联系我们
产品目录
产品展示/Products
产品名称: Ifebemtinib;化合物 IfebemtinibIN-10018|||BI-853520;IN-10018|||BI-853520
产品简介:ifebemtinib (bi-853520) is an orally active and potent inhibitor of adhesion plaque kinase (fak) (ic50=1 nm) with anti-tumour activity that inhibits globule for..产品型号:T64167 原产地:中国大陆价格: ¥0.0
产品名称: EGFR-IN-18;化合物 EGFR-IN-18EGFR-IN-18
产品简介:egfr-in-18 is a potent inhibitor of the enzymatic activity of the l858r/t790m/c797s mutant egfr (4.9 nm) and is also able to reduce the enzymatic activity of wi..产品型号:T64170 原产地:中国大陆价格: ¥0.0
产品名称: LXR antagonist 2;化合物 LXR antagonist 2LXR antagonist 2
产品简介:lxr antagonist 2 (compound 10rr) is a potent lxr (liver x receptor) inverse agonist, acting on lxrβ (ic50: 0.36 μm) and lxrα (ic50: 2.25 μm). lxr antagonist 2 i..产品型号:T64171 原产地:中国大陆价格: ¥0.0
产品名称: Epocholeone;化合物 EpocholeoneEpocholeone
产品简介:epocholeone is a growth regulator and can be used for the control of fungal or physiological diseases of crops...产品型号:T64173 原产地:中国大陆价格: ¥0.0
产品名称: Cobimetinib hemifumarate;化合物 Cobimetinib hemifumarateCobimetinib hemifumarate
产品简介:cobimetinib hemifumarate is a potent and selective mek1 inhibitor with an ic50 value of 4.2 nm for mek1...产品型号:T64175 原产地:中国大陆价格: ¥0.0
产品名称: Vandetanib trifluoroacetate;化合物 Vandetanib trifluoroacetateVandetanib trifluoroacetate
产品简介:vandetanib trifluoroacetate (d6474 trifluoroacetate) is an orally active and potent vegfr2/kdr tyrosine kinase inhibitor with an ic50 value of 40 nm. vandetanib..产品型号:T64176 原产地:中国大陆价格: ¥0.0
产品名称: VGD071;化合物 VGD071VGD071
产品简介:vgd071, a compound that targets sortilin, presents a promising avenue for forthcoming research utilizing mouse models of breast cancer...产品型号:T64206 原产地:中国大陆价格: ¥0.0
产品名称: FAK-IN-6;化合物 FAK-IN-6FAK-IN-6
产品简介:fak-in-6 is a potent inhibitor of fak (ic50: 1.415 nm). fak-in-6 exhibits anti-proliferative effects on certain cancer cell lines and can be used to study pancr..产品型号:T64207 原产地:中国大陆价格: ¥0.0
产品名称: EZH2-IN-9;化合物 EZH2-IN-9EZH2-IN-9
产品简介:ezh2-in-9 is a potent inhibitor of ezh2, whose overexpression or mutations in the set region (y641f, y641n, a687v, a677g point mutations) cause abnormal elevati..产品型号:T64208 原产地:中国大陆价格: ¥0.0
产品名称: Anticancer agent 55;化合物 Anticancer agent 55Anticancer agent 55
产品简介:anticancer agent is a potent anti-cancer agent that exhibits anti-cancer effects by inhibiting cell viability and cell migration in a dose-dependent manner and ..产品型号:T64209 原产地:中国大陆价格: ¥0.0
产品名称: BRD73954;化合物BRD73954BRD73954
产品简介:brd73954, an effective and specific hdac inhibitor, which is with ic50 of 36 nm and 120 nm for hdac6 and hdac8, respectively...产品型号:T6421 原产地:中国大陆价格: ¥0.0
产品名称: ATX inhibitor 13;化合物 ATX inhibitor 13ATX inhibitor 13
产品简介:atx inhibitor 13 (compound 10c) is an orally active atx inhibitor (ic50: 3.4 nm). atx inhibitor 13 is capable of blocking the cell cycle of raw264.7 cells in th..产品型号:T64210 原产地:中国大陆价格: ¥0.0
产品名称: GLS1 Inhibitor-3;化合物 GLS1 Inhibitor-3GLS1 Inhibitor-3
产品简介:gls1 inhibitor-3 (compound c147) is a potent inhibitor of gls1 (ic50: 27.98 nm) and exhibits anti-proliferative effects...产品型号:T64211 原产地:中国大陆价格: ¥0.0
产品名称: Antiproliferative agent-5;化合物 Antiproliferative agent-5Antiproliferative agent-5
产品简介:antiproliferative agent-5 (compound 4o) irreversibly and significantly inhibits the proliferation of gastric cancer cells. antiproliferative agent-5 blocks the ..产品型号:T64212 原产地:中国大陆价格: ¥0.0
产品名称: Cap-dependent endonuclease-IN-3;化合物 Cap-dependent endonuclease-IN-3Cap-dependent endonuclease-IN-3
产品简介:cap-dependent endonuclease-in-3 is a potent inhibitor of cap-dependent nucleic acid endonucleases (cen). cap-dependent endonuclease-in-3 has shown potential for..产品型号:T64213 原产地:中国大陆价格: ¥0.0
产品名称: NXPZ-2;化合物 NXPZ-2NXPZ-2
产品简介:nxpz-2 is an orally active keap1-nrf2protein-protein interaction (ppi) inhibitor (ki: 95 nm, ec50: 120 and 170 nm). nxpz-2 dose-dependently attenuates aβ[1-42]-..产品型号:T64214 原产地:中国大陆价格: ¥0.0
产品名称: TAK-960 hydrochloride;化合物 TAK-960 hydrochlorideTAK-960 hydrochloride
产品简介:tak-960 hydrochloride is a potent, selective, orally active inhibitor of polo-like kinase 1 (plk1) (ic50: 0.8 nm). tak-960 hydrochloride inhibits the proliferat..产品型号:T64216 原产地:中国大陆价格: ¥0.0
产品名称: SM-433 hydrochloride;化合物 SM-433 hydrochlorideSM-433 hydrochloride
产品简介:sm-433 hydrochlorid is a smac mimetic, an inhibitor of inhibitory apoptosis proteins (iaps). sm-433 hydrochlorid is able to bind xiap bir3 protein with a potent..产品型号:T64217 原产地:中国大陆价格: ¥0.0
产品名称: Keap1-Nrf2-IN-1 TFA;化合物 Keap1-Nrf2-IN-1 TFAKeap1-Nrf2-IN-1 TFA
产品简介:keap1-nrf2-in-1 tfa (compound35) is a keap1-nrf2 protein-protein interaction inhibitor (ic50: 43 nm) that activates nrf2-regulated cytoprotective responses. kea..产品型号:T64218 原产地:中国大陆价格: ¥0.0
产品名称: PI3K/mTOR Inhibitor-6;化合物 PI3K/mTOR Inhibitor-6PI3K/mTOR Inhibitor-6
产品简介:pi3k/mtor inhibitor-6 (compound 19c) is a potent dual pi3k/mtor inhibitor that is more stable than gedatolisib in artificial gastric fluid. 10 μm of pi3k/mtor i..产品型号:T64219 原产地:中国大陆价格: ¥0.0