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产品名称: CGP 57380;化合物CGP 57380MNK1 Inhibitor;N3-(4-氟苯基)-1H-吡唑并[3,4-D]嘧啶-3,4-二胺|||MNK1 Inhibitor
产品简介:cgp 57380 (mnk1 inhibitor) is a potent mnk1 inhibitor with ic50 of 2.2 μm, exhibiting no inhibitory activity on p38, jnk1, erk1 and -2, pkc, or c-src-like kinas..产品型号:T6440 原产地:中国大陆价格: ¥0.0
产品名称: WAY-600;化合物WAY600WAY600;6-(1H-吲哚-5-基)-4-(4-吗啉基)-1-[1-(3-吡啶基甲基)-4-哌啶基]-1H-吡唑并[3,4-D]嘧啶|||WAY600
产品简介:way-600 is a potent, atp-competitive and selective inhibitor of mtor with ic50 of 9 nm; blocks mtorc1/p-s6k(t389) and mtorc2/p-akt(s473) but not p-akt(t308); se..产品型号:T6730 原产地:中国大陆价格: ¥0.0
产品名称: WYE-687化合物WYE687N-[4-[4-(4-吗啉基)-1-[1-(3-吡啶甲基)-4-哌啶基]-1H-吡唑并[3,4-D]嘧啶-6-基]苯基]氨基甲酸甲酯
产品简介:wye-687 is an atp-competitive and selective inhibitor of mtor with ic50 of 7 nm; blocks mtorc1/ps6k(t389) and mtorc2/p-akt(s473) but no effect observed on p-akt..产品型号:T6732 原产地:中国大陆价格: ¥0.0
产品名称: WYE-354化合物WYE3544-[6-[4-[(甲氧羰基)氨基]苯基]-4-(4-吗啉基)-1H-吡唑并[3,4-D]嘧啶-1-基]-1-哌啶羧酸甲酯
产品简介:wye-354(ic50=5 nm) is an effective, selective and atp-competitive mtor inhibitor. it blocks mtorc2/p-akt(s473) and mtorc1/p-s6k(t389), not p-akt(t308). the sele..产品型号:T6731 原产地:中国大陆价格: ¥0.0
产品名称: Nelociguat;化合物NelociguatBAY60-4552;N-[4,6-二氨基-2-[1-[(2-氟苯基)甲基]-1H-吡唑并[3,4-B]吡啶-3-基]-5-嘧啶]-氨基甲酸甲酯|||B
产品简介:nelociguat (bay60-4552)(bay60-4552) is a soluble guanylate cyclase stimulator (sgc stimulator). soluble guanylate cyclase (sgc) is a key enzyme in the nitric ox..产品型号:T7201 原产地:中国大陆价格: ¥0.0
产品名称: SD 0006;化合物SD 0006SD-06;SD-06|||3-[N-(2-羟基乙酰基)-4-哌啶基]-4-(4-嘧啶基)-5-(4-氯苯基)吡唑
产品简介:sd 0006 (sd-06) is a mapk p38 alpha inhibitor( ic50 : 110 nm) for the treatment of arthritis...产品型号:T7276 原产地:中国大陆价格: ¥0.0
产品名称: Nelotanserin;化合物NelotanserinAPD125;1-[3-(4-溴-1-甲基-1H-吡唑-5-基)-4-甲氧基苯基]-3-(2,4-二氟苯基)脲|||APD125
产品简介:nelotanserin (apd125) is a potent 5-ht2a inverse agonist(ic50 : 1.7 nm), a moderately potent 5-ht2c partial inverse agonist t(ic50 :79 nm )and a weak 5-ht2b inv..产品型号:T7350 原产地:中国大陆价格: ¥0.0
产品名称: 4-(3-Methyl-5-oxo-2-pyrazolin-1-yl)benzoic acid;1-(4-羧基苯基)-3-甲基-5-吡唑酮4-(3-Methyl-5-oxo-2-pyrazolin-1
产品简介:4-(3-methyl-5-oxo-2-pyrazolin-1-yl)benzoic acid exhibits hypoglycemic activity and operates through a mechanism dependent on the response to oral glucose overlo..产品型号:T40694 原产地:中国大陆价格: ¥0.0
产品名称: 1,3-Dimethylpyrazole;1,3-二甲基吡唑1,3-Dimethyl-1H-pyrazole|||2,5-Dimethylpyrazole;1,3-Dimethyl-1H-pyrazo
产品简介:1,3-dimethylpyrazole (2,5-dimethylpyrazole) is a bioactive compound isolated from moso bamboo root...产品型号:T40807 原产地:中国大陆价格: ¥0.0
产品名称: 1H-pyrazole;吡唑1,2-Diazole|||Pyrazole;1,2-Diazole|||Pyrazole|||吡唑
产品简介:1h-pyrazole (1,2-diazole), is a versatile building block, with a vast applications in organic synthesis. the derivatives of pyrazole are used in medicine, for t..产品型号:T4842 原产地:中国大陆价格: ¥0.0
产品名称: Allopurinol Sodium;1H-吡唑并[3,4-D]嘧啶-4-醇单钠盐Allopurinol sodium salt|||Sodium allopurinol;1H-吡唑并[3,4-D]嘧
产品简介:allopurinol sodium is a xanthine oxidase inhibitor with an ic50 of 7.82±0.12 μm...产品型号:T6376 原产地:中国大陆价格: ¥0.0