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产品名称: AZD3514AZD3514
产品简介:azd3514 is a potent and oral androgen receptor downregulator with ki of 2.2 μm and has ability of reducing ar protein expression.phase 1...产品型号:T6400 原产地:美洲价格: ¥0.0
产品名称: AZD1981AZD1981
产品简介:azd1981 is an effective and specific crth2 (dp2) receptor antagonist (ic50: 4 nm), showing >1000-fold selectivity over more than 340 other enzymes and receptors..产品型号:T6399 原产地:美洲价格: ¥0.0
产品名称: AZD7762AZD7762
产品简介:azd7762, an effective and specific inhibitor of chk1(ic50=5 nm), is equally potent against chk2 and less potent against cam, yes, fyn, lyn, hck and lck...产品型号:T6093 原产地:美洲价格: ¥0.0
产品名称: SapitinibSapitinib,AZD-8931,
产品简介:azd8931, a reversible, atp competitive inhibitor of egfr(ic50=4 nm), erbb2(ic50=3 nm) and erbb3(ic50=4 nm), is more effective over gefitinib or lapatinib agains..产品型号:T6092 原产地:美洲价格: ¥0.0
产品名称: AZD6482AZD6482,KIN 193,
产品简介:azd 6482 is a potent and selective p110β inhibitor with ic50 of 0.69 nm and a pi3kβ inhibitor with ic50 of 10 nm...产品型号:T6087 原产地:美洲价格: ¥0.0
产品名称: AZD-8835;化合物AZD8835AZD8835;AZD8835
产品简介:azd-8835 is a mixed inhibitor of pi3kα/δ (ic50: 6.2/5.7 nm), also with selectivity against pi3kβ/γ (ic50: 431/90 nm)...产品型号:T6774 原产地:中国大陆价格: ¥0.0
产品名称: AZD8926;化合物 T30266AZD 8926|||AZD-8926;AZD 8926|||AZD-8926
产品简介:azd8926 is a potent and selective inhibitor of gsk3β(glycogen synthase kinase-3β). azd8926 is potential for treating alzheimer’s disease (ad), schizophrenia, an..产品型号:T30266 原产地:中国大陆价格: ¥0.0
产品名称: AZD9291-345;化合物 T30268AZD-9291345|||AZD 9291345|||AZD9291345;AZD-9291345|||AZD 9291345|||AZD9291345
产品简介:azd9291-345 is a compound which has a molecule weight 345, and structurally related to azd9291...产品型号:T30268 原产地:中国大陆价格: ¥0.0
产品名称: Olaparib;奥拉帕尼AZD2281|||KU0059436;AZD2281|||奥拉帕尼|||KU0059436
产品简介:olaparib (ku0059436) is a small molecule inhibitor of parp1/parp2 (ic50=5/1 nm), with weak inhibitory activity against parp tankyrase-1 (ic50=1.5 μm), and is se..产品型号:T3015 原产地:中国大陆价格: ¥0.0
产品名称: AZD-1305;化合物AZD-1305UNII-CZO834LXQM|||AZD 1305;UNII-CZO834LXQM|||AZD 1305
产品简介:azd-1305 is a novel anti-arrhythmic compound that primarily blocks the fast component of ikr, l-type calcium currents and intra-ward sodium currents in mammalia..产品型号:T30251 原产地:中国大陆价格: ¥0.0
产品名称: AZD-2327;化合物 T30254AZD-2327
产品简介:azd-2327 is a highly selective agonist of δ-opioid receptor, highly selective to human μ-and κ-opioid receptor subtypes (> 1000 times) and 130 other receptors a..产品型号:T30254 原产地:中国大陆价格: ¥0.0
产品名称: Osimertinib mesylate;奥希替尼甲磺酸盐Mereletinib mesylate|||AZD-9291 mesylate;甲磺酸奥希替尼|||Mereletinib mesylate
产品简介:osimertinib mesylate (mereletinib mesylate) is an irreversible and mutant selective egfr inhibitor (ic50s: 12/1 nm for egfr(l858r) and egfr(l858r/t790m))...产品型号:T3634 原产地:中国大陆价格: ¥0.0
产品名称: AZD 1152 (hydrochloride)AZD 1152 (hydrochloride)AZD 1152 (hydrochloride)
产品简介:azd 1152 is an orally bioavailable prodrug of azd 1152-hqpa, a selective inhibitor of aurora kinase b (ic50= 0.36 nm).1azd 1152 is converted to azd 1152-hqpa in..产品型号:T36199 原产地:中国大陆价格: ¥0.0
产品名称: AZD 3147;化合物AZD 3147AZD 3147
产品简介:azd 3147 is an inhibitor of mtorc with ic50s of 40.7 and 5.75 nm for mtorc1 and mtorc2. azd 3147 shows ic50s of 912, 5495, 9333, and 6310 nm for pi3kα, pi3kβ, p..产品型号:T36200 原产地:中国大陆价格: ¥0.0
产品名称: AZD5582 dihydrochloride;AZD 5582 dihydrochlorideAZD 5582 dihydrochloride;AZD 5582 dihydrochloride
产品简介:dimeric smac mimetic; potent inhibitor of x-linked (xiap) and cellular (ciap) inhibitor of apoptosis protein (ic50 values are 15, 15 and 21 nm for xiap, ciap1 a..产品型号:T36201 原产地:中国大陆价格: ¥0.0
产品名称: AZD5582 TFA;AZD5582 三氟乙酸盐AZD5582 TFA(1258392-53-8 free base);AZD5582 TFA(1258392-53-8 free ba
产品简介:azd5582 tfa is a potent iap antagonist that binds to the bir3 domain of ciap1, ciap2, and xiap with ic50 values of 15, 21, and 15 nm, respectively.azd5582 tfa..产品型号:T36201L 原产地:中国大陆价格: ¥0.0
产品名称: AZD4721;AZD4721RIST4721|||AZD4721;RIST4721|||AZD4721
产品简介:azd4721 (rist4721) is the potent and orally active antagonist of acidic cxc chemokine receptor 2 ( cxcr2 ). azd4721 has the potential for the research of inflam..产品型号:T38850 原产地:中国大陆价格: ¥0.0
产品名称: azd1390;化合物azd1390azd1390|||azd1390|||ATM/ATR|||azd-1390|||ATM and RAD3 related|||AZD 1390|||inhibit
产品简介:azd1390 is an exceptionally potent inhibitor of atm in cells (ic50: 0.78 nm) with >10,000-fold selectivity over closely related members of the pikk family of en..产品型号:T5175 原产地:中国大陆价格: ¥0.0
产品名称: AZD3965;化合物AZD3965AZD 3965|||AZD-3965;AZD 3965|||AZD-3965
产品简介:azd3965 (azd-3965) is a selective inhibitor of monocarboxylate transporter 1 (mct1)...产品型号:T3210 原产地:中国大陆价格: ¥0.0
产品名称: Linaprazan mesylate;化合物 T32760AZD-0865 mesilate|||AR-h044277AW|||Linaprazan mesilate|||AZD-0865 mesy
产品简介:linaprazan mesylate is a bio-active chemical...产品型号:T32760 原产地:中国大陆价格: ¥0.0