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产品名称: Dorsomorphin dihydrochloride6-[4-[2-(1-哌啶基)乙氧基]苯基]-3-(4-吡啶基)吡唑并[1,5-A]嘧啶;Dorsomorphin (Compound C) 2
产品简介:dorsomorphin is a potent, selective and atp-competitive ampk inhibitor (ki: 109 nm) and does not exhibit significant activity on structurally related kinases...产品型号:T6146 原产地:中国大陆价格: ¥0.0
产品名称: CB1-IN-11-(2,4-二氯苯基)-N-1-哌啶基-4-[[(1-吡咯烷基磺酰基)氨基]甲基]-5-[5-[2-[4-(三氟甲基)苯基]乙炔基]-2-噻吩基]-1H-吡唑-3-甲酰胺;DBPR2
产品简介:cb1-in-1 is a peripherally restricted cb1r antagonist, for cb1r and cb2r with ki of 0.3 nm and 21 nm,respectively...产品型号:T5996 原产地:中国大陆价格: ¥0.0
产品名称: Sulfaphenazole磺胺苯吡唑;Raziosulfa;Depotsulfonamide;Depocid;Plisulfan
产品简介:sulfaphenazole is an inhibitor of cyp2c9 (ki: 0.3 μm) that demonstrates at least 100-fold selectivity over other cyp450 isoforms (ki: 63/29 μm for cyp2c8/cyp2c1..产品型号:T4567 原产地:中国大陆价格: ¥0.0
产品名称: 1H-pyrazole1,2-Diazole;Pyrazole;吡唑
产品简介:1h-pyrazole, is a versatile building block, with a vast applications in organic synthesis. the derivatives of pyrazole are used in medicine, for their analgesic..产品型号:T4842 原产地:中国大陆价格: ¥0.0
产品名称: S1RA hydrochlorideE-52862 hydrochloride;4-[2-[[5-甲基-1-(2-萘基)-1H-吡唑-3-基]氧基]乙基]吗啉盐酸盐(1:1)
产品简介:s1ra hcl (e-52862 hcl) is an effective and specific sigma-1 receptor(σ1r, ki: 17 nm) antagonist, and has good selectivity against σ2r (ki > 1000 nm)...产品型号:T4229 原产地:中国大陆价格: ¥0.0
产品名称: Prexasertib5-[[5-[2-(3-氨基丙氧基)-6-甲氧基苯基]-1H-吡唑-3-基]氨基]-2-吡嗪甲腈;LY2606368
产品简介:prexasertib is an inhibitor of checkpoint kinase 1 (chk1) with potential antineoplastic activity...产品型号:T4310 原产地:中国大陆价格: ¥0.0
产品名称: BUR11-{1-苯基-1H-吡唑并[3,4-D]嘧啶-4-基}哌啶;BMP upregulator 1;BUR-1;BUR 1;BMP upregulator-1
产品简介:bur1 is a saccharomyces cerevisiae cyclin-dependent kinase (cdk) and is homologous to mammalian cdk9, which functions in transcriptional elongation...产品型号:T23840 原产地:中国大陆价格: ¥0.0
产品名称: SC-581251-[(4-甲基磺酰基)苯基]-3-三氟甲基-5-(4-氟苯基)吡唑;SC 58125
产品简介:sc-58125 is a selective cyclooxygenase 2 (cox-2) inhibitor, with an ic50 of 0.04 μm. sc-58125 exhibits antitumor activity in vitro and in vivo, and it also can ..产品型号:T23333 原产地:中国大陆价格: ¥0.0
产品名称: SCH4424162-(2-呋喃基)-7-[3-(4-甲氧苯基)丙基]-7H-吡唑并[4,3-E][1,2,4]三唑并[1,5-C]嘧啶-5-胺;SCH 442416
产品简介:sch-442416 is an selective antagonist of adenosine a2a receptor. sch-442416 binds to human and rat a2a receptors with high affinity (ki values are 0.048 and 0.5..产品型号:T23336 原产地:中国大陆价格: ¥0.0
产品名称: INCB0323044-(1H-吡唑-4-基)-7-((2-(三甲基硅烷基)乙氧基)-甲基)-7H-吡咯并[2,3-D]嘧啶;4-(1H-Pyrazol-4-yl)-7-((2-(trimethyls
产品简介:detail unknown...产品型号:T2476 原产地:中国大陆价格: ¥0.0
产品名称: AM2811-(2,4-二氯苯基)-5-(4-碘苯基)-4-甲基-N-4-吗啉基-1H-吡唑-3-甲酰胺
产品简介:am 281, a cannabinoid antagonist, reduces neurologic dysfunction and mortality rate after cecal ligation and puncture in rats...产品型号:T2264 原产地:中国大陆价格: ¥0.0
产品名称: JNJ-10198409JNJ-?10198409;3-氟-N-(6,7-二甲氧基-2,4-二氢茚并[1,2-C〕吡唑-3-基苯基胺
产品简介:jnj- 10198409 is a relatively selective and atp competitive pdgf-rtk inhibitor (ic50=2 nm). jnj-10198409 has good activity against pdgfr-β kinase (ic50=4.2 nm) ..产品型号:T15616 原产地:中国大陆价格: ¥0.0
产品名称: Udenafil3-(6,7-二氢-1-甲基-7-氧代-3-丙基-1H-吡唑并[4,3-D]嘧啶-5-基)-N-[2-(1-甲基-2-吡咯烷基)乙基]-4-丙氧基苯磺酰胺;乌地那非
产品简介:udenafil is an inhibitor of pde5 ...产品型号:T17199 原产地:中国大陆价格: ¥0.0
产品名称: c-Met inhibitor 13-[(2-甲基-2H-吲唑-5-基)硫基]-6-(1-甲基-1H-吡唑-4-基)-1,2,4-三唑并[4,3-B]哒嗪
产品简介:c-met inhibitor 1 is a c-met receptor signaling pathway inhibitor, used for the treatment of cancer including glioblastoma, gastric, and pancreatic cancer...产品型号:T10655 原产地:中国大陆价格: ¥0.0
产品名称: Fomepizole4-Methylpyrazole;Antizol;Antizol-Vet;4-甲基吡唑;甲吡唑
产品简介:fomepizole is used as an antidote in confirmed or suspected methanol or ethylene glycol poisoning. fomepizole is a competitive inhibitor of alcohol dehydrogenas..产品型号:T0765 原产地:中国大陆价格: ¥0.0
产品名称: NVP-BSK805化合物NVP-BSK805NVP-BSK805 2HCl|||8-[3,5-二氟-4-(4-吗啉基甲基)苯基]-2-[1-(4-哌啶基)-1H-吡唑-4-基]喹喔啉|||BSK 8
产品简介:nvp-bsk805 (bsk 805) is an atp-competitive jak2 inhibitor...产品型号:T5049 原产地:中国大陆价格: ¥0.0
产品名称: 1-Methyl-1H-pyrazol-3-amine;N-甲基-3-氨基吡唑1-Methyl-1H-pyrazol-3-amine
产品简介:1-methyl-1h-pyrazol-3-amine is a pyrazole compound. it has been used in the synthesis of various compounds such as drugs, dyes and polymers. it is also an impor..产品型号:T3295 原产地:中国大陆价格: ¥0.0
产品名称: Prexasertib;化合物PrexasertibLY2606368;5-[[5-[2-(3-氨基丙氧基)-6-甲氧基苯基]-1H-吡唑-3-基]氨基]-2-吡嗪甲腈|||LY2606368
产品简介:prexasertib (ly2606368) is an inhibitor of checkpoint kinase 1 (chk1) with potential antineoplastic activity...产品型号:T4310 原产地:中国大陆价格: ¥0.0
产品名称: S1RA hydrochloride;化合物S1RA hydrochlorideE-52862 hydrochloride;4-[2-[[5-甲基-1-(2-萘基)-1H-吡唑-3-基]氧基]乙基]吗
产品简介:s1ra hydrochloride (e-52862 hydrochloride) is an effective and specific sigma-1 receptor(σ1r, ki: 17 nm) antagonist, and has good selectivity against σ2r (ki > ..产品型号:T4229 原产地:中国大陆价格: ¥0.0
产品名称: Sulfaphenazole磺胺苯吡唑Plisulfan|||Raziosulfa|||Depocid|||磺胺苯吡唑|||Depotsulfonamide
产品简介:sulfaphenazole (plisulfan) is an inhibitor of cyp2c9 (ki: 0.3 μm) that demonstrates at least 100-fold selectivity over other cyp450 isoforms (ki: 63/29 μm for c..产品型号:T4567 原产地:中国大陆价格: ¥0.0