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产品名称: RORγt/DHODH-IN-1;化合物 RORγt/DHODH-IN-1RORγt/DHODH-IN-1
产品简介:rorγt/dhodh-in-1 (compound (r)-14d) is a potent, orally active dual inhibitor of rorγt (ic50: 0.083 μm) and dhodh (ic50: 0.172 μm), which exhibits significant i..产品型号:T64145 原产地:中国大陆价格: ¥0.0
产品名称: RORγt/DHODH-IN-3;化合物 RORγt/DHODH-IN-3RORγt/DHODH-IN-3
产品简介:rorγt/dhodh-in-3 (compound (s)-14d) is a potent, orally active dual inhibitor of rorγt (ic50: 0.098 μm) and dhodh (ic50: 0.432 μm).rorγt/dhodh-in-1 has signific..产品型号:T64146 原产地:中国大陆价格: ¥0.0
产品名称: ERK1/2 inhibitor 6;化合物 ERK1/2 inhibitor 6ERK1/2 inhibitor 6
产品简介:erk1/2 inhibitor 6 is a potent inhibitor of erk1/2. erk1/2 inhibitor 6 has shown potential for the study or prevention of cancer, inflammation or other prolifer..产品型号:T64147 原产地:中国大陆价格: ¥0.0
产品名称: LXR agonist 2;化合物 LXR agonist 2LXR agonist 2
产品简介:lxr agonist 2 is a potent agonist of the lxr (liver x receptor). lxr agonist 2 stabilises ncoa1 (coactivator), which in turn agonises the lxr...产品型号:T64148 原产地:中国大陆价格: ¥0.0
产品名称: CX-5461 dihydrochloride;化合物 CX-5461 dihydrochlorideCX-5461 dihydrochloride
产品简介:cx-5461 dihydrochloride is a potent, orally active inhibitor of pol i-mediated rrna synthesis that acts on hct-116 cells (ic50: 142 nm), a375 cells (ic50: 113 n..产品型号:T64150 原产地:中国大陆价格: ¥0.0
产品名称: Mibefradil dihydrochloride hydrate;化合物 Mibefradil dihydrochloride hydrateMibefradil dihydrochloride
产品简介:mibefradil dihydrochloride hydrate (ro 40-5967 dihydrochloride hydrate) is a long-acting calcium channel antagonist. mibefradil dihydrochloride hydrate is an an..产品型号:T64151 原产地:中国大陆价格: ¥0.0
产品名称: Purinostat mesylate;化合物 Purinostat mesylatePurinostat mesylate
产品简介:purinostat mesylate is a selective hdac inhibitor. purinostat mesylate inhibits type i and type iib hdacs (ic50: 0.81-11.5 nm). purinostat mesylate affects the ..产品型号:T64152 原产地:中国大陆价格: ¥0.0
产品名称: Glyoxalase I inhibitor 1;化合物 Glyoxalase I inhibitor 1Glyoxalase I inhibitor 1
产品简介:glyoxalase i inhibitor 1 is a potent inhibitor of glyoxalase i (glo1) (ic50: 26 nm)...产品型号:T64153 原产地:中国大陆价格: ¥0.0
产品名称: CYP51/HDAC-IN-1;化合物 CYP51/HDAC-IN-1CYP51/HDAC-IN-1
产品简介:cyp51/hdac-in-1 is an orally active, potent, dual cyp51/hdac inhibitor that inhibits important virulence factors and down-regulates the expression of associated..产品型号:T64154 原产地:中国大陆价格: ¥0.0
产品名称: AChE/BChE-IN-1;化合物 AChE/BChE-IN-1AChE/BChE-IN-1
产品简介:ache/bche-in-1 is a potent dual inhibitor of acetylcholinesterase and butyrylcholinesterase with blood-brain barrier permeability, exhibiting an ic50 value of 1..产品型号:T64156 原产地:中国大陆价格: ¥0.0
产品名称: OXi8007;化合物 OXi8007OXi8007
产品简介:oxi8007 is a water-soluble phosphate that is a prodrug for oxi8006, a microtubulin-binding compound. oxi8007 is a vascular disrupting agent with potential antic..产品型号:T64157 原产地:中国大陆价格: ¥0.0
产品名称: Nenocorilant;化合物 NenocorilantNenocorilant
产品简介:nenocorilant (relacorilant) is an orally active glucocorticoid receptor (gr) antagonist (ki: 0.15 nm). nenocorilant can be used to study tumours...产品型号:T64158 原产地:中国大陆价格: ¥0.0
产品名称: Cathepsin K inhibitor 2;化合物 Cathepsin K inhibitor 2Cathepsin K inhibitor 2
产品简介:cathepsin k inhibitor 2 is a potent inhibitor of cathepsin k. cathepsin k (cat k) is a cysteine protease expressed under the control of the ctsk gene, which is ..产品型号:T64159 原产地:中国大陆价格: ¥0.0
产品名称: MraY-IN-3;化合物 MraY-IN-3MraY-IN-3
产品简介:mray-in-3 (12a) is a potent inhibitor of the bacterial translocase mray (ic50: 140 μm). 46 μg/ml)...产品型号:T64160 原产地:中国大陆价格: ¥0.0
产品名称: XIAP degrader-1;化合物 XIAP degrader-1XIAP degrader-1
产品简介:xiap degrader-1 is a small primary amine molecule that promotes the degradation of x-linked apoptosis inhibitory protein (xiap)...产品型号:T64161 原产地:中国大陆价格: ¥0.0
产品名称: AChE-IN-5;化合物 AChE-IN-5AChE-IN-5
产品简介:ache-in-5 (compound 5) is an orally active, blood-brain barrier-transparent substance with significant in vitro biological activity against ache/5-ht1a/sert. ic..产品型号:T64162 原产地:中国大陆价格: ¥0.0
产品名称: Aliskiren hydrochloride;化合物 Aliskiren hydrochlorideAliskiren hydrochloride
产品简介:aliskiren (cgp 60536; cgp60536b; spp 100) hydrochloride is a selective, orally active, renin inhibitor (ic50: 1.5 nm). cachexia...产品型号:T64163 原产地:中国大陆价格: ¥0.0
产品名称: Topoisomerase II inhibitor 11;化合物 Topoisomerase II inhibitor 11Topoisomerase II inhibitor 11
产品简介:topoisomerase ii inhibitor 11 (compound 3d) is a potent inhibitor of topoisomerase ii (ic50: 2.89 μm). topoisomerase ii inhibitor 11 inhibits cell proliferation..产品型号:T64164 原产地:中国大陆价格: ¥0.0
产品名称: Gln-AMS TFA;化合物 Gln-AMS TFAGln-AMS TFA
产品简介:gln-ams (tfa) is a type ia amido-trna synthetase (aars) inhibitor with a ki value of 1.32 μm for glutaminyl-trna synthetase...产品型号:T64165 原产地:中国大陆价格: ¥0.0
产品名称: Antiviral agent 20;化合物 Antiviral agent 20Antiviral agent 20
产品简介:antiviral agent 20 (compound 17b) is a selective inhibitor of zika virus (ec50: 4.5 μm) and exhibits low cytotoxicity...产品型号:T64166 原产地:中国大陆价格: ¥0.0