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产品名称: BI 2536化合物BI 25364-[[(7R)-8-环戊基-7-乙基-5,6,7,8-四氢-5-甲基-6-氧代-2-喋啶基]氨基]-3-甲氧基-N-(1-甲基-4-哌啶基)苯甲酰胺
产品简介:bi2536 is an effective plk1 inhibitor (ic50: 0.83 nm). it has 4- and 11-fold greater selectivity than plk2 and plk3...产品型号:T6173 原产地:中国大陆价格: ¥0.0
产品名称: CDK4/6-IN-7;化合物 CDK4/6-IN-7CDK4/6-IN-7
产品简介:cdk4/6-in-7, a highly potent and selective orally active inhibitor of cdk4/6, demonstrates impressive inhibition activity with ic50 values of 1.58 nm and 4.09 n..产品型号:T61738 原产地:中国大陆价格: ¥0.0
产品名称: 5-HT7 receptor ligand 1;化合物 5-HT7 receptor ligand 15-HT7 receptor ligand 1
产品简介:5-ht7 receptor ligand 1 (compound 5c) is a potent ligand for the 5-ht7 receptor, with a k i value of 8 nm. the compound demonstrates non-hepatotoxic properties ..产品型号:T61515 原产地:中国大陆价格: ¥0.0
产品名称: FGFR-IN-7;化合物 FGFR-IN-7FGFR-IN-7
产品简介:fgfr-in-7 (compound 17) is an orally active, potent fgfr modulator with the ability to penetrate the blood-brain barrier. it exhibits neuroprotective properties..产品型号:T61528 原产地:中国大陆价格: ¥0.0
产品名称: ATG7-IN-2;化合物 ATG7-IN-2ATG7-IN-2
产品简介:atg7-in-2 (compound 1) is a highly potent inhibitor of the atg7 protein, displaying an ic 50 value of 0.089 μm. this compound effectively suppresses the activit..产品型号:T61547 原产地:中国大陆价格: ¥0.0
产品名称: ATG7-IN-3;化合物 ATG7-IN-3ATG7-IN-3
产品简介:atg7-in-3 (compound 18) is an effective inhibitor of atg7, with a potency of 0.048 μm as determined by its ic50 value. it exhibits inhibitory actions on autopha..产品型号:T61552 原产地:中国大陆价格: ¥0.0
产品名称: P2X7 receptor antagonist-2;化合物 P2X7 receptor antagonist-2P2X7 receptor antagonist-2
产品简介:p2x7 receptor antagonist-2 is a highly potent antagonist of the p2x7 receptor, exhibiting a pic50 value range of 6.5-7.5. its efficacy in combating neuroinflamm..产品型号:T61566 原产地:中国大陆价格: ¥0.0
产品名称: AKT-IN-7;化合物 AKT-IN-7AKT-IN-7
产品简介:akt-in-7 (compound 1-p1) is a potent inhibitor of akt. akt-in-7 has potential for cancer research...产品型号:T62807 原产地:中国大陆价格: ¥0.0
产品名称: NLRP3-IN-7;化合物 NLRP3-IN-7NLRP3-IN-7
产品简介:nlrp3-in-7 (compound 36) is a selective inhibitor of the nlrp3 inflammasome and is able to assemble the nlrp3 inflammasome...产品型号:T62809 原产地:中国大陆价格: ¥0.0
产品名称: FXIa-IN-7;化合物 FXIa-IN-7FXIa-IN-7
产品简介:fxia-in-7 is an orally active, selective factor xia inhibitor (ic50: 0.4 nm)...产品型号:T62832 原产地:中国大陆价格: ¥0.0
产品名称: CDK7-IN-16;化合物 CDK7-IN-16CDK7-IN-16
产品简介:cdk7-in-16 (compound 9) is a potent inhibitor of cdk 7 (ic50: 1-10 nm). cdk7-in-16 can be used in research against cancer, particularly cancers with transcripti..产品型号:T62791 原产地:中国大陆价格: ¥0.0
产品名称: Rel-5-(4-Chloro-2-fluorophenyl)-2,3-dimethyl-7-[(2R,4S)-tetrahydro-2-(1-methyl-1H-pyrazol-4-yl)-2H-p
产品简介:rel-5-(4-chloro-2-fluorophenyl)-2,3-dimethyl-7-[(2r,4s)-tetrahydro-2-(1-methyl-1h-pyrazol-4-yl)-2h-pyran-4-yl]pyrido[3,4-b]pyrazine has an ec50 value of ≤ 0.05 ..产品型号:T62750L 原产地:中国大陆价格: ¥0.0
产品名称: CDK7-IN-13;化合物 CDK7-IN-13CDK7-IN-13
产品简介:cdk7-in-13 is a pyrimidine-derived compound that is a potent inhibitor of cdk7. cdk7-in-13 has the potential to be investigated in a variety of cancers (particu..产品型号:T62759 原产地:中国大陆价格: ¥0.0
产品名称: Microtubule inhibitor 7;化合物 Microtubule inhibitor 7Microtubule inhibitor 7
产品简介:compounds 17o (ic50= 14.0 nm, nci-h460) and 17p (ic50= 2.9 nm, nci-h460) with furan moieties show potent nanomolar levels of cytotoxic activity against various ..产品型号:T62639 原产地:中国大陆价格: ¥0.0
产品名称: Carbonic anhydrase inhibitor 7;化合物 Carbonic anhydrase inhibitor 7Carbonic anhydrase inhibitor 7
产品简介:carbonic anhydrase inhibitor 7 is a potent inhibitor of human carbonic anhydrase (hca), acting on hca ix (ki: 6.5 nm), hca ii (ki: 7.1 nm), hca xii (ki: 72.1 nm..产品型号:T62666 原产地:中国大陆价格: ¥0.0
产品名称: GSK-3β inhibitor 7;化合物 GSK-3β inhibitor 7GSK-3β inhibitor 7
产品简介:gsk-3β inhibitor 7 is a gsk-3β inhibitor (ic50: 5.25 μm). gsk-3β inhibitor 7 acts by inserting into the atp-binding binding pocket of gsk-3β and forming hydroge..产品型号:T63866 原产地:中国大陆价格: ¥0.0
产品名称: Benzo[b]thiophene-7-propanoic acid, α-methoxy-4-[2-(5-methyl-2-phenyl-4-oxazolyl)ethoxy]-, (αR)-;化合物
产品简介:benzo[b]thiophene-7-propanoic acid, α-methoxy-4-[2-(5-methyl-2-phenyl-4-oxazolyl)ethoxy]-, (αr)- is a dual pparα/γ agonist with ec50 of 0.358μm and 1.21μm. benz..产品型号:T63898 原产地:中国大陆价格: ¥0.0
产品名称: Antiviral agent 7;化合物 Antiviral agent 7Antiviral agent 7
产品简介:antiviral agent 7 is a peptide-based coating that kills viruses...产品型号:T63921 原产地:中国大陆价格: ¥0.0
产品名称: Tubulin polymerization-IN-7;化合物 Tubulin polymerization-IN-7Tubulin polymerization-IN-7
产品简介:tubulin aggregation-in-7 is a potent tubulin aggregation inhibitor that has shown research potential for cancer diseases...产品型号:T63836 原产地:中国大陆价格: ¥0.0
产品名称: HER2-IN-7;化合物 HER2-IN-7HER2-IN-7
产品简介:her2-in-7 is a potent inhibitor of her2. her2-in-7 has shown potential for the study of diseases associated with erbbs, particularly her2, including cancer...产品型号:T64003 原产地:中国大陆价格: ¥0.0