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产品名称: PROTAC TTK degrader-1;化合物 PROTAC TTK degrader-1PROTAC TTK degrader-1
产品简介:protac ttk degrader-1, a potent threonine tyrosine kinase (ttk) protac degrader, demonstrates dc50 values of 1.7 nm in colo-205 cells and 5.8 nm in hct-116 cell..产品型号:T81375 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC SMARCA2 degrader-2;化合物 PROTAC SMARCA2 degrader-2PROTAC SMARCA2 degrader-2
产品简介:protac smarca2 degrader-2, a selective and powerful degrader of smarca2/4, exhibits an ic50 of <0.1 μμ in the hela hibit assay.this compound holds promise for r..产品型号:T81376 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC NSD3 degrader-1;化合物 PROTAC NSD3 degrader-1PROTAC NSD3 degrader-1
产品简介:protac nsd3 degrader-1 (compound 56) is a targeted degradation agent for the nuclear receptor binding set domain protein nsd3. it effectively induces the degrad..产品型号:T81377 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC IRAK4 ligand-3;化合物 PROTAC IRAK4 ligand-3PROTAC IRAK4 ligand-3
产品简介:protac irak4 ligand-3 serves as a ligand for protac irak4 degrader-7 and is utilized in cancer research [1]...产品型号:T81378 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC GDI2 Degrader-1;化合物 PROTAC GDI2 Degrader-1PROTAC GDI2 Degrader-1
产品简介:protac gdi2 degrader-1 (compound 21) is a potent degrader of protac gdi2, demonstrating outstanding antitumor activity in vivo within pancreatic xenograft model..产品型号:T81379 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC EGFR degrader 7 diTFA;化合物 PROTAC EGFR degrader 7 diTFAPROTAC EGFR degrader 7 diTFA
产品简介:protac egfr degrader 7 (compound 13b) is a potent, selective, crbn-recruiting egfrl858r/t790m degrader with a dc50 of 13.2 nm. it effectively inhibits prolifera..产品型号:T81380 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC eDHFR Degrader-1;化合物 PROTAC eDHFR Degrader-1PROTAC eDHFR Degrader-1
产品简介:protac edhfr degrader-1 is a potent degrader targeting edhfr-yfp and various proteins of interest (pois), such as yfp and luciferase [1]...产品型号:T81381 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC BRD9 Degrader-7;化合物 PROTAC BRD9 Degrader-7PROTAC BRD9 Degrader-7
产品简介:protac brd9 degrader-7 is a selective and orally active brd9 degrader with a dc50 of 1.02 nm and demonstrates superior pharmacokinetics, evidenced by a cmax of ..产品型号:T81382 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC BRD9 Degrader-5;化合物 PROTAC BRD9 Degrader-5PROTAC BRD9 Degrader-5
产品简介:protac brd9 degrader-5 is a proteolysis targeting chimera (protac) designed for the specific degradation of bromodomain-containing protein 9 (brd9)...产品型号:T81383 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC BRD9 Degrader-3;化合物 PROTAC BRD9 Degrader-3PROTAC BRD9 Degrader-3
产品简介:protac brd9 degrader-3 is a bifunctional degrader targeting brd9, utilized in cancer research...产品型号:T81384 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC BRD9 Degrader-2;化合物 PROTAC BRD9 Degrader-2PROTAC BRD9 Degrader-2
产品简介:protac brd9 degrader-2 is a bifunctional compound designed for the targeted degradation of brd9 in cancer research applications...产品型号:T81385 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC BRD4 Degrader-22;化合物 PROTAC BRD4 Degrader-22PROTAC BRD4 Degrader-22
产品简介:protac brd4 degrader-22 (compd 44h) is a protac-based degrader targeting brd4, exhibiting a pdc50 of 9.2 in molt4 cells over 24 hours [1]...产品型号:T81386 原产地:中国大陆价格: ¥0.0
产品名称: BT-PROTAC;化合物 BT-PROTACBT-PROTAC
产品简介:bt-protac is a bioorthogonally activatable prodrug that enables precise control over protac (proteolysis targeting chimera) activity...产品型号:T82809 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC BRD4 Degrader-7;化合物 PROTAC BRD4 Degrader-7PROTAC BRD4 Degrader-7
产品简介:protac brd4 degrader-7, a potent bromodomain brd4 inhibitor exemplified by compound 1a, demonstrates half-maximal inhibitory concentrations (ic50s) of 15.5 nm a..产品型号:T74090 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC BRD4 Degrader-11;化合物 PROTAC BRD4 Degrader-11PROTAC BRD4 Degrader-11
产品简介:protac brd4 degrader-11 (compound 9a), a protac linked through ligands to von hippel-lindau and brd4, effectively targets and degrades the brd4 protein in pc3 p..产品型号:T74124 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC EGFR degrader 6;化合物 PROTAC EGFR degrader 6PROTAC EGFR degrader 6
产品简介:protac egfr degrader 6 is a potent protac egfr degrader that effectively reduces egfr del19 levels in hcc827 cells, exhibiting a dc50 of 45.2 nm. it notably pro..产品型号:T74525 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC_ERRα;化合物 PROTAC_ERRαPROTAC_ERRα
产品简介:protac_errα is a potent, selective degrader of errα, efficiently facilitating its proteasomal degradation. this compound specifically targets errα protein, achi..产品型号:T74559 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC EZH2 Degrader-1;化合物 PROTAC EZH2 Degrader-1PROTAC EZH2 Degrader-1
产品简介:protac ezh2 degrader-1 (compound 150d), a potent inhibitor, effectively suppresses ezh2 methyltransferase activity, demonstrating an ic50 of 2.7 nm. ezh2 is cru..产品型号:T74602 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC AR-V7 degrader-1;化合物 PROTAC AR-V7 degrader-1PROTAC AR-V7 degrader-1
产品简介:protac ar-v7 degrader-1 (compound 6) is an orally bioavailable, potent, and selective degrader targeting the androgen receptor (ar) variant v7, achieving degrad..产品型号:T74410 原产地:中国大陆价格: ¥0.0
产品名称: PROTAC IRAK4 degrader-7;化合物 PROTAC IRAK4 degrader-7PROTAC IRAK4 degrader-7
产品简介:protac irak4 degrader-7 (compound i-417) is an orally administered agent with antitumor properties, functioning as a protac irak4 degrader [1]...产品型号:T74411 原产地:中国大陆价格: ¥0.0