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产品名称: Aurora A/PKC-IN-1;化合物 Aurora A/PKC-IN-1Aurora A/PKC-IN-1
产品简介:aurora a/pkc-in-1 (compound 2e) is a potent dual inhibitor of aurora a (aura) and pkc (α, β1, β2, θ), acting on aura (ic50: 6.9 nm) and pkcα (ic50: 16.9 nm). au..产品型号:T62945 原产地:中国大陆价格: ¥0.0
产品名称: Dopamine D3 receptor antagonist-2;化合物 Dopamine D3 receptor antagonist-2Dopamine D3 receptor antagoni
产品简介:dopamine d3 receptor antagonist-2 is a dopamine d3 receptor selective (ki=2.16 nm) or multi-targeting dual ligand that shows potential effects in cns disorders...产品型号:T62946 原产地:中国大陆价格: ¥0.0
产品名称: Lp-PLA2-IN-11;化合物 Lp-PLA2-IN-11Lp-PLA2-IN-11
产品简介:lp-pla2-in-11 is a potent inhibitor of lipoprotein-associated phospholipase a2 (lp-pla2). lp-pla2-in-11 has the potential to be investigated in diseases associa..产品型号:T62947 原产地:中国大陆价格: ¥0.0
产品名称: PI3Kβ-IN-1;化合物 PI3Kβ-IN-1PI3Kβ-IN-1
产品简介:pi3kβ-in-1 is a selective, orally active pi3kβ inhibitor (ic50: 2 nm)...产品型号:T62948 原产地:中国大陆价格: ¥0.0
产品名称: (1R,3S)-THCCA-Asn;化合物 (1R,3S)-THCCA-Asn(1R,3S)-THCCA-Asn
产品简介:(1r,3s)-thcca-asn (4j) is a selective inhibitor of thrombin (ic50: 0.07-0.14 μm) with anti-thrombotic effects...产品型号:T62949 原产地:中国大陆价格: ¥0.0
产品名称: IRAK4-IN-18;化合物 IRAK4-IN-18IRAK4-IN-18
产品简介:irak4-in-18 is a potent inhibitor of interleukin 1 receptor-associated kinase 4 (irak4) (ic50: 15 nm). irak4-in-18 inhibits lps-induced il23 production in thp a..产品型号:T62950 原产地:中国大陆价格: ¥0.0
产品名称: Aldose reductase-IN-2;化合物 Aldose reductase-IN-2Aldose reductase-IN-2
产品简介:aldose reductase-in-2 (compound 5f) is a potent inhibitor of aldose reductase (ar) with antioxidant properties. aldose reductase-in-2 is a promising anti-diabet..产品型号:T62951 原产地:中国大陆价格: ¥0.0
产品名称: Estrogen receptor antagonist 5;化合物 Estrogen receptor antagonist 5Estrogen receptor antagonist 5
产品简介:estrogen receptor antagonist 5 is a potent antagonist of the estrogen receptor. estrogen receptor (estrogen receptor) is a ligand-activated transcriptional regu..产品型号:T62952 原产地:中国大陆价格: ¥0.0
产品名称: Estrogen receptor antagonist 6;化合物 Estrogen receptor antagonist 6Estrogen receptor antagonist 6
产品简介:estrogen receptor antagonist 6 is a potent antagonist of the estrogen receptor. estrogen receptor is a ligand-activated transcriptional regulatory protein that ..产品型号:T62953 原产地:中国大陆价格: ¥0.0
产品名称: Ferroportin-IN-1;化合物 Ferroportin-IN-1Ferroportin-IN-1
产品简介:ferroportin-in-1 is an inhibitor of the iron transport protein ferroportin and can be used to study diseases such as thalassaemia, sickle cell disease and haemo..产品型号:T62954 原产地:中国大陆价格: ¥0.0
产品名称: PARP1-IN-5;化合物 PARP1-IN-5PARP1-IN-5
产品简介:parp1-in-5 is a potent, selective, orally active, low-toxicity parp-1 inhibitor with an ic50 value of 14.7 nm. parp1-in-5 can be used in cancer research...产品型号:T62955 原产地:中国大陆价格: ¥0.0
产品名称: RORγt inverse agonist 29;化合物 RORγt inverse agonist 29RORγt inverse agonist 29
产品简介:rorγt inverse agonist 29 is a potent, selective, orally active rorγt inverse agonist with an ic50 value of 21 nm. rorγt inverse agonist 29 can be used in the st..产品型号:T62956 原产地:中国大陆价格: ¥0.0
产品名称: MRK-740;化合物MRK-740MRK-740
产品简介:mrk-740 is a potent and selective inhibitor of prdm9 histone methyltransferase.mrk-740 inhibits other histone methyltransferases and inhibits prdm9-dependent h3..产品型号:T62957 原产地:中国大陆价格: ¥0.0
产品名称: SARS-CoV-2-IN-31;化合物 SARS-CoV-2-IN-31SARS-CoV-2-IN-31
产品简介:sars-cov-2-in-31 is a potent inhibitor of covid-19. sars-cov-2-in-31 shows excellent to mild activity (ic50: 28.84-38.36 μm) against a variety of cancer cell li..产品型号:T62958 原产地:中国大陆价格: ¥0.0
产品名称: LRH-1 modulator-1;化合物 LRH-1 modulator-1LRH-1 modulator-1
产品简介:lrh-1 modulator-1 is a potent modulator/agonist of lrh-1 (liver receptor homolog-1). lrh-1 modulator-1 induces the anti-inflammatory cytokine il-10 and exhibits..产品型号:T62959 原产地:中国大陆价格: ¥0.0
产品名称: RAF265;化合物RAF265CHIR-265;CHIR-265
产品简介:raf265 (chir-265) (chir-265) is a potent selective inhibitor of c-raf/b-raf/b-raf v600e with ic50 of 3-60 nm, and exhibits potent inhibition on vegfr2 phosphory..产品型号:T6296 原产地:中国大陆价格: ¥0.0
产品名称: ZK824859 hydrochloride;化合物 ZK824859 hydrochlorideZK824859 hydrochloride
产品简介:zk824859 hydrochloride is a selective, orally active inhibitor of urokinase-type fibrinogen activator (upa) with ic50 values of 79 nm, 1580 nm and 1330 nm for h..产品型号:T62961 原产地:中国大陆价格: ¥0.0
产品名称: Axl-IN-3;化合物 Axl-IN-3Axl-IN-3
产品简介:axl-in-3 is a selective, potent and orally active inhibitor of axl kinase (ic50: 41.5 nm) and has a low inhibitory effect on other kinases...产品型号:T62962 原产地:中国大陆价格: ¥0.0
产品名称: Xanthine amine congener hydrochloride;化合物 Xanthine amine congener hydrochlorideXanthine amine congen
产品简介:xanthine amine congener (xac) hydrochloride is a non-selective adenosine receptor antagonist that induces convulsions in mice...产品型号:T62963 原产地:中国大陆价格: ¥0.0
产品名称: AdipoRon hydrochloride;化合物 AdipoRon hydrochlorideAdipoRon hydrochloride
产品简介:adiporon hydrochloride is a specific, orally active adipor agonist, capable of binding adipor1 (kd: 1.8 μm) and adipor2 (kd: 3.1 μm)...产品型号:T62964 原产地:中国大陆价格: ¥0.0