1PROTAC eDHFR Degrader-1
产品简介:protac edhfr degrader-1 is a potent degrader targeting edhfr-yfp and various proteins of interest (pois), such as yfp and luciferase [1]...产品型号:T81381 原产地:中国大陆价格: ¥0.0
产品名称: BRD9 Degrader-1;化合物 BRD9 Degrader-1BRD9 Degrader-1
产品简介:brd9 degrader-1 functions as a brd9 degrader, demonstrating micromolar binding affinity towards brd9 and nanomolar affinity for the ternary complex involving br..产品型号:T82821 原产地:中国大陆价格: ¥0.0
产品名称: STAT3 degrader-1;化合物 STAT3 degrader-1STAT3 degrader-1
产品简介:stat3 degrader-1 (compound 295) is a potent degrader of stat3, utilized in anticancer research [1]...产品型号:T74545 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC EZH2 Degrader-1;化合物 PROTAC EZH2 Degrader-1PROTAC EZH2 Degrader-1
产品简介:protac ezh2 degrader-1 (compound 150d), a potent inhibitor, effectively suppresses ezh2 methyltransferase activity, demonstrating an ic50 of 2.7 nm. ezh2 is cru..产品型号:T74602 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC AR-V7 degrader-1;化合物 PROTAC AR-V7 degrader-1PROTAC AR-V7 degrader-1
产品简介:protac ar-v7 degrader-1 (compound 6) is an orally bioavailable, potent, and selective degrader targeting the androgen receptor (ar) variant v7, achieving degrad..产品型号:T74410 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC ERα Y537S degrader-1;化合物 PROTAC ERα Y537S degrader-1PROTAC ERα Y537S degrader-1
产品简介:protac erα y537s degrader-1 comprises a ubiquitin e3 ligase binding group, a linker and a protein binding group. protac erα y537s degrader-1 is an estrogen rece..产品型号:T74375 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC SOS1 degrader-1;化合物 PROTAC SOS1 degrader-1PROTAC SOS1 degrader-1
产品简介:protac sos1 degrader-1, a potent compound, demonstrates an effective degradation of protac sos1 with a dc50 value of 98.4 nm. it exhibits antiproliferative acti..产品型号:T74439 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC eEF2K degrader-1;化合物 PROTAC eEF2K degrader-1PROTAC eEF2K degrader-1
产品简介:protac eef2k degrader-1 (compound 11l), an eef2k-targeting protac small molecule, effectively induces apoptosis in mda-mb-231 cells through mediating eef2k degr..产品型号:T74512 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC VEGFR-2 degrader-1;化合物 PROTAC VEGFR-2 degrader-1PROTAC VEGFR-2 degrader-1
产品简介:protac vegfr-2 degrader-1 (protac-1), a specific degrader of protac vegfr-2, demonstrates minimal inhibition of vegfr-2 (ic50 > 1 μm) and exhibits low anti-prol..产品型号:T74517 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC CYP1B1 degrader-1;化合物 PROTAC CYP1B1 degrader-1PROTAC CYP1B1 degrader-1
产品简介:protac cyp1b1 degrader-1 (compound 6c), an α-naphthoflavone chimera derivative, effectively targets and degrades cytochrome p450 (cyp) 1b1 to overcome agent res..产品型号:T74519 原产地:中国大陆价格: ¥0.0
产品名称: IRAK degrader-1;化合物 IRAK degrader-1IRAK degrader-1
产品简介:irak degrader-1 (example i-3) is a potent irak degrader [1] ...产品型号:T75136 原产地:中国大陆价格: ¥0.0
产品名称: HDAC6 degrader-1;化合物 HDAC6 degrader-1HDAC6 degrader-1
产品简介:hdac6 degrader-1, a proteolysis-targeting chimeric molecule (protac), incorporates the selective hdac6 inhibitor nexturastat a (nex a) for hdac6 binding, a link..产品型号:T77922 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC KRAS G12C degrader-1;化合物 PROTAC KRAS G12C degrader-1PROTAC KRAS G12C degrader-1
产品简介:protac kras g12c degrader-1, a cereblon-based degrader, promotes crbn/kras g12c dimerization and facilitates the degradation of gfp-kras g12c in reporter cells ..产品型号:T77926 原产地:中国大陆价格: ¥0.0