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产品目录

产品展示/Products

  • AZD8055AZD8055

    产品名称: AZD8055AZD8055

    产品简介:azd8055 is an atp-competitive mtor inhibitor (ic50: 0.8 nm in mda-mb-468 cells). it is ~1,000-fold selective for mtor over all pi3k isoforms...

    产品型号:T1859 原产地:美洲价格: ¥0.0

  • AZD2932AZD2932

    产品名称: AZD2932AZD2932

    产品简介:azd2932 is a potent and multi-targeted kinase inhibitor vegfr2, pdgfβ, flt-3, and c-kit...

    产品型号:T1836 原产地:美洲价格: ¥0.0

  • AZD1080AZD1080

    产品名称: AZD1080AZD1080

    产品简介:azd1080 is a selective, orally active, brain permeable gsk3 inhibitor...

    产品型号:T1741 原产地:美洲价格: ¥0.0

  • CapivasertibCapivasertib,AZD5363,

    产品名称: CapivasertibCapivasertib,AZD5363,

    产品简介:capivasertib (azd5363) is a new-type orally available inhibitor of the serine/threonine protein kinase akt (ic50s: 3/7/7 nm for akt1/2/3)...

    产品型号:T1920 原产地:美洲价格: ¥0.0

  • AZD4547AZD4547

    产品名称: AZD4547AZD4547

    产品简介:azd4547, a new-type specific fgfr inhibitor, targets for fgfr1/2/3 (ic50: 0.2/2.5/1.8 nm in cell-free assays)...

    产品型号:T1948 原产地:美洲价格: ¥0.0

  • VistusertibVistusertib,AZD2014,

    产品名称: VistusertibVistusertib,AZD2014,

    产品简介:azd2014 is an orally bioavailable inhibitor of the mammalian target of rapamycin (mtor) with potential antineoplastic activity...

    产品型号:T1961 原产地:美洲价格: ¥0.0

  • AZD2858AZD2858

    产品名称: AZD2858AZD2858

    产品简介:azd2858 is a selective gsk-3 inhibitor, inhibiting tau phosphorylation at the s396 site and activating wnt signaling pathway...

    产品型号:T1957 原产地:美洲价格: ¥0.0

  • AZD5438AZD5438

    产品名称: AZD5438AZD5438

    产品简介:azd5438 is an effective inhibitor of cdk, for cdk1(ic50=16 nm),cdk2(ic50=6 nm),cdk9(ic50=20 nm)...

    产品型号:T2506 原产地:美洲价格: ¥0.0

  • CediranibCediranib,AZD2171,NSC-732208

    产品名称: CediranibCediranib,AZD2171,NSC-732208

    产品简介:cediranib (azd2171) is a highly potent (ic50 < 1 nmol/l) atp-competitive inhibitor of recombinant kdr tyrosine kinase in vitro, also inhibits flt1/4 (ic50: 5 nm..

    产品型号:T2500 原产地:美洲价格: ¥0.0

  • BarasertibBarasertib,1H-Pyrazole-3-acetamide,AZD1152-HQPA

    产品名称: BarasertibBarasertib,1H-Pyrazole-3-acetamide,AZD1152-HQPA

    产品简介:barasertib (azd1152-hqpa) is a highly selective aurora b inhibitor (ic50: 0.37 nm) and demonstrates ~3,700-fold greater selectivity than aurora a...

    产品型号:T2602 原产地:美洲价格: ¥0.0

  • AZD1208AZD1208

    产品名称: AZD1208AZD1208

    产品简介:azd1208 is a novel, orally bioavailable, highly selective pim kinase inhibitor with single nanomolar potency against all three pim kinases...

    产品型号:T2300 原产地:美洲价格: ¥0.0

  • OsimertinibOsimertinib,Mereletinib,AZD-9291

    产品名称: OsimertinibOsimertinib,Mereletinib,AZD-9291

    产品简介:osimertinib is a small molecule tyrosine kinase receptor inhibitor and antineoplastic agent that is used in the therapy of selected forms of advanced non-small ..

    产品型号:T2490 原产地:美洲价格: ¥0.0

  • AZD2461AZD2461

    产品名称: AZD2461AZD2461

    产品简介:azd2461 is a novel parp inhibitor...

    产品型号:T2484 原产地:美洲价格: ¥0.0

  • AZD7545AZD7545

    产品名称: AZD7545AZD7545

    产品简介:azd7545 is a potent pdhk inhibitor...

    产品型号:T2447 原产地:美洲价格: ¥0.0

  • AdavosertibAdavosertib,MK-1775,AZD1775

    产品名称: AdavosertibAdavosertib,MK-1775,AZD1775

    产品简介:mk-1775 is a small molecule inhibitor of the checkpoint kinase wee1 (ic50: 5.2 nm). it hinders the g2 dna damage checkpoint...

    产品型号:T2077 原产地:美洲价格: ¥0.0

  • AZD3229AZD3229

    产品名称: AZD3229AZD3229

    产品简介:azd3229 is a potent pan-kit mutant inhibitor for the treatment of gastrointestinal stromal tumors. it demonstrates potent single-digit nm growth inhibition acro..

    产品型号:T5409 原产地:美洲价格: ¥0.0

  • azd1390azd1390

    产品名称: azd1390azd1390

    产品简介:azd1390 is an exceptionally potent inhibitor of atm in cells (ic50: 0.78 nm) with >10,000-fold selectivity over closely related members of the pikk family of en..

    产品型号:T5175 原产地:美洲价格: ¥0.0

  • AZD8330AZD8330,ARRY-704,ARRY-424704

    产品名称: AZD8330AZD8330,ARRY-704,ARRY-424704

    产品简介:azd8330 is a novel, selective, non-atp competitive mek 1/2 inhibitor with ic50 of 7 nm. phase 1...

    产品型号:T6083 原产地:美洲价格: ¥0.0

  • SaracatinibSaracatinib,AZD0530,

    产品名称: SaracatinibSaracatinib,AZD0530,

    产品简介:saracatinib (azd0530) is an effective src inhibitor (ic50: 2.7 nm), and effective to lck, fyn, lyn, blk, fgr and c-yes...

    产品型号:T6078 原产地:美洲价格: ¥0.0

  • SelumetinibSelumetinib,ARRY-142886,AZD6244

    产品名称: SelumetinibSelumetinib,ARRY-142886,AZD6244

    产品简介:selumetinib (azd6244) is an effective, specific inhibitor of mek1 and erk1/2 phosphorylation (ic50: 14/10 nm)...

    产品型号:T6218 原产地:美洲价格: ¥0.0

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