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产品目录

产品展示/Products

  • HDAC1/2 and CDK2-IN-1;化合物 HDAC1/2 and CDK2-IN-1HDAC1/2 and CDK2-IN-1

    产品名称: HDAC1/2 and CDK2-IN-1;化合物 HDAC1/2 and CDK2-IN-1HDAC1/2 and CDK2-IN-1

    产品简介:hdac1/2 and cdk2-in-1 (compound 14d) are potent inhibitors of hdac1, hdac2 and cdk2 with ic50 values of 70.7, 23.1 and 0.80 μm, respectively. hdac1/2 and cdk2-i..

    产品型号:T63209 原产地:中国大陆价格: ¥0.0

  • HDAC-IN-45;化合物 HDAC-IN-45HDAC-IN-45

    产品名称: HDAC-IN-45;化合物 HDAC-IN-45HDAC-IN-45

    产品简介:hdac-in -45, a small molecule hdac inhibitor, was able to form hydrogen bonds with y303 residues and exhibited anticancer effects. hdac-in-45 significantly inhi..

    产品型号:T63422 原产地:中国大陆价格: ¥0.0

  • Tubacin;HDAC6 抑制剂Tubacin

    产品名称: Tubacin;HDAC6 抑制剂Tubacin

    产品简介:tubacin is a highly potent and selective, reversible, cell-permeable hdac6 inhibitor with an ic50 of 4 nm, approximately 350-fold selectivity over hdac1...

    产品型号:T6327 原产地:中国大陆价格: ¥0.0

  • mTOR/HDAC-IN-1;化合物 mTOR/HDAC-IN-1mTOR/HDAC-IN-1

    产品名称: mTOR/HDAC-IN-1;化合物 mTOR/HDAC-IN-1mTOR/HDAC-IN-1

    产品简介:mtor/hdac-in-1 (compound 50) is a dual inhibitor targeting both mtor and hdac with respective ic50 values of 0.49 nm and 0.91 nm. it holds potential as an anti-..

    产品型号:T63399 原产地:中国大陆价格: ¥0.0

  • mTOR/HDAC-IN-1 HCl;mTOR/HDAC抑制剂1盐酸盐mTOR/HDAC-IN-1 HCl(2815286-02-1 Free base);mTOR/HDAC-IN-1 HCl(281

    产品名称: mTOR/HDAC-IN-1 HCl;mTOR/HDAC抑制剂1盐酸盐mTOR/HDAC-IN-1 HCl(2815286-02-1 Free base);mTOR/HDAC-IN-1 HCl(281

    产品简介:mtor/hdac-in-1 hcl is a potent dual inhibitor of mtor and hdac with potential anti-inflammatory, anti-proliferative, autophagy and apoptosis-inducing effects fo..

    产品型号:T63399L 原产地:中国大陆价格: ¥0.0

  • HDAC-IN-39;化合物 HDAC-IN-39HDAC-IN-39

    产品名称: HDAC-IN-39;化合物 HDAC-IN-39HDAC-IN-39

    产品简介:hdac-in-39 is a potent inhibitor of hdac and is able to act on hdac1, hdac2 and hdac3 with ic50 values of 1.07 μm, 1.47 μm and 2.27 μm, respectively. hdac-in-39..

    产品型号:T63416 原产地:中国大陆价格: ¥0.0

  • HDAC6-IN-3;化合物 HDAC6-IN-3HDAC6-IN-3

    产品名称: HDAC6-IN-3;化合物 HDAC6-IN-3HDAC6-IN-3

    产品简介:hdac6-in-3 (compound 14) is a potent anti-prostate cancer agent that acts as an orally active inhibitor of hdac6. it has ic50 values ranging from 0.02-1.54 μm f..

    产品型号:T61139 原产地:中国大陆价格: ¥0.0

  • HDAC-IN-27;化合物 HDAC-IN-27HDAC-IN-27

    产品名称: HDAC-IN-27;化合物 HDAC-IN-27HDAC-IN-27

    产品简介:hdac-in-27 是一种有效的口服活性 hdac i 类选择性抑制剂,对 hdac1-3 的 ic 50 值范围为 0.43 至 3.01 nm。抗急性髓系白血病 (aml) 活性。..

    产品型号:T61209 原产地:中国大陆价格: ¥0.0

  • HDAC1/MAO-B-IN-1;化合物 HDAC1/MAO-B-IN-1HDAC1/MAO-B-IN-1

    产品名称: HDAC1/MAO-B-IN-1;化合物 HDAC1/MAO-B-IN-1HDAC1/MAO-B-IN-1

    产品简介:hdac1/mao-b-in-1 has the potential to be used in the alzheimer’s disease research. hdac1/mao-b-in-1 is a potent and selective inhibitor of hdac1/mao-b that can ..

    产品型号:T60947 原产地:中国大陆价格: ¥0.0

  • HDAC6-IN-6;化合物 HDAC6-IN-6HDAC6-IN-6

    产品名称: HDAC6-IN-6;化合物 HDAC6-IN-6HDAC6-IN-6

    产品简介:hdac6-in-6 (compound 6a) is a potent inhibitor of hdac6 that can penetrate bbb with an ic50 value of 0.025 μm. hdac6-in-6 has potent inhibitory activity against..

    产品型号:T60954 原产地:中国大陆价格: ¥0.0

  • HDAC6-IN-11;化合物 HDAC6-IN-11HDAC6-IN-11

    产品名称: HDAC6-IN-11;化合物 HDAC6-IN-11HDAC6-IN-11

    产品简介:hdac6-in-11 (compound 9) has anti-proliferative activities against cancer cells. hdac6-in-11 is a selective inhibitor of hdac6 with the ic50 value of 20.7 nm. t..

    产品型号:T61044 原产地:中国大陆价格: ¥0.0

  • HDAC-IN-47;化合物 HDAC-IN-47HDAC-IN-47

    产品名称: HDAC-IN-47;化合物 HDAC-IN-47HDAC-IN-47

    产品简介:hdac-in-47 is an orally active histone deacetylase (hdac) inhibitor with ic50 values of 19.75 nm, 57.8 nm, 40.27 nm, 5.63 nm and 302.73 nm for hdac1, hdac2, hda..

    产品型号:T62072 原产地:中国大陆价格: ¥0.0

  • HDAC-IN-31;化合物 HDAC-IN-31HDAC-IN-31

    产品名称: HDAC-IN-31;化合物 HDAC-IN-31HDAC-IN-31

    产品简介:hdac-in-31 is a selective, potent, orally active hdac inhibitor that acts on hdac1 (ic50: 84.90 nm), hdac2 (ic50: 168.0 nm), hdac3 (ic50: 442.7 nm), hdac8 (ic50..

    产品型号:T62109 原产地:中国大陆价格: ¥0.0

  • HDAC6-IN-5;化合物 HDAC6-IN-5HDAC6-IN-5

    产品名称: HDAC6-IN-5;化合物 HDAC6-IN-5HDAC6-IN-5

    产品简介:hdac6-in-5 (compound 11b) is a potent and bbb-penetrated inhibitor of hdac6 (ic50= 0.025 μm). hdac6-in-5 inhibits aβ 1-42 self-aggregation and ache, with ic 50s..

    产品型号:T62046 原产地:中国大陆价格: ¥0.0

  • HDAC8/BRPF1-IN-1;化合物 HDAC8/BRPF1-IN-1HDAC8/BRPF1-IN-1

    产品名称: HDAC8/BRPF1-IN-1;化合物 HDAC8/BRPF1-IN-1HDAC8/BRPF1-IN-1

    产品简介:hdac8/brpf1-in-1 (compound 23a) is a dual hdac8 and brpf1 inhibitor that acts on human hdac8 (ic50: 443 nm) and human brpf1 (kd: 67 nm). hdac8/brpf1-in-1 has lo..

    产品型号:T62171 原产地:中国大陆价格: ¥0.0

  • PI3K/HDAC-IN-2;化合物 PI3K/HDAC-IN-2PI3K/HDAC-IN-2

    产品名称: PI3K/HDAC-IN-2;化合物 PI3K/HDAC-IN-2PI3K/HDAC-IN-2

    产品简介:pi3k/hdac-in-2 is a potent dual pi3k/hdac inhibitor, capable of acting on pi3kα (ic50: 226 nm), pi3kβ (ic50: 279 nm), pi3kγ (ic50: 467 nm), pi3kδ (ic50: 29 nm),..

    产品型号:T62912 原产地:中国大陆价格: ¥0.0

  • HDAC-IN-38;化合物 HDAC-IN-38HDAC-IN-38

    产品名称: HDAC-IN-38;化合物 HDAC-IN-38HDAC-IN-38

    产品简介:hdac-in-38 is a potent inhibitor of hdac. hdac-in-38 has similar micromolar inhibitory effects on hdac1, 2, 3, 5, 6 and 8, and also increases histone acetylatio..

    产品型号:T62920 原产地:中国大陆价格: ¥0.0

  • AChE/HDAC-IN-1;化合物 AChE/HDAC-IN-1AChE/HDAC-IN-1

    产品名称: AChE/HDAC-IN-1;化合物 AChE/HDAC-IN-1AChE/HDAC-IN-1

    产品简介:cox-2-in-23 (compound a10) is a potent inhibitor of ache (ic50: 0.12 nm) and hdac (ic50: 0.23 nm).cox-2-in-23 exhibits antioxidant and metal chelating propertie..

    产品型号:T63142 原产地:中国大陆价格: ¥0.0

  • Top/HDAC-IN-2;化合物 Top/HDAC-IN-2Top/HDAC-IN-2

    产品名称: Top/HDAC-IN-2;化合物 Top/HDAC-IN-2Top/HDAC-IN-2

    产品简介:top/hdac-in-2 (45b) is a dual inhibitor of top and hdac that induces apoptosis and exhibits significant anti-tumour effects...

    产品型号:T64025 原产地:中国大陆价格: ¥0.0

  • CYP51/HDAC-IN-1;化合物 CYP51/HDAC-IN-1CYP51/HDAC-IN-1

    产品名称: CYP51/HDAC-IN-1;化合物 CYP51/HDAC-IN-1CYP51/HDAC-IN-1

    产品简介:cyp51/hdac-in-1 is an orally active, potent, dual cyp51/hdac inhibitor that inhibits important virulence factors and down-regulates the expression of associated..

    产品型号:T64154 原产地:中国大陆价格: ¥0.0

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