联系我们
产品目录
产品展示/Products
产品名称: PROTAC HDAC6 degrader 1;化合物 PROTAC HDAC6 degrader 1PROTAC HDAC6 degrader 1
产品简介:compound a6, a potent and selective protac hdac6 degrader, exhibits a dc50 of 3.5 nm. it demonstrates notable antiproliferative activity by inducing apoptosis i..产品型号:T75017 原产地:中国大陆价格: ¥0.0
产品名称: HDAC6 degrader-3;化合物 HDAC6 degrader-3HDAC6 degrader-3
产品简介:hdac6 degrader-3, a selective and potent degrader of hdac6 through ternary complex formation and the ubiquitin-proteasome pathway, exhibits a dc50 value of 19.4..产品型号:T75018 原产地:中国大陆价格: ¥0.0
产品名称: HDAC-IN-57;化合物HDAC-IN-57HDAC-IN-57
产品简介:hdac-in-57 is an orally active pan-inhibitor of histone deacetylase (hdac), inhibiting hdac1, hdac2, hdac6, and hdac8 with ic50 values of 2.07 nm, 4.71 nm, 2.4 ..产品型号:T77334 原产地:中国大陆价格: ¥0.0
产品名称: HDAC6 degrader-1;化合物 HDAC6 degrader-1HDAC6 degrader-1
产品简介:hdac6 degrader-1, a proteolysis-targeting chimeric molecule (protac), incorporates the selective hdac6 inhibitor nexturastat a (nex a) for hdac6 binding, a link..产品型号:T77922 原产地:中国大陆价格: ¥0.0
产品名称: HDAC-IN-55;化合物 HDAC-IN-55HDAC-IN-55
产品简介:hdac-in-55(8j) is a small-molecule inhibitor that enhances e-cadherin expression and suppresses cancer cell proliferation [1]...产品型号:T78532 原产地:中国大陆价格: ¥0.0
产品名称: JAK/HDAC-IN-2;化合物 JAK/HDAC-IN-2JAK/HDAC-IN-2
产品简介:jak/hdac-in-2, a potent 2-amino-4-phenylaminopyrimidine dual-target inhibitor, effectively suppresses jak1/2 and hdac3/6 at nanomolar concentrations. this compo..产品型号:T78708 原产地:中国大陆价格: ¥0.0
产品名称: HDAC8-IN-4;化合物 HDAC8-IN-4HDAC8-IN-4
产品简介:hdac8-in-4 is a selective hdac8 inhibitor, exhibiting inhibitory activity with ic50 values of 0.15 μm for hdac8 and 12 μm for hdac3 [1]...产品型号:T79082 原产地:中国大陆价格: ¥0.0
产品名称: PI3Kα/HDAC6-IN-1;化合物 PI3Kα/HDAC6-IN-1PI3Kα/HDAC6-IN-1
产品简介:pi3kα/hdac6-in-1 (compound 21j) is a dual inhibitor of pi3kα and hdac6, exhibiting ic50 values of 2.9 nm and 26 nm, respectively. it effectively hinders akt(ser..产品型号:T79710 原产地:中国大陆价格: ¥0.0
产品名称: JMJD3/HDAC-IN-1;化合物 JMJD3/HDAC-IN-1JMJD3/HDAC-IN-1
产品简介:compound a5b, also known as jmjd3/hdac-in-1, is a dual inhibitor that targets both jmjd3 (jumonji domain-containing protein demethylase 3) and hadc1 (histone de..产品型号:T79713 原产地:中国大陆价格: ¥0.0
产品名称: HDAC3-IN-2;化合物 HDAC3-IN-2HDAC3-IN-2
产品简介:hdac3-in-2 (compound 4i), a pyrazinyl hydrazide-based hdac3 inhibitor with an ic50 of 14 nm, effectively targets triple-negative breast cancer cells. demonstrat..产品型号:T79714 原产地:中国大陆价格: ¥0.0
产品名称: HDAC-IN-64;化合物 HDAC-IN-64HDAC-IN-64
产品简介:hdac-in-64 (compound 13), an hdac inhibitor, demonstrates potent inhibition of hdac4/5/6/7/9 with ic50 values of 24, 45, 85, 31, and 37 nm, respectively. it exh..产品型号:T79674 原产地:中国大陆价格: ¥0.0
产品名称: HDAC/CD13-IN-1;化合物 HDAC/CD13-IN-1HDAC/CD13-IN-1
产品简介:hdac/cd13-in-1 (compound 12) is an inhibitor of both hdac and cd13, with ic50 values of 0.34 μm for hcd13, 0.53 μm for porcine cd13, and 0.03, 0.06, and 0.02 μm..产品型号:T79683 原产地:中国大陆价格: ¥0.0
产品名称: HDAC/JAK/BRD4-IN-1;化合物 HDAC/JAK/BRD4-IN-1HDAC/JAK/BRD4-IN-1
产品简介:hdac/jak/brd4-in-1 (compound 25ap) is a potent triple inhibitor targeting hdac, jak, and brd4. this compound not only inhibits cell proliferation but also induc..产品型号:T79768 原产地:中国大陆价格: ¥0.0
产品名称: HDAC6-IN-23;化合物 HDAC6-IN-23HDAC6-IN-23
产品简介:hdac6-in-23 (compound 9), an orally active inhibitor of hdac6 [1], displays selective enzymatic inhibition...产品型号:T79769 原产地:中国大陆价格: ¥0.0
产品名称: HDAC6-IN-22;化合物 HDAC6-IN-22HDAC6-IN-22
产品简介:hdac6-in-22 (compound 30), an hdac6 inhibitor, exhibits an ic50 of 4.63 nm and demonstrates antiproliferative effects against multiple myeloma both in vitro and..产品型号:T79771 原产地:中国大陆价格: ¥0.0
产品名称: VEGFR2/HDAC1-IN-1;化合物 VEGFR2/HDAC1-IN-1VEGFR2/HDAC1-IN-1
产品简介:vegfr2/hdac1-in-1 (compound 13) is a potent dual inhibitor of vegfr-2 and hdac, with ic50 values of 57.83 nm for vegfr-2 and 9.82 nm for hdac. it arrests the ..产品型号:T80873 原产地:中国大陆价格: ¥0.0
产品名称: HDAC6-IN-25;化合物 HDAC6-IN-25HDAC6-IN-25
产品简介:hdac6-in-25 (compound 8) is a potent and selective hdac6 inhibitor, exhibiting an ic50 value of 0.6 nm [1]...产品型号:T82224 原产地:中国大陆价格: ¥0.0
产品名称: HDAC6-IN-24;化合物 HDAC6-IN-24HDAC6-IN-24
产品简介:hdac6-in-24 (compound n1) is an inhibitor of histone deacetylase 6 (hdac6) [1]...产品型号:T82225 原产地:中国大陆价格: ¥0.0
产品名称: HDAC6-IN-21;化合物 HDAC6-IN-21HDAC6-IN-21
产品简介:hdac6-in-21 (compound 13) is an irreversible inhibitor of histone deacetylase 6 (hdac6) [1]...产品型号:T82226 原产地:中国大陆价格: ¥0.0
产品名称: HDAC1/CDK7-IN-1;化合物 HDAC1/CDK7-IN-1HDAC1/CDK7-IN-1
产品简介:hdac1/cdk7-in-1 (compound 8e) serves as a dual inhibitor targeting both cdk7 and hdac1, with ic50 values of 893 nm and 248 nm , respectively. this compound eff..产品型号:T82227 原产地:中国大陆价格: ¥0.0