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产品名称: Verosudil;化合物VerosudilAR-12286;AR-12286
产品简介:verosudil (ar-12286) is a highly potent rho kinase (rock) inhibitor with a ki of 2 and 2 nm against rock1 and rock2, respectively. ar-12286 reverses steroid-ind..产品型号:T60924 原产地:中国大陆价格: ¥0.0
产品名称: AR524;化合物 AR524AR524
产品简介:ar524 is a transgenic inhibitor with higher inhibitory activity than the known transgenic inhibitor kifunensine. ar524 inhibits the formation of human malignant..产品型号:T62198 原产地:中国大陆价格: ¥0.0
产品名称: A1/A3 AR antagonist 1;化合物 A1/A3 AR antagonist 1A1/A3 AR antagonist 1
产品简介:a1/a3 ar antagonist 1 (compound 10) is a potent, dual adenosine 1 (a1) and adenosine 3 (a3) receptor antagonist that acts on human a1 (ki: 37.6 nm), human a3 (k..产品型号:T62134 原产地:中国大陆价格: ¥0.0
产品名称: AR antagonist 2;化合物 AR antagonist 2AR antagonist 2
产品简介:ar antagonist 2 (compound 58) is a potent inhibitor of the androgen receptor (ar) (ic50: 0.95 μm)...产品型号:T63030 原产地:中国大陆价格: ¥0.0
产品名称: β2AR/M-receptor agonist-1;化合物 β2AR/M-receptor agonist-1β2AR/M-receptor agonist-1
产品简介:β2ar/m-receptor agonist-1 (example 131), a muscarinic antagonist and β2 adrenoceptor agonist (maba), exhibits dual potency towards β2 adrenoceptor and muscarini..产品型号:T74708 原产地:中国大陆价格: ¥0.0
产品名称: (3aR,9aR)-Fluparoxan;化合物(3aR, 9aR)-Fluparoxan(3aR,9aR)-Fluparoxan
产品简介:(3ar,9ar)-fluparoxan is a highly selective and potent adrenergic receptor α2b antagonist for the prevention, amelioration or treatment of neurodevelopmental dis..产品型号:T77566 原产地:中国大陆价格: ¥0.0
产品名称: cis-ent-Tadalafil;他达拉非EP杂质C(6S,12aR)-Tadalafil|||Tadalafil, (6S,12aR)-|||cis-ent-IC-351;(6S,12aR)-Ta
产品简介:cis-ent-tadalafil (cis-ent-ic-351) is a potent and selective pde5 inhibitor that lowers blood pressure. cis-ent-tadalafil is a potent and selective pde5 inhibit..产品型号:T78216 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC AR-NTD degrader 1;化合物 PROTAC AR-NTD degrader 1PROTAC AR-NTD degrader 1
产品简介:protac ar-ntd antagonist 1 (compound 18) is a small molecule belonging to the protein-targeting chimeras (protacs) that selectively targets the n-terminal domai..产品型号:T78811 原产地:中国大陆价格: ¥0.0
产品名称: A1/A3 AR antagonist 3;化合物 A1/A3 AR antagonist 3A1/A3 AR antagonist 3
产品简介:a1/a3 ar antagonist 3 is a dual a1r/a3r antagonist that demonstrates high affinity within the low-micromolar to nanomolar range, and is potentially useful in th..产品型号:T79027 原产地:中国大陆价格: ¥0.0
产品名称: A3AR agonist 1;化合物 A3AR agonist 1A3AR agonist 1
产品简介:a3ar agonist 1 (compound 12), with a ki of 25.8 nm, is a potent a3 adenosine receptor (a3ar) agonist that promotes β-arrestin2 recruitment with an effective con..产品型号:T79372 原产地:中国大陆价格: ¥0.0
产品名称: A3AR agonist 2;化合物 A3AR agonist 2A3AR agonist 2
产品简介:compound 19, a selective a3 adenosine receptor (a3ar) agonist (k i : 22.1 nm), effectively stimulates β-arrestin2 recruitment with an ec 50 value of 4.36 nm. th..产品型号:T79373 原产地:中国大陆价格: ¥0.0
产品名称: α1A-AR Degrader 9c;化合物 α1A-AR Degrader 9cα1A-AR Degrader 9c
产品简介:α1a-ar degrader 9c is a potent, selective, and reversible protac degrader targeting the α1a adrenergic receptor (α1a-ar) with a dc50 of 2.86 μm. it promotes the..产品型号:T74557 原产地:中国大陆价格: ¥0.0
产品名称: A2A/A3u00A0AR antagonist-1;化合物 A2A/A3u00A0AR antagonist-1A2A/A3u00A0AR antagonist-1
产品简介:compound 23, designated as a2a/a3 ar antagonist-1, is a dual fluorescent ligand targeting a2a and a3 adenosine receptors (ar), exhibiting dissociation constants..产品型号:T74606 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC AR-V7 degrader-1;化合物 PROTAC AR-V7 degrader-1PROTAC AR-V7 degrader-1
产品简介:protac ar-v7 degrader-1 (compound 6) is an orally bioavailable, potent, and selective degrader targeting the androgen receptor (ar) variant v7, achieving degrad..产品型号:T74410 原产地:中国大陆价格: ¥0.0
产品名称: A3AR modulator 1;化合物 A3AR modulator 1A3AR modulator 1
产品简介:a3ar modulator 1 (mrs8054), an orally active positive allosteric modulator (pam) of the a3 adenosine receptor (a3ar) (adenosine receptor), significantly enhance..产品型号:T74993 原产地:中国大陆价格: ¥0.0
产品名称: Mca-PLGL-Dpa-AR-NH2;化合物 Mca-PLGL-Dpa-AR-NH2Mca-PLGL-Dpa-AR-NH2
产品简介:mca-plgl-dpa-ar-nh2 is a fluorescent peptide mmp substrate [1] ...产品型号:T76267 原产地:中国大陆价格: ¥0.0
产品名称: C5aR1 antagonist peptide;化合物 C5aR1 antagonist peptideC5aR1 antagonist peptide
产品简介:c5ar1 antagonist peptide, a biologically active linear peptide originating from the c-terminus of the chemokine complement fragment 5 anaphylatoxin (c5a), inhib..产品型号:T82797 原产地:中国大陆价格: ¥0.0
产品名称: Mca-KPLGL-Dap(Dnp)-AR-NH2 TFA;化合物 Mca-KPLGL-Dap(Dnp)-AR-NH2 TFAMca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-N
产品简介:mca-kplgl-dap(dnp)-ar-nh2 serves as a fluorogenic substrate specifically designed for matrix metalloproteinases (mmps). this compound facilitates the quantifica..产品型号:T83708 原产地:中国大陆价格: ¥0.0
产品名称: (4R,4aS,5aS,6aR,6bS,7aR)-4-Hydroxy-3,6b-dimethyl-5-methylene-4,4a,5,5a,6,6a,7,7a-octahydrocyclopropa
产品简介:(4r,4as,5as,6ar,6bs,7ar)-4-hydroxy-3,6b-dimethyl-5-methylene-4,4a,5,5a,6,6a,7,7a-octahydrocyclopropa[2,3]indeno[5,6-b]furan-2(6bh)-one is a sesquiterpene lacton..产品型号:T83554 原产地:中国大陆价格: ¥0.0
产品名称: (Z)-(1R,3R,4R,4aS,8R,8aR)-3,4,8,8a-Tetramethyl-7-oxo-4-(2-(5-oxo-2,5-dihydrofuran-3-yl)ethyl)decahyd
产品简介:compound 7a, (z)-(1r,3r,4r,4as,8r,8ar)-3,4,8,8a-tetramethyl-7-oxo-4-(2-(5-oxo-2,5-dihydrofuran-3-yl)ethyl)decahydronaphthalen-1-yl 2-methylbut-2-enoate, is a cl..产品型号:T83517 原产地:中国大陆价格: ¥0.0