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产品名称: Topotecan hydrochloride hydrate;化合物 Topotecan hydrochloride hydrateTopotecan hydrochloride hydrate
产品简介:topotecan hydrochloride hydrate is an orally active topoisomerase i inhibitor with anticancer properties. topotecan hydrochloride hydrate is capable of blocking..产品型号:T63105 原产地:中国大陆价格: ¥0.0
产品名称: Estrogen receptor antagonist 4;化合物 Estrogen receptor antagonist 4Estrogen receptor antagonist 4
产品简介:estrogen receptor antagonist 4 is a potent inhibitor of the estrogen receptor (er), crucial for regulating cell growth, differentiation, and apoptosis. this com..产品型号:T63106 原产地:中国大陆价格: ¥0.0
产品名称: Anti-inflammatory agent 6;化合物 Anti-inflammatory agent 6Anti-inflammatory agent 6
产品简介:anti-inflammatory agent 6 exhibits anti-inflammatory potential by blocking the phosphorylation of iκb kinase α/β (ikkα/β), iκbα and nuclear factor kb p65 (nf-κb..产品型号:T63107 原产地:中国大陆价格: ¥0.0
产品名称: AKT-IN-13;化合物 AKT-IN-13AKT-IN-13
产品简介:akt-in-13 (compound 4b) is a potent inhibitor of akt, acting on akt1 (ic50: 1.6 nm), akt2 (ic50: 2.4 nm) and akt3 (ic50: 0.3 nm). akt-in-13 can be used in antic..产品型号:T63039 原产地:中国大陆价格: ¥0.0
产品名称: CCT128930 hydrochloride;化合物CCT128930 hydrochlorideCCT128930 hydrochloride(885499-61-6 Free base);CCT
产品简介:cct128930 hydrochloride (cct128930 hydrochloride) is a potent and selective inhibitor of akt with ic50 of 6 nm. cct128930 hydrochloride induces cell cycle arres..产品型号:T6303L 原产地:中国大陆价格: ¥0.0
产品名称: AT7867;化合物AT7867AT7867
产品简介:at7867 is a potent atp-competitive inhibitor of akt1/2/3 and p70s6k/pka with ic50 of 32 nm/17 nm/47 nm and 85 nm/20 nm, respectively; little activity outside th..产品型号:T6304 原产地:中国大陆价格: ¥0.0
产品名称: GNF2133 hydrochloride;化合物 GNF2133 hydrochlorideGNF2133 hydrochloride
产品简介:gnf2133 hydrochloride is a selective, effective, and orally active dyrk1a inhibitor, able to act on dyrk1a (ic50: 0.0062 μm) and gsk3β (ic50> 50 μm); gnf2133 hy..产品型号:T63040 原产地:中国大陆价格: ¥0.0
产品名称: DS01080522;化合物 DS01080522DS01080522
产品简介:ds01080522 is an inhibitor of prkaca. ds01080522 inhibited prkaca kinase activity (ic50.0.8 nm) and creb phosphorylation (ic50.66 nm). ds0108052 can be used to ..产品型号:T63041 原产地:中国大陆价格: ¥0.0
产品名称: NDB;化合物NDBNDB
产品简介:ndb is a selective and potent hfxrα antagonist that inhibits gw4064-stimulated fxr/rxr interactions and fxrα target gene expression in primary mouse hepatocytes..产品型号:T63042 原产地:中国大陆价格: ¥0.0
产品名称: Antimalarial agent 2;化合物 Antimalarial agent 2Antimalarial agent 2
产品简介:antimalarial agent 2 is an orally active, novel antimalarial agent that exhibits rapid in vitro killing effects...产品型号:T63043 原产地:中国大陆价格: ¥0.0
产品名称: SOS1-IN-6;化合物 SOS1-IN-6SOS1-IN-6
产品简介:sos1-in-6 (compound 33-p1) is a potent inhibitor of sos1, acting on sos1-g12d (ic50: 14.9 nm) and sos1-g12v (ic50: 73.3 nm)...产品型号:T63044 原产地:中国大陆价格: ¥0.0
产品名称: (1S,3R)-GNE-502;化合物 (1S,3R)-GNE-502(1S,3R)-GNE-502
产品简介:(1s,3r)-gne-502 (compound 179) is a potent degradation agent of erα and is able to degrade erα in mcf7 hcs cells (ec50: 13 nm). (1s,3r)-gne-502 can be used in t..产品型号:T63045 原产地:中国大陆价格: ¥0.0
产品名称: HPK1-IN-15;化合物 HPK1-IN-15HPK1-IN-15
产品简介:hpk1-in-15 is a selective and effective inhibitor of hpk1. hematopoietic progenitor kinase 1 (hpk1), which was originally cloned from hematopoietic progenitor c..产品型号:T63046 原产地:中国大陆价格: ¥0.0
产品名称: SLP9101555;化合物SLP9101555SLP9101555
产品简介:slp9101555 is a potent and selective sphingosine kinase 2 (sphk2) inhibitor with a ki of 90 nm.slp9101555 has a high affinity for sphk2, which is 200-fold highe..产品型号:T63047 原产地:中国大陆价格: ¥0.0
产品名称: Sigma-LIGAND-1 hydrochloride;化合物 Sigma-LIGAND-1 hydrochlorideSigma-LIGAND-1 hydrochloride
产品简介:sigma-ligand-1 hydrochloride is a selective sigma receptor ligand that acts at the dtg (ic50: 16 nm) and ppp (ic50: 19 nm) sites. sigma-ligand-1 hydrochloride i..产品型号:T63048 原产地:中国大陆价格: ¥0.0
产品名称: CHD1Li 6.11;化合物CHD1Li 6.11CHD1Li 6.11
产品简介:chd1li 6.11 is a potent inhibitor of oncogenic chd1l, acting on the cat-chd1l recombinant protein (ic50: 3.3 μm). chd1li 6.11 is an orally active antitumour age..产品型号:T63049 原产地:中国大陆价格: ¥0.0
产品名称: SNX2112;化合物SNX2112SNX-2112|||PF 04928473|||SNX 2112;SNX-2112|||PF 04928473|||SNX 2112
产品简介:snx2112 (pf 04928473) is an orally active hsp90 inhibitor, with a kd of 16 nm...产品型号:T6305 原产地:中国大陆价格: ¥0.0
产品名称: JH-XVII-10;化合物 JH-XVII-10JH-XVII-10
产品简介:jh-xvii-10 is a selective, orally active and potent inhibitor of dyrk1a (ic50: 3 nm) and dyrk1b (ic50: 5 nm).jh-xvii-10 exhibits antitumor effects in squamous c..产品型号:T63050 原产地:中国大陆价格: ¥0.0
产品名称: (R)-MALT1-IN-3;化合物 (R)-MALT1-IN-3(R)-MALT1-IN-3
产品简介:(r)-malt1-in-3 (compound 121) is a potent inhibitor of malt1 protease (ic50: 20 nm) with ic50 values of 60 nm and 40 nm for human il6/il10 in oci-ly3 cells, res..产品型号:T63051 原产地:中国大陆价格: ¥0.0
产品名称: Antimalarial agent 10;化合物 Antimalarial agent 10Antimalarial agent 10
产品简介:antimalarial agent 10 (compound 17b) is an amino alcohol-quinoline compound. antimalarial agent 10 is also an antimalarial agent capable of acting on pf3d7 (ic5..产品型号:T63052 原产地:中国大陆价格: ¥0.0